ECSP034653A - Inhibidores de girasa y usos del mismo - Google Patents

Inhibidores de girasa y usos del mismo

Info

Publication number
ECSP034653A
ECSP034653A EC2003004653A ECSP034653A ECSP034653A EC SP034653 A ECSP034653 A EC SP034653A EC 2003004653 A EC2003004653 A EC 2003004653A EC SP034653 A ECSP034653 A EC SP034653A EC SP034653 A ECSP034653 A EC SP034653A
Authority
EC
Ecuador
Prior art keywords
inhibitors
relates
girasa
same
compounds
Prior art date
Application number
EC2003004653A
Other languages
English (en)
Inventor
Anne-Laure Grillot
Paul Charifson
Yusheng Liao
Michael Badia
Martin Trudeau
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of ECSP034653A publication Critical patent/ECSP034653A/es

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Esta invención se refiere a compuestos de la formula I o un derivado farmacéuticamente aceptable o prodroga del mismo. Los compuestos son útiles como inhibidores de actividad de girasas bacterianas. La presente invención también se refiere a métodos de tratamiento de infecciones bacterianas en mamíferos. La presente invención también se refiere a métodos por decrecimiento de cantidad bacteriana en una muestra biológica.
EC2003004653A 2000-12-15 2003-06-12 Inhibidores de girasa y usos del mismo ECSP034653A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25609400P 2000-12-15 2000-12-15

Publications (1)

Publication Number Publication Date
ECSP034653A true ECSP034653A (es) 2003-07-25

Family

ID=33449456

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2003004653A ECSP034653A (es) 2000-12-15 2003-06-12 Inhibidores de girasa y usos del mismo

Country Status (2)

Country Link
EC (1) ECSP034653A (es)
ZA (1) ZA200303933B (es)

Also Published As

Publication number Publication date
ZA200303933B (en) 2004-05-21

Similar Documents

Publication Publication Date Title
BR0116216A (pt) Inibidores de girase e seus usos
PL374191A1 (en) 2-ureido-6-heteroaryl-3h-benzoimidazole-4-carboxylic acid derivatives and related compounds as gyrase and/or topoisomerase iv inhibitors for the treatment of bacterial infections
MXPA05008126A (es) Inhibidores de girasa y uso de los mismos.
UY29458A1 (es) Heterociclos sustituidos y usos de los mismos
ECSP003699A (es) Inhibidores de fab i
ATE433980T1 (de) Gyraseinhibitoren und deren verwendungen
CR6577A (es) Inhibidores triciclicos de poli(adp-ribosa) polimerasas
TR200201505T2 (tr) Terapötik maddeler olarak pirazolopirimidinler
ECSP055640A (es) Composiciones de pirazol útiles como inhibidores de gsk-3
ATE370139T1 (de) Pyrazolopyridin derivate als tgf beta hemmstoffe zur behandlung von krebs
EA200802213A1 (ru) Способы лечения заболеваний крови
CY1107747T1 (el) Υποκατεστημενα τετρακυκλικα παραγωγα πυρρολοκινολονης χρησιμα ως αναστολεις της φωσφοδιεστερασης
ATE307810T1 (de) Imidazol-2-carbonsäureamid derivate als raf- kinase-inhibitoren
DE602004020070D1 (de) Thienopyrimidin-derivate als kaliumkanal-inhibitoren
ATE433963T1 (de) Fab-i inhibitoren
BRPI0519267A2 (pt) derivado de quinolina, seu uso, produÇço e medicamento contendo o mesmo
ATE509018T1 (de) Als antimikrobielle mittel geeignete bisindolpyrrole
UY30014A1 (es) Subgrupo de compuestos basados en oxabispidina comprendiendo un grupo alquilo amidasustituido, proceso de preparación, composiciones farmacéuticas conteniéndolos y aplicaciones
AR064152A1 (es) Derivados de quinolina antibacterianos,composiciones farmaceuticas que los contienen y metodo de preparacion.
ATE335739T1 (de) Cak inhibitoren und deren verwendungen
UY29012A1 (es) "oxazolididonas y composiciones y metodos relacionados"
SE0004101D0 (sv) New use
ES2182035T3 (es) Derivados del bisarilciclobuteno como inhibidores de ciclooxigenasa.
ATE419242T1 (de) Pyrrolidinylharnstoffderivate als angiogeneseinhibitoren
ECSP034653A (es) Inhibidores de girasa y usos del mismo