EA202092184A2 - Антагонисты рецептора нейрокинина-3 для терапевтического или косметологического лечения излишних жировых отложений на теле - Google Patents
Антагонисты рецептора нейрокинина-3 для терапевтического или косметологического лечения излишних жировых отложений на телеInfo
- Publication number
- EA202092184A2 EA202092184A2 EA202092184A EA202092184A EA202092184A2 EA 202092184 A2 EA202092184 A2 EA 202092184A2 EA 202092184 A EA202092184 A EA 202092184A EA 202092184 A EA202092184 A EA 202092184A EA 202092184 A2 EA202092184 A2 EA 202092184A2
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- neurokinin
- receptor
- antagonists
- therapeutic
- body fat
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Child & Adolescent Psychology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Настоящее изобретение относится к применению антагонистов рецептора нейрокинина-3 (NK3R) для терапевтического лечения патологических излишних жировых отложений на теле и/или предотвращения прибавления жировых отложений на теле у пациентов. Также настоящее изобретение относится к косметологическому способу для стимулирования потери избытка жировых отложений на теле, согласно которому вводят антагонист рецептора NK-3.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP15193513 | 2015-11-06 |
Publications (2)
Publication Number | Publication Date |
---|---|
EA202092184A2 true EA202092184A2 (ru) | 2021-03-31 |
EA202092184A3 EA202092184A3 (ru) | 2021-06-30 |
Family
ID=75262255
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202092184A EA202092184A3 (ru) | 2015-11-06 | 2016-03-16 | Антагонисты рецептора нейрокинина-3 для терапевтического или косметологического лечения излишних жировых отложений на теле |
Country Status (1)
Country | Link |
---|---|
EA (1) | EA202092184A3 (ru) |
-
2016
- 2016-03-16 EA EA202092184A patent/EA202092184A3/ru unknown
Also Published As
Publication number | Publication date |
---|---|
EA202092184A3 (ru) | 2021-06-30 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201791901A1 (ru) | Антагонисты рецептора нейрокинина-3 для терапевтического или косметологического лечения излишних жировых отложений на теле | |
EA202091134A1 (ru) | Экзосомы для иммуноонкологической и противовоспалительной терапии | |
PH12019501339A1 (en) | Amino acid compositions and methods for the treatment of muscle diseases and disorders | |
PT3377637T (pt) | Composições para uso em métodos para o tratamento de ferimentos, transtornos e doenças da pele | |
EA201792304A1 (ru) | Комбинированная терапия для лечения рака | |
IL276383B1 (en) | Treatment of ophthalmological diseases | |
EA201691567A1 (ru) | Способы лечения легких травм головного мозга | |
IL264069A (en) | Trpa1 antagonists for treatment of dry eye, ocular pain and inflammation | |
EA201891609A1 (ru) | Производные 3-((гетеро-)арил)алкил-8-амино-2-оксо-1,3-диазаспиро[4.5]декана | |
EA201792571A1 (ru) | Терапевтическое применение l-4-хлорокинуренина | |
EA202190281A1 (ru) | Производные 3-((гетеро-)арил)-8-амино-2-оксо-1,3-диаза-спиро[4,5]декана | |
MX2018000262A (es) | Usos terapeuticos de formulaciones de berberina. | |
ZA202002075B (en) | Compounds, compositions and methods for treatment of eye disorders and skin diseases | |
EA202091307A1 (ru) | Накожная система мониторинга состояния человека | |
EA201792560A1 (ru) | Наночастицы для применения в качестве терапевтической вакцины | |
EA201792445A1 (ru) | Новые амидогетероарилароилгидразидэтины | |
EA202090266A1 (ru) | Ингибиторы mpo для применения в медицине | |
MX2019000600A (es) | Agente estimulador del receptor 5-hidroxitriptamina 1b para reparación de piel y/o cabello. | |
SG11202007082PA (en) | Composition used for therapeutic treatment of skin disease | |
EA202092184A2 (ru) | Антагонисты рецептора нейрокинина-3 для терапевтического или косметологического лечения излишних жировых отложений на теле | |
PT3271015T (pt) | Antagonistas do recetor nk-3 para tratamento terapêutico ou cosmético do excesso de gordura corporal | |
IL274132A (en) | Treatment of skin problems | |
GB201904012D0 (en) | Regulation of blood glucoe via human microbioma | |
IT201700070978A1 (it) | Apparecchiatura per il trattamento terapeutico del corpo umano | |
EA201991866A1 (ru) | Комбинированная терапия |