EA201992839A1 - Кристаллические формы селеталисиба - Google Patents
Кристаллические формы селеталисибаInfo
- Publication number
- EA201992839A1 EA201992839A1 EA201992839A EA201992839A EA201992839A1 EA 201992839 A1 EA201992839 A1 EA 201992839A1 EA 201992839 A EA201992839 A EA 201992839A EA 201992839 A EA201992839 A EA 201992839A EA 201992839 A1 EA201992839 A1 EA 201992839A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- celetalisib
- crystal forms
- pathological conditions
- isophome
- seletalisib
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Transplantation (AREA)
- Ophthalmology & Optometry (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
В заявке описаны кристаллические формы селеталисиба, обозначенные как форма В и форма F и охарактеризованные в настоящем изобретении, которые являются селективными ингибиторами ферментов киназы PI3, в частности изофомы PI3K человека, и поэтому полезны для применения в медицине, например, для лечения воспалительных, аутоиммунных, сердечно-сосудистых, нейродегенеративных, метаболических, онкологических, ноцицептивных патологических состояний или патологических состояний глаз.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB1708856.8A GB201708856D0 (en) | 2017-06-02 | 2017-06-02 | Seletalisib crystalline forms |
PCT/EP2018/063640 WO2018219772A1 (en) | 2017-06-02 | 2018-05-24 | Crystalline forms of seletalisib |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201992839A1 true EA201992839A1 (ru) | 2020-04-08 |
Family
ID=59349914
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201992839A EA201992839A1 (ru) | 2017-06-02 | 2018-05-24 | Кристаллические формы селеталисиба |
Country Status (17)
Country | Link |
---|---|
US (1) | US11059820B2 (ru) |
EP (1) | EP3630760A1 (ru) |
JP (1) | JP7264829B2 (ru) |
KR (1) | KR102591329B1 (ru) |
CN (2) | CN110709399A (ru) |
AR (1) | AR112062A1 (ru) |
AU (1) | AU2018276243B2 (ru) |
BR (1) | BR112019023592A8 (ru) |
CA (1) | CA3062533A1 (ru) |
CL (1) | CL2019003510A1 (ru) |
CO (1) | CO2019014026A2 (ru) |
EA (1) | EA201992839A1 (ru) |
GB (1) | GB201708856D0 (ru) |
IL (1) | IL270937A (ru) |
MX (1) | MX2019013518A (ru) |
RU (1) | RU2019143761A (ru) |
WO (1) | WO2018219772A1 (ru) |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5620981A (en) * | 1995-05-03 | 1997-04-15 | Warner-Lambert Company | Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation |
US20040106794A1 (en) * | 2001-04-16 | 2004-06-03 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
GB0428475D0 (en) * | 2004-12-30 | 2005-02-02 | 4 Aza Bioscience Nv | Pyrido(3,2-D)pyrimidine derivatives and pharmaceutical compositions useful as medicines for the treatment of autoimmune disorders |
AR082799A1 (es) * | 2010-09-08 | 2013-01-09 | Ucb Pharma Sa | Derivados de quinolina y quinoxalina como inhibidores de quinasa |
KR20170010369A (ko) * | 2014-05-27 | 2017-01-31 | 알미랄, 에스.에이. | 병용물 |
GB201506786D0 (en) | 2015-04-21 | 2015-06-03 | Ucb Biopharma Sprl | Therapeutic use |
GB201608797D0 (en) | 2016-05-19 | 2016-07-06 | Ucb Biopharma Sprl | Therapeutic use |
-
2017
- 2017-06-02 GB GBGB1708856.8A patent/GB201708856D0/en not_active Ceased
-
2018
- 2018-05-24 WO PCT/EP2018/063640 patent/WO2018219772A1/en active Application Filing
- 2018-05-24 EA EA201992839A patent/EA201992839A1/ru unknown
- 2018-05-24 MX MX2019013518A patent/MX2019013518A/es unknown
- 2018-05-24 RU RU2019143761A patent/RU2019143761A/ru unknown
- 2018-05-24 CA CA3062533A patent/CA3062533A1/en active Pending
- 2018-05-24 KR KR1020197037460A patent/KR102591329B1/ko active IP Right Grant
- 2018-05-24 CN CN201880036440.9A patent/CN110709399A/zh active Pending
- 2018-05-24 CN CN202210296993.6A patent/CN114573580A/zh active Pending
- 2018-05-24 JP JP2019566167A patent/JP7264829B2/ja active Active
- 2018-05-24 AU AU2018276243A patent/AU2018276243B2/en active Active
- 2018-05-24 EP EP18728337.9A patent/EP3630760A1/en active Pending
- 2018-05-24 US US16/615,992 patent/US11059820B2/en active Active
- 2018-05-24 BR BR112019023592A patent/BR112019023592A8/pt unknown
- 2018-06-01 AR ARP180101467A patent/AR112062A1/es unknown
-
2019
- 2019-11-26 IL IL270937A patent/IL270937A/en unknown
- 2019-11-29 CL CL2019003510A patent/CL2019003510A1/es unknown
- 2019-12-12 CO CONC2019/0014026A patent/CO2019014026A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
US11059820B2 (en) | 2021-07-13 |
KR102591329B1 (ko) | 2023-10-18 |
CA3062533A1 (en) | 2018-12-06 |
IL270937A (en) | 2020-01-30 |
CN110709399A (zh) | 2020-01-17 |
CN114573580A (zh) | 2022-06-03 |
BR112019023592A8 (pt) | 2023-05-09 |
KR20200012902A (ko) | 2020-02-05 |
MX2019013518A (es) | 2020-02-10 |
US20200095246A1 (en) | 2020-03-26 |
WO2018219772A1 (en) | 2018-12-06 |
AU2018276243B2 (en) | 2021-11-25 |
JP7264829B2 (ja) | 2023-04-25 |
AR112062A1 (es) | 2019-09-18 |
CL2019003510A1 (es) | 2020-04-17 |
CO2019014026A2 (es) | 2020-01-17 |
JP2020521793A (ja) | 2020-07-27 |
EP3630760A1 (en) | 2020-04-08 |
AU2018276243A1 (en) | 2019-12-19 |
BR112019023592A2 (pt) | 2020-05-26 |
RU2019143761A (ru) | 2021-07-09 |
GB201708856D0 (en) | 2017-07-19 |
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