EA201270786A1 - α-КРИСТАЛЛИЧЕСКАЯ ФОРМА КАРБАБЕНЗПИРИДА - Google Patents
α-КРИСТАЛЛИЧЕСКАЯ ФОРМА КАРБАБЕНЗПИРИДАInfo
- Publication number
- EA201270786A1 EA201270786A1 EA201270786A EA201270786A EA201270786A1 EA 201270786 A1 EA201270786 A1 EA 201270786A1 EA 201270786 A EA201270786 A EA 201270786A EA 201270786 A EA201270786 A EA 201270786A EA 201270786 A1 EA201270786 A1 EA 201270786A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- carbabenzpyrid
- crystal form
- carbabenzopyrid
- relates
- crystalline form
- Prior art date
Links
- 208000036142 Viral infection Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 230000009385 viral infection Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4425—Pyridinium derivatives, e.g. pralidoxime, pyridostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Virology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyridine Compounds (AREA)
Abstract
Настоящее изобретение относится к новой кристаллической форме карбабензпирида формулы (I)и способу ее получения. Также изобретение касается применения новой кристаллической формы карбабензпирида для лечения и предупреждения вирусных инфекций.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IB2010/001956 WO2011158058A1 (en) | 2010-06-17 | 2010-06-17 | α-CRYSTALLINE FORM OF CARBABENZPYRIDE |
PCT/EP2011/059922 WO2011157743A1 (en) | 2010-06-17 | 2011-06-15 | Alpha-crystalline form of carbabenzpyride |
Publications (3)
Publication Number | Publication Date |
---|---|
EA201270786A1 true EA201270786A1 (ru) | 2013-02-28 |
EA019080B1 EA019080B1 (ru) | 2013-12-30 |
EA019080B9 EA019080B9 (ru) | 2014-03-31 |
Family
ID=43607637
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201270786A EA019080B9 (ru) | 2010-06-17 | 2011-06-15 | α-КРИСТАЛЛИЧЕСКАЯ ФОРМА КАРБАБЕНЗПИРИДА |
Country Status (7)
Country | Link |
---|---|
US (1) | US8404857B2 (ru) |
EP (1) | EP2513060B1 (ru) |
CA (1) | CA2790294C (ru) |
EA (1) | EA019080B9 (ru) |
PL (1) | PL2513060T3 (ru) |
UA (1) | UA104102C2 (ru) |
WO (2) | WO2011158058A1 (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013170901A1 (en) * | 2012-05-18 | 2013-11-21 | Farmak International Holding Gmbh | N-methyl-4-benzylcarbamidopyridinium chloride and a process for its preparation |
EA201792455A1 (ru) * | 2017-12-06 | 2019-06-28 | Открытое акционерное общество "Авексима" | Нобазит кристаллический в форме ромбической сингонии и способ его получения |
RU2689775C1 (ru) * | 2018-11-02 | 2019-05-29 | Открытое акционерное общество "Авексима" | Способ промышленного производства N-метил-4-бензилкарбамидопиридиния йодида |
-
2010
- 2010-06-17 WO PCT/IB2010/001956 patent/WO2011158058A1/en active Application Filing
-
2011
- 2011-06-15 EP EP11725450.8A patent/EP2513060B1/en active Active
- 2011-06-15 UA UAA201215039A patent/UA104102C2/ru unknown
- 2011-06-15 PL PL11725450T patent/PL2513060T3/pl unknown
- 2011-06-15 EA EA201270786A patent/EA019080B9/ru not_active IP Right Cessation
- 2011-06-15 WO PCT/EP2011/059922 patent/WO2011157743A1/en active Application Filing
- 2011-06-15 US US13/576,885 patent/US8404857B2/en active Active
- 2011-06-15 CA CA2790294A patent/CA2790294C/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EA019080B1 (ru) | 2013-12-30 |
US8404857B2 (en) | 2013-03-26 |
EP2513060B1 (en) | 2013-09-11 |
CA2790294A1 (en) | 2011-12-22 |
WO2011158058A1 (en) | 2011-12-22 |
CA2790294C (en) | 2013-05-28 |
EA019080B9 (ru) | 2014-03-31 |
EP2513060A1 (en) | 2012-10-24 |
UA104102C2 (en) | 2013-12-25 |
US20120309978A1 (en) | 2012-12-06 |
PL2513060T3 (pl) | 2014-02-28 |
WO2011157743A1 (en) | 2011-12-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201290632A1 (ru) | Производные бетулина | |
EA201301320A1 (ru) | 4-арил-n-фенил-1,3,5-триазин-2-амины, которые содержат сульфоксиминную группу | |
EA201490724A1 (ru) | Замещенные соединения тетрагидроизохинолина в качестве ингибиторов фактора xia | |
PH12015500347A1 (en) | 6-amino acid heteroaryldihydropyrimidines for the treatment and prophylaxis of hepatitis b virus infection | |
MD20140136A2 (ru) | Ингибиторы вируса гепатита С | |
EA201490474A1 (ru) | Аминохиназолины в качестве ингибиторов киназ | |
EA201390576A1 (ru) | Противовирусные соединения | |
UA111841C2 (uk) | Сполуки бензотіазолу та їх фармацевтичне застосування | |
IN2014MN02652A (ru) | ||
UA111626C2 (uk) | Похідні дигідрохінолін-2-ону | |
EA201101026A1 (ru) | Ингибиторы бета-секретазы | |
EA201591527A1 (ru) | Новые производные пиридина | |
EA201590890A1 (ru) | Производные 5-фтор-n-(пиридин-2-ил)пиридин-2-амина, содержащие сульфоксиминовую группу | |
EA201490854A1 (ru) | Противовирусные соединения | |
EA201270149A1 (ru) | Ингибиторы bace | |
EA201300604A1 (ru) | Соединения, предназначенные для лечения респираторно-синцитиальных вирусных инфекций | |
EA201590979A1 (ru) | Способы и промежуточные химические соединения для получения фармацевтических средств | |
EA201490567A1 (ru) | Новые бициклические производные дигидрохинолин-2-она | |
EA201300388A1 (ru) | Соединения замещенного бензамида | |
AU2011286276A8 (en) | Substituted Biphenylene Compounds and methods of use thereof for the treatment of viral diseases | |
EA201490650A1 (ru) | Фармацевтические композиции | |
EA201190293A1 (ru) | Пролекарства триптолида | |
EA201300034A1 (ru) | Фармацевтические композиции, содержащие иматиниб или его фармацевтически приемлемую соль, и способы их получения | |
IN2014CN04449A (ru) | ||
EA201590364A1 (ru) | Применение орвепитанта, его солей и кристаллических форм и композиций, его содержащих, для лечения зуда |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
TH4A | Publication of the corrected specification to eurasian patent | ||
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM TJ |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AZ BY KZ KG MD TM RU |