EA201170880A1 - Таблетка с контролируемым высвобождением с малой дозой активного вещества - Google Patents

Таблетка с контролируемым высвобождением с малой дозой активного вещества

Info

Publication number
EA201170880A1
EA201170880A1 EA201170880A EA201170880A EA201170880A1 EA 201170880 A1 EA201170880 A1 EA 201170880A1 EA 201170880 A EA201170880 A EA 201170880A EA 201170880 A EA201170880 A EA 201170880A EA 201170880 A1 EA201170880 A1 EA 201170880A1
Authority
EA
Eurasian Patent Office
Prior art keywords
tablet
active substance
low dose
controlled shipping
shipping
Prior art date
Application number
EA201170880A
Other languages
English (en)
Inventor
Коринде Аннемари Янсен
Дирк Памперин
Original Assignee
Синтон Б.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42099055&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201170880(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Синтон Б.В. filed Critical Синтон Б.В.
Publication of EA201170880A1 publication Critical patent/EA201170880A1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Настоящее изобретение относится к лекарственным средствам с малой дозой активного вещества, которые обладают пролонгированным действием благодаря конструкции "таблетка-в-таблетке", в соответствии с которой лекарственное средство содержится в матрице с контролируемым высвобождением, находящейся в наружном напрессованном покрывающем слое, а не во внутренней сердцевине таблетки.
EA201170880A 2008-12-24 2009-12-21 Таблетка с контролируемым высвобождением с малой дозой активного вещества EA201170880A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14071208P 2008-12-24 2008-12-24
PCT/EP2009/009206 WO2010072401A1 (en) 2008-12-24 2009-12-21 Low dose controlled release tablet

Publications (1)

Publication Number Publication Date
EA201170880A1 true EA201170880A1 (ru) 2012-02-28

Family

ID=42099055

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201170880A EA201170880A1 (ru) 2008-12-24 2009-12-21 Таблетка с контролируемым высвобождением с малой дозой активного вещества

Country Status (11)

Country Link
US (1) US8465770B2 (ru)
EP (1) EP2376066A1 (ru)
KR (1) KR20110104076A (ru)
BR (1) BRPI0922623A2 (ru)
CL (1) CL2011001554A1 (ru)
CO (1) CO6390099A2 (ru)
EA (1) EA201170880A1 (ru)
EC (1) ECSP11011188A (ru)
MX (1) MX2011006679A (ru)
WO (1) WO2010072401A1 (ru)
ZA (1) ZA201104564B (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA110933C2 (uk) * 2010-03-25 2016-03-10 Аоп Орфан Фармацойтікальс Аг Композиція для лікування есенціальної тромбоцитемії
KR20160100570A (ko) * 2015-02-16 2016-08-24 한미약품 주식회사 탐수로신 염산염 함유 서방성 과립을 포함하는 경구용 약제학적 제제
RU2018142485A (ru) * 2016-05-04 2020-06-04 Эспен Парк Фармасьютикалз, Инк. Отсроченное высвобождение тамсулозина гидрохлорида после перорального введения

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1147342A (en) * 1977-10-12 1983-05-31 Kazuo Imai Process of producing novel phenylethanolamine derivatives
JPS56110665A (en) * 1980-02-08 1981-09-01 Yamanouchi Pharmaceut Co Ltd Sulfamoyl-substituted phenetylamine derivative and its preparation
US4772475A (en) 1985-03-08 1988-09-20 Yamanouchi Pharmaceutical Co., Ltd. Controlled-release multiple units pharmaceutical formulation
JPH066565B2 (ja) 1986-07-21 1994-01-26 山之内製薬株式会社 光学活性なベンゼンスルホンアミド誘導体の製造法
FI95572C (fi) * 1987-06-22 1996-02-26 Eisai Co Ltd Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi
IE60311B1 (en) 1987-09-24 1994-06-29 American Home Prod Sustained release etodolac
RO112991B1 (ro) 1992-09-18 1998-03-30 Yamanouchi Pharma Co Ltd Preparat tip hidrogel, cu eliberare sustinuta
ES2098069T3 (es) * 1993-02-23 1997-04-16 Hoechst Ag Bencenosulfonil-ureas y -tioureas sustituidas, procedimiento para su preparacion y su utilizacion como agentes farmaceuticos.
US5877218A (en) * 1994-01-10 1999-03-02 Teva Pharmaceutical Industries, Ltd. Compositions containing and methods of using 1-aminoindan and derivatives thereof and process for preparing optically active 1-aminoindan derivatives
US6177430B1 (en) * 1997-03-27 2001-01-23 Pfizer Inc Use of α1-adrenoreceptor antagonists in the prevention and treatment of benign prostatic hyperplasia
SE9803871D0 (sv) 1998-11-11 1998-11-11 Pharmacia & Upjohn Ab Therapeutic method and formulation
US20030180352A1 (en) * 1999-11-23 2003-09-25 Patel Mahesh V. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
US6368628B1 (en) * 2000-05-26 2002-04-09 Pharma Pass Llc Sustained release pharmaceutical composition free of food effect
US6287599B1 (en) * 2000-12-20 2001-09-11 Shire Laboratories, Inc. Sustained release pharmaceutical dosage forms with minimized pH dependent dissolution profiles
US6835853B2 (en) * 2001-10-31 2004-12-28 Synthon Bv Process for resolution of tamsulosin and compounds, compositions, and processes associated therewith
PT1443917E (pt) * 2001-11-07 2006-06-30 Synthon Bv Comprimidos de tamsulosina
US7018658B2 (en) * 2002-11-14 2006-03-28 Synthon Bv Pharmaceutical pellets comprising tamsulosin
US7442387B2 (en) 2003-03-06 2008-10-28 Astellas Pharma Inc. Pharmaceutical composition for controlled release of active substances and manufacturing method thereof
US8197846B2 (en) * 2003-11-10 2012-06-12 Astellas Pharma Inc. Sustained release pharmaceutical composition
US8128958B2 (en) * 2003-11-10 2012-03-06 Astellas Pharma Inc. Sustained release pharmaceutical composition
KR20070044911A (ko) * 2005-10-26 2007-05-02 주식회사 씨티씨바이오 염산 탐스로신 함유 방출조절 제제
EP2026766A1 (en) 2006-05-17 2009-02-25 Synthon B.V. Tablet composition with a prolonged release of tamsulosin
KR100885029B1 (ko) * 2007-02-07 2009-02-23 지엘팜텍 주식회사 경구투여용 서방성 삼중정제

Also Published As

Publication number Publication date
EP2376066A1 (en) 2011-10-19
US20100092552A1 (en) 2010-04-15
WO2010072401A1 (en) 2010-07-01
US8465770B2 (en) 2013-06-18
ECSP11011188A (es) 2011-08-31
KR20110104076A (ko) 2011-09-21
CO6390099A2 (es) 2012-02-29
ZA201104564B (en) 2012-09-26
BRPI0922623A2 (pt) 2016-09-13
MX2011006679A (es) 2011-09-28
CL2011001554A1 (es) 2012-04-09

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