EA200970097A1 - Фармацевтическая композиция, содержащая бикалутамид, и способ её применения - Google Patents

Фармацевтическая композиция, содержащая бикалутамид, и способ её применения

Info

Publication number
EA200970097A1
EA200970097A1 EA200970097A EA200970097A EA200970097A1 EA 200970097 A1 EA200970097 A1 EA 200970097A1 EA 200970097 A EA200970097 A EA 200970097A EA 200970097 A EA200970097 A EA 200970097A EA 200970097 A1 EA200970097 A1 EA 200970097A1
Authority
EA
Eurasian Patent Office
Prior art keywords
application
pharmaceutical composition
composition containing
containing bicalutamide
week
Prior art date
Application number
EA200970097A
Other languages
English (en)
Inventor
Амарджит Сингх
Сарабджит Сингх
Шивананд Путхли
Original Assignee
Панацея Биотек Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Панацея Биотек Лимитед filed Critical Панацея Биотек Лимитед
Publication of EA200970097A1 publication Critical patent/EA200970097A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/095Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10Sulfides; Sulfoxides; Sulfones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28Antiandrogens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Настоящее изобретение относится к пероральному препарату, содержащему бикалутамид, для введения в режиме дозирования трижды в неделю, дважды в неделю и один раз в неделю. Данную композицию используют для достижения антиандрогенного эффекта.
EA200970097A 2006-07-07 2007-07-05 Фармацевтическая композиция, содержащая бикалутамид, и способ её применения EA200970097A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1074MU2006 2006-07-07
PCT/IN2007/000274 WO2008068770A2 (en) 2006-07-07 2007-07-05 Pharmaceutical composition containing bicalutamide and a method for its use

Publications (1)

Publication Number Publication Date
EA200970097A1 true EA200970097A1 (ru) 2009-06-30

Family

ID=39492731

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200970097A EA200970097A1 (ru) 2006-07-07 2007-07-05 Фармацевтическая композиция, содержащая бикалутамид, и способ её применения

Country Status (16)

Country Link
US (1) US20090317464A1 (ru)
EP (1) EP2046321A4 (ru)
JP (1) JP2009542627A (ru)
KR (1) KR20090057214A (ru)
CN (1) CN101478963A (ru)
AR (1) AR061853A1 (ru)
BR (1) BRPI0714053A2 (ru)
CA (1) CA2655541A1 (ru)
CO (1) CO6150137A2 (ru)
EA (1) EA200970097A1 (ru)
MA (1) MA30692B1 (ru)
MX (1) MX2009000268A (ru)
TN (1) TNSN08530A1 (ru)
UA (1) UA92233C2 (ru)
WO (1) WO2008068770A2 (ru)
ZA (1) ZA200900502B (ru)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103860487B (zh) * 2012-12-10 2016-07-06 天津市汉康医药生物技术有限公司 一种比卡鲁胺片及其制备工艺

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050008691A1 (en) * 2003-05-14 2005-01-13 Arturo Siles Ortega Bicalutamide compositions
JP2005060302A (ja) * 2003-08-12 2005-03-10 Sumitomo Chemical Co Ltd N−メタクリロイル−4−シアノ−3−トリフルオロメチルアニリンの製造方法および安定化方法
US20060269596A1 (en) * 2005-01-12 2006-11-30 Gary Liversidge Controlled release compositions comprising an acylanilide

Also Published As

Publication number Publication date
US20090317464A1 (en) 2009-12-24
AR061853A1 (es) 2008-09-24
CN101478963A (zh) 2009-07-08
TNSN08530A1 (en) 2010-04-14
EP2046321A4 (en) 2011-08-31
BRPI0714053A2 (pt) 2012-12-18
CA2655541A1 (en) 2008-06-12
KR20090057214A (ko) 2009-06-04
MA30692B1 (fr) 2009-09-01
EP2046321A2 (en) 2009-04-15
WO2008068770A2 (en) 2008-06-12
MX2009000268A (es) 2009-01-26
JP2009542627A (ja) 2009-12-03
CO6150137A2 (es) 2010-04-20
WO2008068770A3 (en) 2008-10-16
ZA200900502B (en) 2010-06-30
UA92233C2 (ru) 2010-10-11

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