EA200700600A1 - Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент - Google Patents
Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агентInfo
- Publication number
- EA200700600A1 EA200700600A1 EA200700600A EA200700600A EA200700600A1 EA 200700600 A1 EA200700600 A1 EA 200700600A1 EA 200700600 A EA200700600 A EA 200700600A EA 200700600 A EA200700600 A EA 200700600A EA 200700600 A1 EA200700600 A1 EA 200700600A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- agent
- pharmaceutical composition
- betumepholic
- composition containing
- cholinergic
- Prior art date
Links
- 239000003795 chemical substances by application Substances 0.000 title abstract 4
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940121948 Muscarinic receptor antagonist Drugs 0.000 title 1
- 239000000812 cholinergic antagonist Substances 0.000 title 1
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- NDAUXUAQIAJITI-LBPRGKRZSA-N (R)-salbutamol Chemical compound CC(C)(C)NC[C@H](O)C1=CC=C(O)C(CO)=C1 NDAUXUAQIAJITI-LBPRGKRZSA-N 0.000 abstract 1
- 230000001078 anti-cholinergic effect Effects 0.000 abstract 1
- 230000003454 betamimetic effect Effects 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229960001361 ipratropium bromide Drugs 0.000 abstract 1
- KEWHKYJURDBRMN-ZEODDXGYSA-M ipratropium bromide hydrate Chemical compound O.[Br-].O([C@H]1C[C@H]2CC[C@@H](C1)[N@@+]2(C)C(C)C)C(=O)C(CO)C1=CC=CC=C1 KEWHKYJURDBRMN-ZEODDXGYSA-M 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Фармацевтическая композиция в дозированной форме, приемлемой для ингаляции, содержащая терапевтически эффективный изомер бета-миметического агента или его соль, сольват, эфир, производное или полиморф, по существу, свободный от менее терапевтически эффективного(ых) изомера(ов) указанного агента и необязательно антихолинергический агент или его соль, сольват, эфир, производное, изомер или полиморф. Предпочтительно композиция содержит сульфат R-сальбутамола и бромид ипратропия. Также представлены способы получения композиций по изобретению.
Applications Claiming Priority (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN970MU2004 | 2004-09-09 | ||
IN1004MU2004 | 2004-09-17 | ||
IN1077MU2004 | 2004-10-08 | ||
IN1088MU2004 | 2004-10-11 | ||
IN1089MU2004 | 2004-10-11 | ||
IN93MU2005 | 2005-01-31 | ||
IN222MU2005 | 2005-02-28 | ||
PCT/GB2005/003475 WO2006027595A1 (en) | 2004-09-09 | 2005-09-09 | Pharmaceutical composition comprising an isomer of a betamimetic agent and an anti-cholinergic agent |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200700600A1 true EA200700600A1 (ru) | 2008-02-28 |
Family
ID=35311711
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200700600A EA200700600A1 (ru) | 2004-09-09 | 2005-09-09 | Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент |
Country Status (11)
Country | Link |
---|---|
US (1) | US20070264202A1 (ru) |
EP (1) | EP1791534A1 (ru) |
JP (1) | JP2008512434A (ru) |
KR (1) | KR20070102659A (ru) |
AU (1) | AU2005281511B2 (ru) |
BR (1) | BRPI0515103A (ru) |
CA (1) | CA2580019A1 (ru) |
EA (1) | EA200700600A1 (ru) |
IL (1) | IL181828A0 (ru) |
MX (1) | MX2007002899A (ru) |
WO (1) | WO2006027595A1 (ru) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0501956D0 (en) * | 2005-01-31 | 2005-03-09 | Arrow Internat | Nebulizer formulation |
CA2652699C (en) | 2006-05-19 | 2014-11-04 | Boehringer Ingelheim International Gmbh | Propellant-free inhalation aerosol formulation containing ipratropium bromide and salbutamol sulfate |
EP2026784A1 (de) * | 2006-05-19 | 2009-02-25 | Boehringer Ingelheim International GmbH | Aerosolformulierung enthaltend ipratropiumbromid und salbutamolsulfat |
US20070286814A1 (en) * | 2006-06-12 | 2007-12-13 | Medispray Laboratories Pvt. Ltd. | Stable aerosol pharmaceutical formulations |
EP2077132A1 (en) | 2008-01-02 | 2009-07-08 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dispensing device, storage device and method for dispensing a formulation |
US20110250242A1 (en) * | 2008-10-23 | 2011-10-13 | Sunovion Pharmaceuticals Inc. | Arformoterol and tiotropium compositions and methods for use |
EP2414560B1 (de) | 2009-03-31 | 2013-10-23 | Boehringer Ingelheim International GmbH | Verfahren zur beschichtung einer oberfläche eines bauteils |
JP5763053B2 (ja) | 2009-05-18 | 2015-08-12 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | アダプタ、吸入器具及びアトマイザ |
US10016568B2 (en) | 2009-11-25 | 2018-07-10 | Boehringer Ingelheim International Gmbh | Nebulizer |
WO2011064163A1 (en) | 2009-11-25 | 2011-06-03 | Boehringer Ingelheim International Gmbh | Nebulizer |
PE20130036A1 (es) | 2009-11-25 | 2013-02-03 | Boehringer Ingelheim Int | Nebulizador |
JP5874724B2 (ja) | 2010-06-24 | 2016-03-02 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ネブライザ |
WO2012130757A1 (de) | 2011-04-01 | 2012-10-04 | Boehringer Ingelheim International Gmbh | Medizinisches gerät mit behälter |
US9827384B2 (en) | 2011-05-23 | 2017-11-28 | Boehringer Ingelheim International Gmbh | Nebulizer |
WO2013152894A1 (de) | 2012-04-13 | 2013-10-17 | Boehringer Ingelheim International Gmbh | Zerstäuber mit kodiermitteln |
PL2835146T3 (pl) | 2013-08-09 | 2021-04-06 | Boehringer Ingelheim International Gmbh | Nebulizator |
JP6643231B2 (ja) | 2013-08-09 | 2020-02-12 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ネブライザ |
CN106255554B (zh) | 2014-05-07 | 2021-05-04 | 勃林格殷格翰国际有限公司 | 容器、喷雾器及用途 |
DK3139984T3 (da) | 2014-05-07 | 2021-07-19 | Boehringer Ingelheim Int | Forstøver |
ES2957901T3 (es) | 2014-05-07 | 2024-01-29 | Boehringer Ingelheim Int | Recipiente y dispositivo indicador y nebulizador |
EP3569221A1 (en) * | 2018-05-17 | 2019-11-20 | Notoxins IP B.V. | Aqueous formulations comprising ipratropium for topical treatment of hyperhidrosis |
CN113018280A (zh) * | 2021-03-01 | 2021-06-25 | 石家庄四药有限公司 | 一种异丙托溴铵吸入用溶液制剂及其制备方法 |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5192528A (en) * | 1985-05-22 | 1993-03-09 | Liposome Technology, Inc. | Corticosteroid inhalation treatment method |
US5919827A (en) * | 1990-07-11 | 1999-07-06 | Sepracor Inc. | Method for treating asthma using optically pure R(-) salmeterol |
US5795564A (en) * | 1991-04-05 | 1998-08-18 | Sepracor, Inc. | Methods and compositions for treating pulmonary disorders using optically pure (R,R)-formoterol |
US6299863B1 (en) * | 1992-04-03 | 2001-10-09 | Sepracor Inc. | Aerosol formulations containing micronized optically pure (R,R) formoterol for bronchodilating therapy |
US6423298B2 (en) * | 1998-06-18 | 2002-07-23 | Boehringer Ingelheim Pharmaceuticals, Inc. | Pharmaceutical formulations for aerosols with two or more active substances |
GB9827200D0 (en) * | 1998-12-11 | 1999-02-03 | Glaxo Group Ltd | Dry powder inhaler |
WO2001064274A2 (en) * | 2000-03-01 | 2001-09-07 | Glaxo Group Limited | Metered dose inhaler |
US20040019025A1 (en) * | 2000-04-18 | 2004-01-29 | Gavin Brian Charles | Medical compositions comprising (r,r)-formoterol and rofleponide |
GB0009607D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Medical compositions |
US20020076382A1 (en) * | 2000-08-04 | 2002-06-20 | Kaplan Leonard W. | Formulations of mometasone and a bronchodilator for pulmonary administration |
US20040050385A1 (en) * | 2000-10-20 | 2004-03-18 | Bonney Stanley George | Inhaler |
GB0030171D0 (en) * | 2000-12-11 | 2001-01-24 | Cipla Ltd | Process for preparing isomers of salbutamol |
US20020189610A1 (en) * | 2001-02-01 | 2002-12-19 | Karl-Heinz Bozung | Pharmaceutical compositions containing an ipratropium salt and a betamimetic |
GB0105560D0 (en) * | 2001-03-07 | 2001-04-25 | Glaxo Group Ltd | Pharmaceutical formulations |
US6667344B2 (en) * | 2001-04-17 | 2003-12-23 | Dey, L.P. | Bronchodilating compositions and methods |
JP2003221335A (ja) * | 2001-10-26 | 2003-08-05 | Dey Lp | 慢性閉塞性肺疾患の症状を緩和するためのアルブテロールおよびイプラトロピウム吸入溶液、システム、キットおよび方法 |
NZ541168A (en) * | 2002-12-10 | 2008-10-31 | Sepracor Inc | Levalbuterol salt |
US20040191176A1 (en) * | 2003-03-28 | 2004-09-30 | Kaplan Leonard W | Formulations for treatment of pulmonary disorders |
-
2005
- 2005-09-09 AU AU2005281511A patent/AU2005281511B2/en not_active Ceased
- 2005-09-09 BR BRPI0515103-1A patent/BRPI0515103A/pt not_active IP Right Cessation
- 2005-09-09 JP JP2007530766A patent/JP2008512434A/ja active Pending
- 2005-09-09 EP EP05786158A patent/EP1791534A1/en not_active Withdrawn
- 2005-09-09 MX MX2007002899A patent/MX2007002899A/es not_active Application Discontinuation
- 2005-09-09 WO PCT/GB2005/003475 patent/WO2006027595A1/en active Application Filing
- 2005-09-09 US US11/574,902 patent/US20070264202A1/en not_active Abandoned
- 2005-09-09 CA CA002580019A patent/CA2580019A1/en not_active Abandoned
- 2005-09-09 EA EA200700600A patent/EA200700600A1/ru unknown
- 2005-09-09 KR KR1020077008004A patent/KR20070102659A/ko not_active Application Discontinuation
-
2007
- 2007-03-08 IL IL181828A patent/IL181828A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
AU2005281511B2 (en) | 2011-03-31 |
KR20070102659A (ko) | 2007-10-19 |
MX2007002899A (es) | 2007-05-16 |
AU2005281511A1 (en) | 2006-03-16 |
CA2580019A1 (en) | 2006-03-16 |
BRPI0515103A (pt) | 2008-07-08 |
EP1791534A1 (en) | 2007-06-06 |
JP2008512434A (ja) | 2008-04-24 |
WO2006027595A1 (en) | 2006-03-16 |
IL181828A0 (en) | 2007-07-04 |
US20070264202A1 (en) | 2007-11-15 |
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