BRPI0515103A - composição farmacêutica, inalador, processos para preparar o mesmo, e uma composição farmacêutica, e, uso de uma composição farmacêutica - Google Patents
composição farmacêutica, inalador, processos para preparar o mesmo, e uma composição farmacêutica, e, uso de uma composição farmacêuticaInfo
- Publication number
- BRPI0515103A BRPI0515103A BRPI0515103-1A BRPI0515103A BRPI0515103A BR PI0515103 A BRPI0515103 A BR PI0515103A BR PI0515103 A BRPI0515103 A BR PI0515103A BR PI0515103 A BRPI0515103 A BR PI0515103A
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical composition
- preparing
- inhaler
- processes
- solvate
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 7
- 150000003839 salts Chemical class 0.000 abstract 3
- 239000012453 solvate Substances 0.000 abstract 3
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- NDAUXUAQIAJITI-LBPRGKRZSA-N (R)-salbutamol Chemical compound CC(C)(C)NC[C@H](O)C1=CC=C(O)C(CO)=C1 NDAUXUAQIAJITI-LBPRGKRZSA-N 0.000 abstract 1
- 229940121948 Muscarinic receptor antagonist Drugs 0.000 abstract 1
- 230000003454 betamimetic effect Effects 0.000 abstract 1
- 239000000812 cholinergic antagonist Substances 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229960001361 ipratropium bromide Drugs 0.000 abstract 1
- KEWHKYJURDBRMN-ZEODDXGYSA-M ipratropium bromide hydrate Chemical compound O.[Br-].O([C@H]1C[C@H]2CC[C@@H](C1)[N@@+]2(C)C(C)C)C(=O)C(CO)C1=CC=CC=C1 KEWHKYJURDBRMN-ZEODDXGYSA-M 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
COMPOSIçãO FARMACêUTICA, INALADOR, PROCESSOS PARA PREPARAR O MESMO, E UMA COMPOSIçãO FARMACêUTICA, E, USO DE UMA COMPOSIçãO FARMACêUTICA Uma composição farmacêutica em uma forma de dosagem adequada para inalação compreende um isómero terapêutico de um agente betamimético ou uni seu sal, solvato, éster, derivado, ou polimorfo substancialmente livre de isómero(s) menos terapeuticamente eficaz(s) de citado agente e opcionalmente um agente anticolinérgico ou um seu sal, solvato, éster, derivado, isómero ou polimorfo. Uma composição preferida compreende sulfato de R-salbutamol e brometo de ipratrópio. Métodos de preparar as composição da invenção também são proporcionados.
Applications Claiming Priority (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN970MU2004 | 2004-09-09 | ||
IN1004MU2004 | 2004-09-17 | ||
IN1077MU2004 | 2004-10-08 | ||
IN1089MU2004 | 2004-10-11 | ||
IN1088MU2004 | 2004-10-11 | ||
IN93MU2005 | 2005-01-31 | ||
IN222MU2005 | 2005-02-28 | ||
PCT/GB2005/003475 WO2006027595A1 (en) | 2004-09-09 | 2005-09-09 | Pharmaceutical composition comprising an isomer of a betamimetic agent and an anti-cholinergic agent |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0515103A true BRPI0515103A (pt) | 2008-07-08 |
Family
ID=35311711
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0515103-1A BRPI0515103A (pt) | 2004-09-09 | 2005-09-09 | composição farmacêutica, inalador, processos para preparar o mesmo, e uma composição farmacêutica, e, uso de uma composição farmacêutica |
Country Status (11)
Country | Link |
---|---|
US (1) | US20070264202A1 (pt) |
EP (1) | EP1791534A1 (pt) |
JP (1) | JP2008512434A (pt) |
KR (1) | KR20070102659A (pt) |
AU (1) | AU2005281511B2 (pt) |
BR (1) | BRPI0515103A (pt) |
CA (1) | CA2580019A1 (pt) |
EA (1) | EA200700600A1 (pt) |
IL (1) | IL181828A0 (pt) |
MX (1) | MX2007002899A (pt) |
WO (1) | WO2006027595A1 (pt) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0501956D0 (en) * | 2005-01-31 | 2005-03-09 | Arrow Internat | Nebulizer formulation |
US20100144784A1 (en) * | 2006-05-19 | 2010-06-10 | Boehringer Ingelheim International Gmbh | Aerosol formulation |
JP5317961B2 (ja) * | 2006-05-19 | 2013-10-16 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 推進剤を含まないイプラトロピウムブロマイド及びサルブタモールスルフェート含有吸入エアロゾル製剤 |
US20070286814A1 (en) * | 2006-06-12 | 2007-12-13 | Medispray Laboratories Pvt. Ltd. | Stable aerosol pharmaceutical formulations |
EP2077132A1 (en) | 2008-01-02 | 2009-07-08 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dispensing device, storage device and method for dispensing a formulation |
US20110250242A1 (en) * | 2008-10-23 | 2011-10-13 | Sunovion Pharmaceuticals Inc. | Arformoterol and tiotropium compositions and methods for use |
JP5670421B2 (ja) | 2009-03-31 | 2015-02-18 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | コンポーネント表面のコーティング方法 |
EP2432531B1 (de) | 2009-05-18 | 2019-03-06 | Boehringer Ingelheim International GmbH | Adapter, inhalationseinrichtung und zerstäuber |
EP2504051B1 (en) | 2009-11-25 | 2019-09-04 | Boehringer Ingelheim International GmbH | Nebulizer |
US10016568B2 (en) | 2009-11-25 | 2018-07-10 | Boehringer Ingelheim International Gmbh | Nebulizer |
JP5715640B2 (ja) | 2009-11-25 | 2015-05-13 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ネブライザ |
US9943654B2 (en) | 2010-06-24 | 2018-04-17 | Boehringer Ingelheim International Gmbh | Nebulizer |
EP2694220B1 (de) | 2011-04-01 | 2020-05-06 | Boehringer Ingelheim International GmbH | Medizinisches gerät mit behälter |
US9827384B2 (en) | 2011-05-23 | 2017-11-28 | Boehringer Ingelheim International Gmbh | Nebulizer |
WO2013152894A1 (de) | 2012-04-13 | 2013-10-17 | Boehringer Ingelheim International Gmbh | Zerstäuber mit kodiermitteln |
EP3030298B1 (en) | 2013-08-09 | 2017-10-11 | Boehringer Ingelheim International GmbH | Nebulizer |
ES2836977T3 (es) | 2013-08-09 | 2021-06-28 | Boehringer Ingelheim Int | Nebulizador |
CN106232166B (zh) | 2014-05-07 | 2020-04-14 | 勃林格殷格翰国际有限公司 | 喷雾器 |
PL3139984T3 (pl) | 2014-05-07 | 2021-11-08 | Boehringer Ingelheim International Gmbh | Nebulizator |
CN106255554B (zh) | 2014-05-07 | 2021-05-04 | 勃林格殷格翰国际有限公司 | 容器、喷雾器及用途 |
EP3569221A1 (en) * | 2018-05-17 | 2019-11-20 | Notoxins IP B.V. | Aqueous formulations comprising ipratropium for topical treatment of hyperhidrosis |
CN113018280A (zh) * | 2021-03-01 | 2021-06-25 | 石家庄四药有限公司 | 一种异丙托溴铵吸入用溶液制剂及其制备方法 |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5192528A (en) * | 1985-05-22 | 1993-03-09 | Liposome Technology, Inc. | Corticosteroid inhalation treatment method |
US5919827A (en) * | 1990-07-11 | 1999-07-06 | Sepracor Inc. | Method for treating asthma using optically pure R(-) salmeterol |
US5795564A (en) * | 1991-04-05 | 1998-08-18 | Sepracor, Inc. | Methods and compositions for treating pulmonary disorders using optically pure (R,R)-formoterol |
US6299863B1 (en) * | 1992-04-03 | 2001-10-09 | Sepracor Inc. | Aerosol formulations containing micronized optically pure (R,R) formoterol for bronchodilating therapy |
US6423298B2 (en) * | 1998-06-18 | 2002-07-23 | Boehringer Ingelheim Pharmaceuticals, Inc. | Pharmaceutical formulations for aerosols with two or more active substances |
GB9827200D0 (en) * | 1998-12-11 | 1999-02-03 | Glaxo Group Ltd | Dry powder inhaler |
WO2001064274A2 (en) * | 2000-03-01 | 2001-09-07 | Glaxo Group Limited | Metered dose inhaler |
US20040019025A1 (en) * | 2000-04-18 | 2004-01-29 | Gavin Brian Charles | Medical compositions comprising (r,r)-formoterol and rofleponide |
GB0009607D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Medical compositions |
CA2417973A1 (en) * | 2000-08-04 | 2002-02-14 | Longwood Pharmaceutical Research, Inc. | Formulations of mometasone and a bronchodilator for pulmonary administration |
US20040050385A1 (en) * | 2000-10-20 | 2004-03-18 | Bonney Stanley George | Inhaler |
GB0030171D0 (en) * | 2000-12-11 | 2001-01-24 | Cipla Ltd | Process for preparing isomers of salbutamol |
US20020189610A1 (en) * | 2001-02-01 | 2002-12-19 | Karl-Heinz Bozung | Pharmaceutical compositions containing an ipratropium salt and a betamimetic |
GB0105560D0 (en) * | 2001-03-07 | 2001-04-25 | Glaxo Group Ltd | Pharmaceutical formulations |
US6667344B2 (en) * | 2001-04-17 | 2003-12-23 | Dey, L.P. | Bronchodilating compositions and methods |
JP2003221335A (ja) * | 2001-10-26 | 2003-08-05 | Dey Lp | 慢性閉塞性肺疾患の症状を緩和するためのアルブテロールおよびイプラトロピウム吸入溶液、システム、キットおよび方法 |
EP1671942B2 (en) * | 2002-12-10 | 2014-07-23 | Sunovion Pharmaceuticals Inc. | Aerosol formulation comprising levalbuterol L-tartrate salt |
US20040191176A1 (en) * | 2003-03-28 | 2004-09-30 | Kaplan Leonard W | Formulations for treatment of pulmonary disorders |
-
2005
- 2005-09-09 BR BRPI0515103-1A patent/BRPI0515103A/pt not_active IP Right Cessation
- 2005-09-09 EP EP05786158A patent/EP1791534A1/en not_active Withdrawn
- 2005-09-09 WO PCT/GB2005/003475 patent/WO2006027595A1/en active Application Filing
- 2005-09-09 CA CA002580019A patent/CA2580019A1/en not_active Abandoned
- 2005-09-09 JP JP2007530766A patent/JP2008512434A/ja active Pending
- 2005-09-09 MX MX2007002899A patent/MX2007002899A/es not_active Application Discontinuation
- 2005-09-09 US US11/574,902 patent/US20070264202A1/en not_active Abandoned
- 2005-09-09 AU AU2005281511A patent/AU2005281511B2/en not_active Ceased
- 2005-09-09 KR KR1020077008004A patent/KR20070102659A/ko not_active Application Discontinuation
- 2005-09-09 EA EA200700600A patent/EA200700600A1/ru unknown
-
2007
- 2007-03-08 IL IL181828A patent/IL181828A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
KR20070102659A (ko) | 2007-10-19 |
EP1791534A1 (en) | 2007-06-06 |
CA2580019A1 (en) | 2006-03-16 |
IL181828A0 (en) | 2007-07-04 |
EA200700600A1 (ru) | 2008-02-28 |
JP2008512434A (ja) | 2008-04-24 |
US20070264202A1 (en) | 2007-11-15 |
AU2005281511B2 (en) | 2011-03-31 |
AU2005281511A1 (en) | 2006-03-16 |
MX2007002899A (es) | 2007-05-16 |
WO2006027595A1 (en) | 2006-03-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2260 DE 29/04/2014. |