EA200000946A1 - Кристаллическая форма пароксетина - Google Patents
Кристаллическая форма пароксетинаInfo
- Publication number
- EA200000946A1 EA200000946A1 EA200000946A EA200000946A EA200000946A1 EA 200000946 A1 EA200000946 A1 EA 200000946A1 EA 200000946 A EA200000946 A EA 200000946A EA 200000946 A EA200000946 A EA 200000946A EA 200000946 A1 EA200000946 A1 EA 200000946A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- paroxetin
- crystal form
- paroxetine
- depression
- therapy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Настоящее изобретение относится к чистому, не содержащему растворителя, например, кристаллическому свободному основанию пароксетина и его применению в терапии для лечения депрессии.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9805581.7A GB9805581D0 (en) | 1998-03-16 | 1998-03-16 | Novel compounds |
GBGB9813054.5A GB9813054D0 (en) | 1998-06-17 | 1998-06-17 | Novel compounds |
GBGB9817115.0A GB9817115D0 (en) | 1998-08-06 | 1998-08-06 | Novel compounds |
PCT/GB1999/000793 WO1999047519A1 (en) | 1998-03-16 | 1999-03-16 | Crystalline form of paroxetine |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200000946A1 true EA200000946A1 (ru) | 2001-02-26 |
Family
ID=27269245
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200000946A EA200000946A1 (ru) | 1998-03-16 | 1999-03-16 | Кристаллическая форма пароксетина |
Country Status (18)
Country | Link |
---|---|
EP (1) | EP1064282A1 (ru) |
JP (1) | JP2002506865A (ru) |
KR (1) | KR20010041947A (ru) |
CN (1) | CN1300286A (ru) |
AP (1) | AP2000001907A0 (ru) |
AU (1) | AU2847199A (ru) |
BG (1) | BG104839A (ru) |
BR (1) | BR9908825A (ru) |
CA (1) | CA2323896A1 (ru) |
EA (1) | EA200000946A1 (ru) |
HU (1) | HUP0101215A3 (ru) |
ID (1) | ID27596A (ru) |
IL (1) | IL138390A0 (ru) |
NO (1) | NO20004583L (ru) |
PL (1) | PL342931A1 (ru) |
SK (1) | SK13622000A3 (ru) |
TR (1) | TR200002675T2 (ru) |
WO (1) | WO1999047519A1 (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH689805A8 (fr) * | 1998-07-02 | 2000-02-29 | Smithkline Beecham Plc | Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant. |
GB9919052D0 (en) * | 1999-08-12 | 1999-10-13 | Smithkline Beecham Plc | Novel compound composition and process |
US20080033050A1 (en) | 2006-08-04 | 2008-02-07 | Richards Patricia Allison Tewe | Method of treating thermoregulatory disfunction with paroxetine |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1422263A (en) * | 1973-01-30 | 1976-01-21 | Ferrosan As | 4-phenyl-piperidine compounds |
EP0223403B1 (en) * | 1985-10-25 | 1993-08-04 | Beecham Group Plc | Piperidine derivative, its preparation, and its use as medicament |
SK283608B6 (sk) * | 1995-02-06 | 2003-10-07 | Smithkline Beecham Plc | Bezvodý hydrochlorid paroxetínu, spôsob jeho výroby a použitie |
-
1999
- 1999-03-16 IL IL13839099A patent/IL138390A0/xx unknown
- 1999-03-16 EP EP99909104A patent/EP1064282A1/en not_active Withdrawn
- 1999-03-16 EA EA200000946A patent/EA200000946A1/ru unknown
- 1999-03-16 ID IDW20001813A patent/ID27596A/id unknown
- 1999-03-16 WO PCT/GB1999/000793 patent/WO1999047519A1/en not_active Application Discontinuation
- 1999-03-16 AP APAP/P/2000/001907A patent/AP2000001907A0/en unknown
- 1999-03-16 SK SK1362-2000A patent/SK13622000A3/sk unknown
- 1999-03-16 JP JP2000536714A patent/JP2002506865A/ja active Pending
- 1999-03-16 CN CN99806077A patent/CN1300286A/zh active Pending
- 1999-03-16 AU AU28471/99A patent/AU2847199A/en not_active Abandoned
- 1999-03-16 TR TR2000/02675T patent/TR200002675T2/xx unknown
- 1999-03-16 CA CA002323896A patent/CA2323896A1/en not_active Abandoned
- 1999-03-16 KR KR1020007010260A patent/KR20010041947A/ko not_active Application Discontinuation
- 1999-03-16 HU HU0101215A patent/HUP0101215A3/hu unknown
- 1999-03-16 PL PL99342931A patent/PL342931A1/xx unknown
- 1999-03-16 BR BR9908825-8A patent/BR9908825A/pt not_active Application Discontinuation
-
2000
- 2000-09-14 NO NO20004583A patent/NO20004583L/no not_active Application Discontinuation
- 2000-10-11 BG BG104839A patent/BG104839A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
BG104839A (en) | 2001-09-28 |
SK13622000A3 (sk) | 2001-03-12 |
TR200002675T2 (tr) | 2000-12-21 |
AU2847199A (en) | 1999-10-11 |
CN1300286A (zh) | 2001-06-20 |
HUP0101215A2 (hu) | 2002-04-29 |
BR9908825A (pt) | 2000-11-21 |
PL342931A1 (en) | 2001-07-16 |
CA2323896A1 (en) | 1999-09-23 |
KR20010041947A (ko) | 2001-05-25 |
NO20004583L (no) | 2000-09-15 |
AP2000001907A0 (en) | 2000-09-30 |
ID27596A (id) | 2001-04-12 |
WO1999047519A1 (en) | 1999-09-23 |
JP2002506865A (ja) | 2002-03-05 |
HUP0101215A3 (en) | 2002-05-28 |
EP1064282A1 (en) | 2001-01-03 |
NO20004583D0 (no) | 2000-09-14 |
IL138390A0 (en) | 2001-10-31 |
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