DK634689D0 - Anvendelse af castanospermin-estere eller deres salte til fremstilling af laegemidler, der inhiberer tumor-metastaser - Google Patents

Anvendelse af castanospermin-estere eller deres salte til fremstilling af laegemidler, der inhiberer tumor-metastaser

Info

Publication number
DK634689D0
DK634689D0 DK634689A DK634689A DK634689D0 DK 634689 D0 DK634689 D0 DK 634689D0 DK 634689 A DK634689 A DK 634689A DK 634689 A DK634689 A DK 634689A DK 634689 D0 DK634689 D0 DK 634689D0
Authority
DK
Denmark
Prior art keywords
esters
salts
castanospermin
preparation
tumor metastases
Prior art date
Application number
DK634689A
Other languages
English (en)
Other versions
DK634689A (da
Inventor
Sai Prasad Sunkara
Paul Saiho Liu
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of DK634689D0 publication Critical patent/DK634689D0/da
Publication of DK634689A publication Critical patent/DK634689A/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK634689A 1988-12-15 1989-12-14 Anvendelse af castanospermin-estere eller deres salte til fremstilling af laegemidler, der inhiberer tumor-metastaser DK634689A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/284,510 US4952585A (en) 1988-12-15 1988-12-15 Castanospermine esters in the inhibition of tumor metastasis

Publications (2)

Publication Number Publication Date
DK634689D0 true DK634689D0 (da) 1989-12-14
DK634689A DK634689A (da) 1990-06-16

Family

ID=23090466

Family Applications (1)

Application Number Title Priority Date Filing Date
DK634689A DK634689A (da) 1988-12-15 1989-12-14 Anvendelse af castanospermin-estere eller deres salte til fremstilling af laegemidler, der inhiberer tumor-metastaser

Country Status (12)

Country Link
US (1) US4952585A (da)
EP (1) EP0373663B1 (da)
JP (1) JP2963476B2 (da)
KR (1) KR0135278B1 (da)
AT (1) ATE96320T1 (da)
AU (1) AU621431B2 (da)
DE (1) DE68910287T2 (da)
DK (1) DK634689A (da)
ES (1) ES2061912T3 (da)
IE (1) IE62014B1 (da)
PH (1) PH26024A (da)
ZA (1) ZA899451B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5004746A (en) * 1987-09-29 1991-04-02 Merrell Dow Pharmaceuticals Inc. Anti-retroviral castanospermine esters
US4970317A (en) * 1989-08-08 1990-11-13 Merrell Dow Pharmaceuticals Inc. Process for the preparation of castanospermine esters
DK0983270T3 (da) * 1997-05-22 2004-05-10 Aventis Pharma Inc Fremgangsmåde til fremstilling af 6-O-monoestere af castanospermin
US5959111A (en) * 1997-05-22 1999-09-28 Hoechst Marion Roussel, Inc. Process for preparing 6-0-monoesters of castanospermine
US6013459A (en) * 1997-06-12 2000-01-11 Clinical Micro Sensors, Inc. Detection of analytes using reorganization energy
EP2049126A2 (en) * 2006-08-02 2009-04-22 United Therapeutics Corporation Liposome treatment of viral infections
WO2009118658A2 (en) * 2008-03-26 2009-10-01 University Of Oxford Endoplasmic reticulum targeting liposomes
US8226684B2 (en) * 2008-12-22 2012-07-24 Ethicon, Inc. Surgical sutures having collapsible tissue anchoring protrusions and methods therefor
WO2010109330A2 (en) * 2009-03-27 2010-09-30 University Of Oxford Cholesterol level lowering liposomes
WO2017138008A2 (en) * 2016-02-14 2017-08-17 Yeda Research And Development Co. Ltd. Methods of modulating protein exocytosis and uses of same in therapy
WO2018059214A1 (zh) 2016-09-29 2018-04-05 广州君赫生物科技有限公司 影响saicar合成的化合物及应用
KR20190122242A (ko) 2017-04-20 2019-10-29 진힐 바이오테크놀로지 컴퍼니 리미티드 항종양 약물의 제조에서의 스페르민 및 그 유도체의 응용
EP3613731A4 (en) 2017-04-20 2021-01-13 Geneheal Biotechnology Co., Ltd. APPLICATIONS OF SPERMIDINE AND ITS DERIVATIVE

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4792558A (en) * 1987-05-29 1988-12-20 Merrell Dow Pharmaceuticals Inc. Castanospermine for inhibiting tumor metastasis
CA1315276C (en) * 1987-07-02 1993-03-30 Paul S. Liu Castanospermine esters and glycosides
US5004746A (en) * 1987-09-29 1991-04-02 Merrell Dow Pharmaceuticals Inc. Anti-retroviral castanospermine esters
AU618838B2 (en) * 1988-08-10 1992-01-09 Praxis Pharmaceuticals, Inc. Use of castanospermine as an anti-inflammatory and immunosuppressant agent

Also Published As

Publication number Publication date
DE68910287D1 (de) 1993-12-02
IE894009L (en) 1990-06-15
DE68910287T2 (de) 1994-03-10
IE62014B1 (en) 1994-12-14
EP0373663A3 (en) 1990-09-12
AU4670789A (en) 1990-06-21
AU621431B2 (en) 1992-03-12
KR910011256A (ko) 1991-08-07
EP0373663A2 (en) 1990-06-20
KR0135278B1 (ko) 1998-04-23
DK634689A (da) 1990-06-16
US4952585A (en) 1990-08-28
ZA899451B (en) 1990-09-26
ES2061912T3 (es) 1994-12-16
JP2963476B2 (ja) 1999-10-18
EP0373663B1 (en) 1993-10-27
PH26024A (en) 1992-01-24
ATE96320T1 (de) 1993-11-15
JPH02212427A (ja) 1990-08-23

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment