DK530480A - Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin - Google Patents

Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin

Info

Publication number
DK530480A
DK530480A DK530480A DK530480A DK530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A
Authority
DK
Denmark
Prior art keywords
ethanon
piperidyl
quinolyl
intermediates
medicine
Prior art date
Application number
DK530480A
Other languages
English (en)
Inventor
A Champseix
G L Fur
C Renault
Original Assignee
Pharmindustrie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmindustrie filed Critical Pharmindustrie
Publication of DK530480A publication Critical patent/DK530480A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/34Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK530480A 1979-12-21 1980-12-12 Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin DK530480A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7931396A FR2471981A1 (fr) 1979-12-21 1979-12-21 Nouveaux derives de la (piperidyl-4)-2 (quinolyl-4)-1 ethanone, produits intermediaires et procedes pour leur preparation, et leur utilisation comme medicaments

Publications (1)

Publication Number Publication Date
DK530480A true DK530480A (da) 1981-06-22

Family

ID=9233056

Family Applications (1)

Application Number Title Priority Date Filing Date
DK530480A DK530480A (da) 1979-12-21 1980-12-12 Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin

Country Status (12)

Country Link
US (2) US4433150A (da)
EP (1) EP0031753B1 (da)
JP (1) JPS5699476A (da)
AT (1) AT376670B (da)
CA (1) CA1178589A (da)
DE (1) DE3069243D1 (da)
DK (1) DK530480A (da)
ES (3) ES498017A0 (da)
FR (1) FR2471981A1 (da)
IE (1) IE51124B1 (da)
NO (1) NO155137C (da)
PT (1) PT72212A (da)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7908031A (nl) * 1979-11-01 1981-06-01 Acf Chemiefarma Nv Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
US4442107A (en) * 1980-03-06 1984-04-10 Acf Chemiefarma N.V. Quinoline derivatives, pharmaceutical compositions containing such compounds, and methods for treating cardiovascular conditions with them
FR2495470A1 (fr) * 1980-12-05 1982-06-11 Pharmindustrie Nouveaux medicaments a base de derives de (quinolyl-4)-1 (piperidyl-4)-2 ethanol ou (quinolyl-4)-1 (piperidyl-4)-3 propanol
FR2582514B1 (fr) * 1985-05-30 1988-02-19 Rhone Poulenc Sante Medicaments a base d'amides, nouveaux amides et leur preparation
US6103903A (en) 1998-02-26 2000-08-15 Neurogen Corporation 4-(4-piperidylmethyhlamino) substituted heteroaryl fused pyridines: GABA brain receptor ligands
GB9917406D0 (en) 1999-07-23 1999-09-22 Smithkline Beecham Plc Compounds
GB9917408D0 (en) 1999-07-23 1999-09-22 Smithkline Beecham Plc Compounds
US6693099B2 (en) * 2000-10-17 2004-02-17 The Procter & Gamble Company Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
US6376514B1 (en) * 2000-10-17 2002-04-23 The Procter & Gamble Co. Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof
AU2002365611A1 (en) * 2001-12-05 2003-06-17 F. Hoffmann - La Roche Ag Inflammation modulators
EP2181996A1 (en) 2002-01-29 2010-05-05 Glaxo Group Limited Aminopiperidine derivatives
FR2858619B1 (fr) * 2003-08-08 2006-12-22 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
US7348434B2 (en) 2003-08-08 2008-03-25 Antony Bigot 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
MX2009012117A (es) * 2007-05-09 2009-11-23 Pfizer Composiciones y derivados heterociclicos sustituidos y su uso farmaceutico como antibacterianos.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR31753E (fr) * 1925-12-03 1927-06-11 Appareil photographique pour prise de vues, agrandissement et projection
FR42781E (fr) * 1932-05-23 1933-10-10 Perfectionnements aux machines rotatives à capsuler les bouteilles
FR959917A (da) * 1946-06-25 1950-04-07
FR2177511A1 (en) * 1972-03-28 1973-11-09 Omnium Chimique Sa Quinolyl pipiridylethyl ketones - with vasodilatory and antispasmodic activity
PT66682B (pt) * 1976-06-18 1978-11-15 Ind Biolog Francaise /(quinolyl-4)-propyl-1/-4 piperidines leur preparation et leur utilisation comme medicaments /(quinolyl-4)-propyl/-4 piperidines leur preparation et leur utilisation comme medicaments
FR2354771A1 (fr) * 1976-06-18 1978-01-13 Mar Pha Etu Expl Marques ((quinolyl-4)-3 propyl-1) -4 piperidines, leur preparation et leur utilisation comme medicaments
FR2485014A1 (fr) * 1980-06-20 1981-12-24 Pharmindustrie Nouveaux derives de (quinolyl-2, -3 ou -4)-1 (piperidyl ou pyrrolidinyl-2 ou -3)-2 ou -3 ethanone ou propanone, procedes pour leur preparation, et leur utilisation comme medicaments

Also Published As

Publication number Publication date
NO803881L (no) 1981-06-22
ES507997A0 (es) 1982-10-01
EP0031753B1 (fr) 1984-09-19
ES8300745A1 (es) 1982-11-01
ATA609680A (de) 1984-05-15
JPS5699476A (en) 1981-08-10
FR2471981A1 (fr) 1981-06-26
US4505916A (en) 1985-03-19
ES507998A0 (es) 1982-10-01
DE3069243D1 (en) 1984-10-25
ES8207526A1 (es) 1982-10-01
CA1178589A (fr) 1984-11-27
IE51124B1 (en) 1986-10-15
EP0031753A1 (fr) 1981-07-08
NO155137C (no) 1987-02-18
US4433150A (en) 1984-02-21
FR2471981B1 (da) 1983-03-25
IE802684L (en) 1981-06-21
AT376670B (de) 1984-12-27
ES8207525A1 (es) 1982-10-01
ES498017A0 (es) 1982-11-01
PT72212A (pt) 1981-01-01
NO155137B (no) 1986-11-10

Similar Documents

Publication Publication Date Title
DK530480A (da) Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin
DK3880A (da) Fremgangsmaade til fremstilling af peptidylargininaldehydderivater og disses anvendelse
DK519481A (da) Carboxylkylaminosyrederivater af substituerede proliner fremgangsmaade til fremstilling heraf samt deres anvendelse som laegemidler
DK445280A (da) Fremgangsmaade til fremstilling af quinolinderivater
DK214480A (da) Fremgangsmaade til fremstilling af 2-(pyrimidinylamino)-1,3-diaza-2-cycloalkenforbindelser deres tautomere forbindelser og syreadditionssalte deraf
DK265780A (da) Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling
DK271981A (da) Hidtil ukendte derivater af 1-(2-, 3- eller 4-quinolyl)-2- eller -3(2- eller 3-piperidyl eller- pyrrolidimyl)-ethanon eller propanon fremgangsmaader til deres fremstilling og deres anvendelse som laegemidler
NO793993L (no) Nye silyl-glucoseaminderivater og fremgangsmaate til deres fremstilling
DK379380A (da) Fremgangsmaade til fremstilling af 1-aminocyclopropan-carbolsyre og derivater deraf
DK570486D0 (da) Heterocyclisk substituerede 2(1h)-quinoloner, deres anvendelse til fremstilling af hjertestimulerende laegemidler, farmaceutiske praeparater indeholdende forbindelserne og mellemprodukter ved deres fremstilling
DK11480A (da) Fremgangsmaade til fremstilling af anthracyclinderivater og syreadditionssalte deraf
DK205180A (da) Fluorerede 1-triazolyl-butan-derivater deres fremstilling og anvendelse som fungicider
DK528381A (da) Substituerede phenoxykanelsyrederivater fremgangsmaade til fremstilling deraf samt deres anvendelse som herbicider samt mellemprodukter og deres fremstilling
DK154382A (da) Hidtil ukendte derivater af 2-piperazinopyrimidin,fremgangsmaader til deres fremstilling og deres anvendelse som laegemidlereller mellemprodukter til fremstilling af laegemidler
DK154650C (da) Analogifremgangsmaade til fremstilling af sukkerderivater
DK258381A (da) Hidtil ukendte indenderivater fremgangsmaader til deres fremstilling og deres anvendelse som laegemidler
DK289585D0 (da) Arylderivater af heterobicycliske forbindelser, deres farmaceutiske anvendelse og deres fremstilling
DK148680A (da) Fremgangsmaade til fremstilling af xanthinderivater
DK287681A (da) Metaphenylendiaminer fremgangsmaade til deres fremstilling farvningskompositioner indeholdende forbindelserne og fremgangsmaade til farvning dermed
DK101481A (da) Hidtil ukendte derivater af 3-chlorquinolin fremgangsmaader til deres fremstilling og deres anvendelse som laegemidler
DK317678A (da) Fremgangsmaade til fremstilling af 3-(1-pyrazolyl)-pyridazindf erivater eller farmaceutisk acceptable syreaddtionssalte dera
DK433381A (da) Fremgangsmaade til fremstilling af 3-brom-4-fluorbenzylalkohol3-brom-4-fluorbenozesyre-derivater og fremgangsmaade til deres fremstilling
DK401280A (da) Acylerede imidazolyl-gamma-fluorpinacolyl-derivater fremgangsmaade til deres fremstilling og deres anvendelse som fungicider
DK284780A (da) Fremgangsmaade til fremstilling af cyclopropan-1-carboxyl-syrederivater perfluoralkylsulfonmellemprodukter hertil og disses fremstilling
NO790564L (no) Nye nitrosourinstoff-derivater og fremgangsmaate til deres fremstilling.

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment