DK529585A - N-(6-methoxy-5-(perflouralkyl)-1-naphtholyl)-n-methylglyciner og deres thionaphthoyl analoge, deres fremstilling og anvendelse som laegemidler - Google Patents

N-(6-methoxy-5-(perflouralkyl)-1-naphtholyl)-n-methylglyciner og deres thionaphthoyl analoge, deres fremstilling og anvendelse som laegemidler Download PDF

Info

Publication number
DK529585A
DK529585A DK529585A DK529585A DK529585A DK 529585 A DK529585 A DK 529585A DK 529585 A DK529585 A DK 529585A DK 529585 A DK529585 A DK 529585A DK 529585 A DK529585 A DK 529585A
Authority
DK
Denmark
Prior art keywords
preparation
perflouralkyl
methylgylines
thionaphthoyl
naphtholyl
Prior art date
Application number
DK529585A
Other languages
English (en)
Other versions
DK166147C (da
DK166147B (da
DK529585D0 (da
Inventor
Francesco Bellini
Kazimir Sestanj
Original Assignee
Ayerst Mckenna & Harrison
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ayerst Mckenna & Harrison filed Critical Ayerst Mckenna & Harrison
Publication of DK529585D0 publication Critical patent/DK529585D0/da
Publication of DK529585A publication Critical patent/DK529585A/da
Publication of DK166147B publication Critical patent/DK166147B/da
Application granted granted Critical
Publication of DK166147C publication Critical patent/DK166147C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/83—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/12—Ophthalmic agents for cataracts
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Seasonings (AREA)
DK529585A 1984-11-16 1985-11-15 N-oe6-methoxy-5-(perflouralkyl)-1-naphthoylaa-n-methylglyciner og deres thionaphthoylanaloge, deres fremstilling og farmaceutiske praeparater indeholdende dem DK166147C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67201584 1984-11-16
US06/672,015 US4604406A (en) 1984-11-16 1984-11-16 N-[6-methoxy-5-(perfluoroalkyl)-1-naphtholyl]-N-methylglycines and their thionaphthoyl analogs

Publications (4)

Publication Number Publication Date
DK529585D0 DK529585D0 (da) 1985-11-15
DK529585A true DK529585A (da) 1986-05-17
DK166147B DK166147B (da) 1993-03-15
DK166147C DK166147C (da) 1993-08-09

Family

ID=24696806

Family Applications (1)

Application Number Title Priority Date Filing Date
DK529585A DK166147C (da) 1984-11-16 1985-11-15 N-oe6-methoxy-5-(perflouralkyl)-1-naphthoylaa-n-methylglyciner og deres thionaphthoylanaloge, deres fremstilling og farmaceutiske praeparater indeholdende dem

Country Status (18)

Country Link
US (1) US4604406A (da)
EP (1) EP0182499B1 (da)
JP (1) JPH0611739B2 (da)
KR (1) KR900006128B1 (da)
AT (1) ATE42091T1 (da)
AU (1) AU583311B2 (da)
CA (1) CA1253520A (da)
DE (1) DE3569367D1 (da)
DK (1) DK166147C (da)
ES (1) ES8801619A1 (da)
GE (1) GEP19981385B (da)
GR (1) GR852726B (da)
HU (1) HU194159B (da)
IE (1) IE58620B1 (da)
PH (1) PH21450A (da)
SU (1) SU1468897A1 (da)
UA (1) UA7051A1 (da)
ZA (1) ZA858186B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4699993A (en) * 1985-12-12 1987-10-13 Ethyl Corporation Perfluoroalkylnaphthalene compounds
US4822904A (en) * 1985-12-12 1989-04-18 Ethyl Corporation Perfluoroalkylation process
US4734435A (en) * 1986-04-07 1988-03-29 American Home Products Corp. N-[[6-methoxy-5-(trifluoromethyl)-1-naphthalenyl]-thioxomethyl]-N-methylglycine S-oxide and the amide thereof
JPS6399057A (ja) * 1986-06-27 1988-04-30 Nippon Shinyaku Co Ltd グリシン誘導体
US4731380A (en) * 1986-08-26 1988-03-15 American Home Products Corporation (Del.) Tolerstat as an agent for diabetic periodontitis
EP0306525A4 (en) * 1987-03-20 1991-04-24 Alcon Laboratories Inc Use of aldose reductase inhibitors to enhance insulin sensitivity in diabetes mellitus
JP2548258Y2 (ja) * 1990-12-21 1997-09-17 ペガサスミシン製造株式会社 自動口伏せ縫い装置
US5388146A (en) * 1991-11-12 1995-02-07 Microlog Corporation Automated telephone system using multiple languages
US5337844A (en) * 1992-07-16 1994-08-16 Baker Hughes, Incorporated Drill bit having diamond film cutting elements
US20150057452A1 (en) 2012-04-04 2015-02-26 Catylix, Inc. Selective androgen receptor modulators

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4254108A (en) * 1979-11-08 1981-03-03 Ayerst, Mckenna & Harrison Inc. Thioxo-1H-benz[de]isoquinoline-2(3H)-acetic acid derivatives and antidiabetic use thereof
US4254109A (en) * 1979-11-08 1981-03-03 Ayerst, Mckenna & Harrison Inc. 1H-Benz[de]isoquinoline-2(3H)-acetic acid derivatives
CA1191156A (en) * 1981-10-15 1985-07-30 Francesco Bellini N-((6-(lower alkoxy)-5-(trifluoromethylthio)-1- naphthalenyl)-thioxomethyl)-n-(lower alkyl)glycines
AU544067B2 (en) * 1981-03-02 1985-05-16 Wyeth-Ayerst Canada Inc. Thioamides and amides. treatment of diabetes
CA1182472A (en) * 1981-03-02 1985-02-12 Kazimir Sestanj N-[(2-naphthalenyl)thioxomethyl]glycine derivatives
CA1176269A (en) * 1981-03-02 1984-10-16 Kazimir Sestanj N-naphthoylglycine derivatives
CA1147739A (en) * 1981-03-02 1983-06-07 Kazimir Sestanj N-(naphthalenylthioxomethyl)aminoacid derivatives
US4369188A (en) * 1981-07-17 1983-01-18 Ayerst, Mckenna & Harrison Inc. 2-Thioxobenz[cd]indole-1(2H)-acetic acid derivatives

Also Published As

Publication number Publication date
DK166147C (da) 1993-08-09
PH21450A (en) 1987-10-28
DK166147B (da) 1993-03-15
ZA858186B (en) 1987-06-24
KR860004010A (ko) 1986-06-16
CA1253520A (en) 1989-05-02
JPS61122256A (ja) 1986-06-10
JPH0611739B2 (ja) 1994-02-16
ATE42091T1 (de) 1989-04-15
GR852726B (da) 1986-03-13
DE3569367D1 (en) 1989-05-18
HU194159B (en) 1988-01-28
IE852598L (en) 1986-05-16
AU4898185A (en) 1986-05-22
UA7051A1 (uk) 1995-03-31
HUT42059A (en) 1987-06-29
EP0182499B1 (en) 1989-04-12
AU583311B2 (en) 1989-04-27
DK529585D0 (da) 1985-11-15
ES548914A0 (es) 1988-02-16
KR900006128B1 (ko) 1990-08-24
ES8801619A1 (es) 1988-02-16
IE58620B1 (en) 1993-10-20
EP0182499A1 (en) 1986-05-28
US4604406A (en) 1986-08-05
SU1468897A1 (ru) 1989-03-30
GEP19981385B (en) 1998-11-10

Similar Documents

Publication Publication Date Title
ES539658A0 (es) Procedimiento de preparacion de nuevos derivados de la xan- tina y de sus sales de adicion con acidos apropiados
DK13382A (da) (2-halogenergolinyl)-n!,n!-diethylurinstofderivater fremgangsmaade til deres fremstilling og deres anvendelse som laegemiddel
ES2064461T3 (es) Derivados de xantina, procedimiento para su preparacion y composicion farmaceutica.
ES8609204A1 (es) Procedimiento de preparar derivados aminicos
DK529585D0 (da) N-(6-methoxy-5-(perflouralkyl)-1-naphtholyl)-n-methylglyciner og deres thionaphthoyl analoge, deres fremstilling og anvendelse som laegemidler
DK0508740T3 (da) Thiazolidindionderivater, deres fremstilling og anvendelse.
DK0392560T3 (da) Diaminoethylenforbindelser
DK592688D0 (da) Benz(thi)amidderivater, deres fremstilling og anvendelse som fungicider
BR8404861A (pt) Processo para obtencao de derivados de ciclo-hexenona,e,composicoes herbicidas a base dos mesmos
PT89757A (pt) Processo para a preparacao de novos derivados da xantina e de composicoes farmaceuticas que os contem, uteis no tratamento da ulcera peptica
DK440987D0 (da) Thyroninderivater, deres fremstilling og anvendelse
FI854512A (fi) Ny kristallform av benzotiazin-dioxidsaltet.
FI874311A0 (fi) 7-/(meta-substituerade)fenylglysin/ -1-karba-1-detiakefalosporiner.
NZ240404A (en) Oxysulphonyl (thio)carbamate derivatives and pharmaceutical
ES2053079T3 (es) Piridazinaminas con actividad anti-rinoviral.
DK0432841T3 (da) Spiro-indolin-oxazin-forbindelser med fotokromatiske og fotosensibiliserende egenskaber samt fremgangsmåde til deres fremstilling
DK455185A (da) Pyridinderivater
ATE144900T1 (de) Verwendung von xanthinderivaten gegen magengeschwüre
DK311284A (da) 3-(4'-aminobutylamino)-propylamino-bleomycin-derivater, deres fremstilling og deres anvendelse som laegemidler
DK162715C (da) 2-nitromethylen-tetrahydro-2h-1,3-thiazinderivater, en fremgangsmaade til deres fremstilling og deres anvendelse som pesticider
DK0565579T3 (da) 2-Imino-6-polyfluoralkyl-3-heterocyclylalkylbenzothiazolin-derivater, deres fremstilling og lægemidler med indhold deraf

Legal Events

Date Code Title Description
PBP Patent lapsed