DK468184D0 - Fremgangsmaade til fremstilling af substituerede 4-alkyl-2(1h)-quinazolinon-1-alkansyrederivater - Google Patents

Fremgangsmaade til fremstilling af substituerede 4-alkyl-2(1h)-quinazolinon-1-alkansyrederivater

Info

Publication number
DK468184D0
DK468184D0 DK468184A DK468184A DK468184D0 DK 468184 D0 DK468184 D0 DK 468184D0 DK 468184 A DK468184 A DK 468184A DK 468184 A DK468184 A DK 468184A DK 468184 D0 DK468184 D0 DK 468184D0
Authority
DK
Denmark
Prior art keywords
quinazolinon
alkyl
acid derivatives
preparing substituted
alkanic acid
Prior art date
Application number
DK468184A
Other languages
English (en)
Other versions
DK468184A (da
Inventor
Ramesh M Kanojia
Victor T Bandurco
Seymour D Levine
Alfonso J Tobia
Dennis M Mulvey
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/537,232 external-priority patent/US4555570A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK468184D0 publication Critical patent/DK468184D0/da
Publication of DK468184A publication Critical patent/DK468184A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK468184A 1983-09-29 1984-09-28 Fremgangsmaade til fremstilling af substituerede 4-alkyl-2(1h)-quinazolinon-1-alkansyrederivater DK468184A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/537,232 US4555570A (en) 1983-09-29 1983-09-29 Substituted 4-alkyl-2-(1H) quinazolinone-1-alkanoic acid derivatives
US06/627,139 US4556739A (en) 1983-09-29 1984-07-02 3,4-Dialkoxy-2-alkylcarbonyl analino compounds

Publications (2)

Publication Number Publication Date
DK468184D0 true DK468184D0 (da) 1984-09-28
DK468184A DK468184A (da) 1985-03-30

Family

ID=27065422

Family Applications (1)

Application Number Title Priority Date Filing Date
DK468184A DK468184A (da) 1983-09-29 1984-09-28 Fremgangsmaade til fremstilling af substituerede 4-alkyl-2(1h)-quinazolinon-1-alkansyrederivater

Country Status (7)

Country Link
US (1) US4556739A (da)
EP (1) EP0138492A3 (da)
KR (1) KR900001200B1 (da)
AU (1) AU565001B2 (da)
DK (1) DK468184A (da)
GR (1) GR80505B (da)
NO (1) NO843908L (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4731480A (en) * 1985-07-29 1988-03-15 Ortho Pharmaceutical Corporation Process for preparing 2-acyl-3,4-dialkoxyanilines
KR900003529B1 (ko) * 1985-07-29 1990-05-21 오르토 파마슈티컬 코포레이션 2-아실-3,4-디알콕시아닐린의 제조방법
JPH0747582B2 (ja) * 1989-12-11 1995-05-24 杏林製薬株式会社 キナゾリン―3―アルカン酸誘導体とその塩およびその製造法
AU6870600A (en) * 1999-09-06 2001-04-10 Takeda Chemical Industries Ltd. Process for the preparation of 2,3-dihydroazepine compounds
EP2147679B1 (en) 2001-07-25 2014-06-25 Raptor Pharmaceutical, Inc. Compositions for blood-brain barrier transport
WO2006116718A2 (en) 2005-04-28 2006-11-02 Proteus Biomedical, Inc. Pharma-informatics system
US8795627B2 (en) 2007-03-21 2014-08-05 Raptor Pharmaceuticals Inc. Treatment of liver disorders by administration of RAP conjugates
JP5564517B2 (ja) 2009-02-20 2014-07-30 ティーオー − ビービービー ホールディング ベスローテン フェンノートシャップ グルタチオンをベースとする薬物送達システム
CN102458374A (zh) 2009-05-06 2012-05-16 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其使用方法
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143588A (da) * 1965-05-06
US4202895A (en) * 1971-06-04 1980-05-13 Sumitomo Chemical Company, Limited 1-Polyhaloalkyl-2(1H)-quinazolinone derivatives
US4146717A (en) * 1972-04-07 1979-03-27 Sumitomo Chemical Company, Limited Nitroquinazolinone compounds having antiviral properties
JPS555506B2 (da) * 1972-09-07 1980-02-07
US3983120A (en) * 1974-11-06 1976-09-28 Bristol-Myers Company Process for the preparation of optionally substituted 1,2,3,5-tetrahydroimidazo[2,1-b]quinazolin-2-ones
US3988340A (en) * 1975-01-23 1976-10-26 Bristol-Myers Company 6-Alkoxymethyl-1,2,3,5-tetrahydroimidazo[2,1-b]quinazolin-2-ones and 7-alkoxymethyl-6-[H]-1,2,3,4-tetrahydropyrimido[2,1-b]quinazolin-2-ones
JPS5795966A (en) * 1980-12-04 1982-06-15 Sumitomo Chem Co Ltd Novel 2(1h)-quinazolinone derivative
US4490374A (en) * 1982-09-30 1984-12-25 Ortho Pharmaceutical Corporation 5,6-Dialkoxy-3,4-optionally substituted-2(1H)quinazolinones, composition and method of use

Also Published As

Publication number Publication date
DK468184A (da) 1985-03-30
EP0138492A2 (en) 1985-04-24
US4556739A (en) 1985-12-03
AU565001B2 (en) 1987-09-03
EP0138492A3 (en) 1986-01-02
KR850002260A (ko) 1985-05-10
AU3371584A (en) 1985-04-18
GR80505B (en) 1985-01-30
KR900001200B1 (ko) 1990-02-28
NO843908L (no) 1985-04-01

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Legal Events

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AHB Application shelved due to non-payment