DK4271674T6 - Carboxy-benzimidazol-forbindelser til modulering af glp-1r - Google Patents

Carboxy-benzimidazol-forbindelser til modulering af glp-1r

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Publication number
DK4271674T6
DK4271674T6 DK22723850.8T DK22723850T DK4271674T6 DK 4271674 T6 DK4271674 T6 DK 4271674T6 DK 22723850 T DK22723850 T DK 22723850T DK 4271674 T6 DK4271674 T6 DK 4271674T6
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DK
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Prior art keywords
glp
carboxy
modulation
benzimidazole compounds
benzimidazole
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Application number
DK22723850.8T
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Danish (da)
English (en)
Other versions
DK4271674T3 (da
Inventor
Megan K Armstrong
Gediminas J Brizgys
James S Cassidy
Elbert Chin
Chienhung Chou
Chao-I Hung
David W Lin
Michael L Mitchell
Ezra Roberts
Scott D Schroeder
James G Taylor
Rhiannon Thomas-Tran
Nathan E Wright
Zheng-Yu Yang
Original Assignee
Gilead Sciences Inc
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Publication of DK4271674T3 publication Critical patent/DK4271674T3/da
Publication of DK4271674T6 publication Critical patent/DK4271674T6/da

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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
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EP4247804A1 (en) 2020-11-20 2023-09-27 Gilead Sciences, Inc. Polyheterocyclic glp-1 r modulating compounds
WO2022192428A1 (en) 2021-03-11 2022-09-15 Gilead Sciences, Inc. Glp-1r modulating compounds
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IL306110A (en) 2021-04-21 2023-11-01 Gilead Sciences Inc Carboxy-benzimidazole glp-1r modulating compounds
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WO2023111144A1 (en) 2021-12-16 2023-06-22 Astrazeneca Ab Certain 3-azabicyclo[3.1.0]hexanes as glp-1 receptor modulators
US20250042882A1 (en) 2021-12-16 2025-02-06 Astrazeneca Ab Certain 3-azabicyclo[3.1.0]hexanes as glp-1 receptor modulators
EP4592285A1 (en) 2022-09-22 2025-07-30 Shionogi & Co., Ltd. Fused ring compound having glp-1 receptor agonist effect
WO2024102625A1 (en) 2022-11-11 2024-05-16 Eli Lilly And Company Glucagon-like peptide 1 receptor agonists
KR20250085816A (ko) 2022-11-16 2025-06-12 일라이 릴리 앤드 캄파니 글루카곤-유사 펩티드 1 수용체 효능제
CN118496200A (zh) * 2023-02-14 2024-08-16 成都康弘药业集团股份有限公司 吲唑啉酮类化合物及其制备方法和用途
EP4731245A1 (en) * 2023-06-23 2026-04-29 Merck Sharp & Dohme LLC Use of a long-acting oxyntomodulin derivative for treament of fatty liver disease
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TW202521534A (zh) 2023-11-24 2025-06-01 香港商歌禮製藥(中國)有限公司 Glp-1r 激動劑及其治療方法
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