DK417785D0 - 3,4-dihydro-2(lh)-pyridon- og 2(lh)-pyridonderivater samt fremgangsmaade til fremstilling deraf - Google Patents

3,4-dihydro-2(lh)-pyridon- og 2(lh)-pyridonderivater samt fremgangsmaade til fremstilling deraf

Info

Publication number
DK417785D0
DK417785D0 DK417785A DK417785A DK417785D0 DK 417785 D0 DK417785 D0 DK 417785D0 DK 417785 A DK417785 A DK 417785A DK 417785 A DK417785 A DK 417785A DK 417785 D0 DK417785 D0 DK 417785D0
Authority
DK
Denmark
Prior art keywords
pyridon
dihydro
procedures
preparing
pyridone derivatives
Prior art date
Application number
DK417785A
Other languages
English (en)
Other versions
DK417785A (da
Inventor
Gerd Hilboll
Ille-Stephanie Doppelfeld
Gerrit Prop
Original Assignee
Nattermann A & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nattermann A & Cie filed Critical Nattermann A & Cie
Publication of DK417785D0 publication Critical patent/DK417785D0/da
Publication of DK417785A publication Critical patent/DK417785A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hospice & Palliative Care (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cosmetics (AREA)
DK417785A 1984-09-15 1985-09-13 3,4-dihydro-2(lh)-pyridon- og 2(lh)-pyridonderivater samt fremgangsmaade til fremstilling deraf DK417785A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843433953 DE3433953A1 (de) 1984-09-15 1984-09-15 Neue, eine imidazol-gruppe enthaltende 3,4-dihydro-2(1h)-pyridone und2(1h)-pyridone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
DK417785D0 true DK417785D0 (da) 1985-09-13
DK417785A DK417785A (da) 1986-03-16

Family

ID=6245507

Family Applications (1)

Application Number Title Priority Date Filing Date
DK417785A DK417785A (da) 1984-09-15 1985-09-13 3,4-dihydro-2(lh)-pyridon- og 2(lh)-pyridonderivater samt fremgangsmaade til fremstilling deraf

Country Status (10)

Country Link
US (1) US4699914A (da)
EP (1) EP0175187B1 (da)
JP (1) JPS6172781A (da)
AT (1) ATE49408T1 (da)
DE (2) DE3433953A1 (da)
DK (1) DK417785A (da)
ES (2) ES8705424A1 (da)
GR (1) GR852181B (da)
PT (1) PT81128B (da)
ZA (1) ZA857059B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4743608A (en) * 1986-07-15 1988-05-10 Rorer Pharmaceutical Corporation Pyridone-pyridyl-imidazolyl and triazolyl compounds and their use as cardiotonic agents
US4708958A (en) * 1986-09-24 1987-11-24 G. D. Searle & Co. 6-(imidazolyphenyl)-4-iminopyrimidinones useful as hypotensive agents
US4737511A (en) * 1986-11-03 1988-04-12 Schering A.G. Cardiotonic imidazolylphenylpyrrol-2-ones
EP0891360A4 (en) * 1996-04-03 2002-05-15 Merck & Co Inc FARNESYL PROTEIN TRANSFERASE INHIBITORS
US6001835A (en) * 1996-04-03 1999-12-14 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
DE19627310A1 (de) * 1996-06-27 1998-01-02 Schering Ag Imidazolderivate als Stickstoffmonoxid-Synthase-Inhibitoren
KR100388790B1 (ko) * 1998-03-06 2003-10-04 주식회사 엘지생명과학 파네실전이효소저해제로서유용한피리딘-2-온유도체
PE20060285A1 (es) 2004-03-30 2006-05-08 Aventis Pharma Inc Piridonas sustituidas como inhibidores de pol(adp-ribosa)-polimerasa (parp)
BRPI0518096A (pt) * 2004-12-01 2008-10-28 Kalypsys Inc composto, composição farmacêutica, uso de um composto para a preparação de um medicamento para o tratamento de uma condição resultante de uma anormalidade na produção de óxido nìtrico, uso de um composto para a preparação de um medicamento para o tratamento da dor em um indivìduo com necessidade do mesmo e uso de um composto para a preparação de um medicamento para o tratamento de inibição da dimerização de inos
CN101454317A (zh) * 2005-11-28 2009-06-10 凯利普西斯公司 作为一氧化氮合酶二聚化抑制剂的咪唑衍生物
BR112014031068A2 (pt) * 2012-06-12 2017-06-27 Abbvie Inc derivados piridinona e piridazinona

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE790106A (fr) * 1971-10-14 1973-04-13 Basf Ag Dihydropyridazones, leur preparation et leurs utilisations therapeutiques
DE3016874A1 (de) * 1980-05-02 1981-11-05 Bayer Ag, 5090 Leverkusen Substituierte 2-amino-3,4-dihydropyridinderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
IL69407A (en) * 1982-08-23 1987-10-20 Warner Lambert Co 2(1h)-pyridinones,their preparation and pharmaceutical compositions containing them
US4503061A (en) * 1983-07-22 1985-03-05 Warner-Lambert Company Substituted phenyl-pyridinones as cardiotonic agents
IL70169A0 (en) * 1982-11-18 1984-02-29 Sterling Drug Inc 2(1h)-pyridinones,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EP0175187A1 (de) 1986-03-26
DE3575300D1 (de) 1990-02-15
DE3433953A1 (de) 1986-03-27
ES554634A0 (es) 1987-04-16
ATE49408T1 (de) 1990-01-15
ES546965A0 (es) 1987-05-01
ES8704927A1 (es) 1987-04-16
PT81128A (en) 1985-10-01
ES8705424A1 (es) 1987-05-01
PT81128B (pt) 1987-10-20
EP0175187B1 (de) 1990-01-10
GR852181B (da) 1986-01-10
DK417785A (da) 1986-03-16
ZA857059B (en) 1986-04-30
JPS6172781A (ja) 1986-04-14
US4699914A (en) 1987-10-13

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment