DK303178A - Benzylpyrimidiner samt fremgangsmaade til fremstilling deraf - Google Patents

Benzylpyrimidiner samt fremgangsmaade til fremstilling deraf

Info

Publication number
DK303178A
DK303178A DK783031A DK303178A DK303178A DK 303178 A DK303178 A DK 303178A DK 783031 A DK783031 A DK 783031A DK 303178 A DK303178 A DK 303178A DK 303178 A DK303178 A DK 303178A
Authority
DK
Denmark
Prior art keywords
benzylpyrimidines
procedures
preparation
Prior art date
Application number
DK783031A
Other languages
English (en)
Other versions
DK142578C (da
DK142578B (da
Inventor
K Gutsche
P Scharwaechter
W Kohlmann
G Kromemer
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of DK303178A publication Critical patent/DK303178A/da
Publication of DK142578B publication Critical patent/DK142578B/da
Application granted granted Critical
Publication of DK142578C publication Critical patent/DK142578C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK303178A 1977-07-06 1978-07-05 Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf DK142578C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19772730467 DE2730467A1 (de) 1977-07-06 1977-07-06 Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2730467 1977-07-06

Publications (3)

Publication Number Publication Date
DK303178A true DK303178A (da) 1979-01-07
DK142578B DK142578B (da) 1980-11-24
DK142578C DK142578C (da) 1981-07-20

Family

ID=6013252

Family Applications (1)

Application Number Title Priority Date Filing Date
DK303178A DK142578C (da) 1977-07-06 1978-07-05 Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf

Country Status (17)

Country Link
US (1) US4279899A (da)
EP (1) EP0000334B1 (da)
JP (1) JPS5416482A (da)
AR (1) AR223465A1 (da)
AT (1) AT361931B (da)
AU (1) AU515661B2 (da)
CA (1) CA1102324A (da)
DE (2) DE2730467A1 (da)
DK (1) DK142578C (da)
FI (1) FI782173A7 (da)
HU (1) HU179407B (da)
IE (1) IE781308L (da)
IL (1) IL55018A (da)
IN (1) IN149577B (da)
IT (1) IT7825220A0 (da)
NO (1) NO782340L (da)
ZA (1) ZA783873B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4438267A (en) * 1980-11-11 1984-03-20 Daluge Susan M Monoheteroring compounds and their use
DE3045720A1 (de) * 1980-12-04 1982-07-08 Basf Ag, 6700 Ludwigshafen N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
HU186413B (en) * 1981-06-26 1985-07-29 Egyt Gyogyszervegyeszeti Gyar Process for producing 2,4-diamino-5-bracket-3-comma above,4-comma above,5-comma above-trimethoxy-benzyl-bracket closed-pyrimidine
HU187370B (en) * 1981-06-26 1985-12-28 Egyt Gyogyszervegyeszeti Gyar Improved process for producing 2,4-diamino-5-bracket-3-comma above, 4-comma above,5-comma above-trimethoxy-benzyl-bracket closed-pyrimidine
EP2090571B1 (de) * 2001-10-17 2012-05-16 Boehringer Ingelheim Pharma GmbH & Co. KG Pyrimidinderivate, Arzneimittel enthaltend diese Verbindungen, deren Verwendung und Verfahren zu ihrer Herstellung
AR081626A1 (es) 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
AR081331A1 (es) * 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3049544A (en) * 1962-08-14 Method for the preparation of
US2723975A (en) * 1952-04-03 1955-11-15 Nepera Chemical Co Inc 2, 4-di-piperidino-5-benzylpyrimidine
US2649449A (en) * 1952-04-04 1953-08-18 Nepera Chemical Co Inc 2-cyclohexylamino-4-amino-5-benzylpyrimidine
CH376115A (de) * 1957-12-06 1964-03-31 Ciba Geigy Verfahren zur Herstellung neuer substituierter Pyrimidine
US3515783A (en) 1967-10-20 1970-06-02 Hoffmann La Roche Antibacterial composition containing 5-methyl - 3 - sulfanilamidoisoxazole and trimethoxybenzyl pyrimidine
US4115650A (en) * 1976-11-17 1978-09-19 Hoffmann-La Roche Inc. Process for preparing 2,4-diamino-5-(substituted benzyl)-pyrimidines

Also Published As

Publication number Publication date
JPS5416482A (en) 1979-02-07
DE2730467A1 (de) 1979-01-18
DK142578C (da) 1981-07-20
IL55018A (en) 1983-03-31
NO782340L (no) 1979-01-09
DK142578B (da) 1980-11-24
CA1102324A (en) 1981-06-02
US4279899A (en) 1981-07-21
IT7825220A0 (it) 1978-06-30
IE781308L (en) 1979-01-06
IN149577B (da) 1982-01-30
AT361931B (de) 1981-04-10
DE2860928D1 (en) 1981-11-12
HU179407B (en) 1982-10-28
ATA487478A (de) 1980-09-15
AU515661B2 (en) 1981-04-16
FI782173A7 (fi) 1979-01-07
IL55018A0 (en) 1978-08-31
EP0000334A1 (de) 1979-01-24
AU3764478A (en) 1980-01-03
ZA783873B (en) 1979-08-29
EP0000334B1 (de) 1981-08-12
AR223465A1 (es) 1981-08-31

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