DK2650274T3 - Thionyleringsfremgangsmåde og et thionyleringsmiddel - Google Patents

Thionyleringsfremgangsmåde og et thionyleringsmiddel Download PDF

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DK2650274T3
DK2650274T3 DK13175186.9T DK13175186T DK2650274T3 DK 2650274 T3 DK2650274 T3 DK 2650274T3 DK 13175186 T DK13175186 T DK 13175186T DK 2650274 T3 DK2650274 T3 DK 2650274T3
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thionylation
thionylating
agent
thionylating agent
thionylation process
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DK13175186.9T
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Danish (da)
English (en)
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Birgitta Pettersson
Per H Svensson
Vedran Hasimbegovic
Jan Bergman
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Vironova Thionation Ab
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
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    • C07F9/58—Pyridine rings
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    • C07C327/40—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/34—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D309/36—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C07D311/82—Xanthenes
    • C07D311/84—Xanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D341/00—Heterocyclic compounds containing rings having three or more sulfur atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/36—Sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Detergent Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Lubricants (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
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US9520617B2 (en) 2013-03-14 2016-12-13 Advanced Technology Materials, Inc. Sulfolane mixtures as ambient aprotic polar solvents
CN103641834B (zh) * 2013-12-12 2015-12-09 沈阳药科大学 吡咯并苯并二氮杂*类化合物及其制备方法和应用
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EP2650274B1 (en) 2019-05-01
EP2569263B1 (en) 2013-11-13
ES2445024T3 (es) 2014-02-27
CA2825257C (en) 2020-01-07
BR112013019821A2 (pt) 2020-08-18
JP5989674B2 (ja) 2016-09-07
KR20140042789A (ko) 2014-04-07
HUE044332T2 (hu) 2019-10-28
AU2012213417A1 (en) 2013-04-04
EP2569263A1 (en) 2013-03-20
DK2569263T3 (da) 2014-02-10
US20130303767A1 (en) 2013-11-14
US20130102774A1 (en) 2013-04-25
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PL2569263T3 (pl) 2014-04-30
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RU2605412C2 (ru) 2016-12-20
US9115158B2 (en) 2015-08-25
CN104829405A (zh) 2015-08-12
SMT201400054B (it) 2014-07-07
JP2014510043A (ja) 2014-04-24
RS53186B (sr) 2014-06-30
EP2650274A3 (en) 2013-12-18
US9221855B2 (en) 2015-12-29
PT2569263E (pt) 2014-02-05
AU2012213417B2 (en) 2015-05-07
BR112013019821B1 (pt) 2021-04-20
KR101978703B1 (ko) 2019-05-15
HK1183474A1 (en) 2013-12-27
ES2737680T3 (es) 2020-01-15
EP2484655A1 (en) 2012-08-08
CY1115067T1 (el) 2016-12-14
EP2650274A2 (en) 2013-10-16
CN103153917A (zh) 2013-06-12
SI2569263T1 (sl) 2014-03-31
RU2013140771A (ru) 2015-03-10

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