DK236877A - PROCEDURE FOR THE PREPARATION OF 17BETA ESTERS OF TESTOSTERONE AND 5ALFA-DIHYDROTESTOSTERONE - Google Patents

PROCEDURE FOR THE PREPARATION OF 17BETA ESTERS OF TESTOSTERONE AND 5ALFA-DIHYDROTESTOSTERONE

Info

Publication number
DK236877A
DK236877A DK236877A DK236877A DK236877A DK 236877 A DK236877 A DK 236877A DK 236877 A DK236877 A DK 236877A DK 236877 A DK236877 A DK 236877A DK 236877 A DK236877 A DK 236877A
Authority
DK
Denmark
Prior art keywords
5alfa
17beta
dihydrotestosterone
testosterone
esters
Prior art date
Application number
DK236877A
Other languages
Danish (da)
Other versions
DK146096B (en
DK146096C (en
Inventor
J Vies
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/691,103 external-priority patent/US4098802A/en
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of DK236877A publication Critical patent/DK236877A/en
Publication of DK146096B publication Critical patent/DK146096B/en
Application granted granted Critical
Publication of DK146096C publication Critical patent/DK146096C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0025Esters

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK236877A 1976-05-28 1977-05-27 METHOD OF ANALOGUE FOR THE PREPARATION OF 17BETA ESTERS OF TESTOSTERON DK146096C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/691,103 US4098802A (en) 1975-02-18 1976-05-28 Oral pharmaceutical preparation having androgenic activity
US69110376 1976-05-28

Publications (3)

Publication Number Publication Date
DK236877A true DK236877A (en) 1977-11-29
DK146096B DK146096B (en) 1983-06-27
DK146096C DK146096C (en) 1983-11-21

Family

ID=24775172

Family Applications (1)

Application Number Title Priority Date Filing Date
DK236877A DK146096C (en) 1976-05-28 1977-05-27 METHOD OF ANALOGUE FOR THE PREPARATION OF 17BETA ESTERS OF TESTOSTERON

Country Status (12)

Country Link
JP (1) JPS52148060A (en)
AR (1) AR214323A1 (en)
BE (1) BE855163A (en)
CH (1) CH627761A5 (en)
DE (1) DE2723876C2 (en)
DK (1) DK146096C (en)
ES (1) ES459230A1 (en)
FI (1) FI57597C (en)
FR (1) FR2352832A1 (en)
GB (1) GB1567515A (en)
NL (1) NL7705790A (en)
SE (1) SE425493B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2253423T3 (en) * 2000-08-23 2006-06-01 Akzo Nobel N.V. FORMULATION OF A TESTOSTERONE ESTER FOR HUMAN USE.
JO2505B1 (en) 2003-03-14 2009-10-05 باير شيرنغ فارما اكتنجيسيلشافت method and pharmaceutical compositions for reliable achievements of acceptable serum testosterone levels
GB0807605D0 (en) * 2008-04-28 2008-06-04 Diurnal Ltd Lipid composition
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US9034858B2 (en) 2010-11-30 2015-05-19 Lipocine Inc. High-strength testosterone undecanoate compositions
US20120148675A1 (en) 2010-12-10 2012-06-14 Basawaraj Chickmath Testosterone undecanoate compositions
TW201521731A (en) * 2013-03-15 2015-06-16 利波辛股份有限公司 Lipobalanced long chain testosterone esters for oral delivery
EP3544614A4 (en) 2016-11-28 2020-08-05 Lipocine Inc. Oral testosterone undecanoate therapy

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL189235C (en) * 1974-02-28 1993-02-16 Akzo Nv METHOD FOR THE PREPARATION OF AN ORAL PHARMACEUTICAL PREPARATION WITH ANDROGENIC ACTION

Also Published As

Publication number Publication date
DE2723876A1 (en) 1977-12-15
SE425493B (en) 1982-10-04
GB1567515A (en) 1980-05-14
JPS52148060A (en) 1977-12-08
JPS6145637B2 (en) 1986-10-08
AR214323A1 (en) 1979-05-31
FI57597C (en) 1980-09-10
FI57597B (en) 1980-05-30
CH627761A5 (en) 1982-01-29
DE2723876C2 (en) 1986-10-30
NL7705790A (en) 1977-11-30
DK146096B (en) 1983-06-27
SE7706235L (en) 1977-11-29
ES459230A1 (en) 1978-11-16
BE855163A (en) 1977-11-28
FR2352832B1 (en) 1980-07-11
DK146096C (en) 1983-11-21
FR2352832A1 (en) 1977-12-23
FI771684A (en) 1977-11-29

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Legal Events

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