DK152049C - Analogifremgangsmaade til fremstilling af monoacyl-derivater af c-076 makrolider - Google Patents
Analogifremgangsmaade til fremstilling af monoacyl-derivater af c-076 makroliderInfo
- Publication number
- DK152049C DK152049C DK434478A DK434478A DK152049C DK 152049 C DK152049 C DK 152049C DK 434478 A DK434478 A DK 434478A DK 434478 A DK434478 A DK 434478A DK 152049 C DK152049 C DK 152049C
- Authority
- DK
- Denmark
- Prior art keywords
- macrolides
- preparing
- analogy procedure
- monoacyl derivatives
- monoacyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P17/00—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
- C12P17/18—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms containing at least two hetero rings condensed among themselves or condensed with a common carbocyclic ring system, e.g. rifamycin
- C12P17/181—Heterocyclic compounds containing oxygen atoms as the only ring heteroatoms in the condensed system, e.g. Salinomycin, Septamycin
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P19/00—Preparation of compounds containing saccharide radicals
- C12P19/44—Preparation of O-glycosides, e.g. glucosides
- C12P19/60—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
- C12P19/62—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
- C12P19/623—Avermectin; Milbemycin; Ivermectin; C-076
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Wood Science & Technology (AREA)
- General Health & Medical Sciences (AREA)
- Zoology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Microbiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Agronomy & Crop Science (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US83909977A | 1977-10-03 | 1977-10-03 | |
| US83860277A | 1977-10-03 | 1977-10-03 | |
| US83909977 | 1977-10-03 | ||
| US83860277 | 1977-10-03 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK434478A DK434478A (da) | 1979-04-04 |
| DK152049B DK152049B (da) | 1988-01-25 |
| DK152049C true DK152049C (da) | 1988-06-20 |
Family
ID=27126041
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK434478A DK152049C (da) | 1977-10-03 | 1978-10-02 | Analogifremgangsmaade til fremstilling af monoacyl-derivater af c-076 makrolider |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0001688B1 (da) |
| JP (1) | JPS5461197A (da) |
| AU (1) | AU519570B2 (da) |
| DE (1) | DE2861286D1 (da) |
| DK (1) | DK152049C (da) |
| IE (1) | IE47570B1 (da) |
| IT (1) | IT1157353B (da) |
| NZ (1) | NZ188459A (da) |
| OA (1) | OA06063A (da) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4203976A (en) * | 1978-08-02 | 1980-05-20 | Merck & Co., Inc. | Sugar derivatives of C-076 compounds |
| US4200581A (en) * | 1978-08-04 | 1980-04-29 | Merck & Co., Inc. | Alkyl derivatives of C-076 compounds |
| US4289760A (en) * | 1980-05-02 | 1981-09-15 | Merck & Co., Inc. | 23-Keto derivatives of C-076 compounds |
| US4285963A (en) * | 1980-08-07 | 1981-08-25 | Merck & Co., Inc. | Novel derivatives of C-076 compounds |
| US4412991A (en) * | 1981-08-28 | 1983-11-01 | Merck & Co., Inc. | 22-Hydroxy derivatives of C-076 compounds, pharmaceutical compositions and method of use |
| US4427663A (en) * | 1982-03-16 | 1984-01-24 | Merck & Co., Inc. | 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof |
| US4846789A (en) * | 1982-07-19 | 1989-07-11 | L. S. Van Landingham, Jr. | Combatting internal parasites in warm blooded animals |
| US4469682A (en) * | 1983-01-28 | 1984-09-04 | Merck & Co., Inc. | Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use |
| JPS60126289A (ja) * | 1983-11-14 | 1985-07-05 | Sankyo Co Ltd | ミルベマイシン類の５−カ−ボネ−ト誘導体 |
| GB2168345B (en) * | 1984-12-14 | 1988-05-25 | Ciba Geigy Ag | Pesticidal 13b-substituted milbemycin derivatives |
| ES8605582A1 (es) * | 1985-12-11 | 1986-03-16 | Antibioticos Sa | Un procedimiento para la preparacion de avermectinas |
| JPH0819133B2 (ja) * | 1986-03-25 | 1996-02-28 | 三共株式会社 | １３−置換ミルベマイシン類の５−オキシム誘導体 |
| RU2024527C1 (ru) * | 1986-03-25 | 1994-12-15 | Санкио Компани Лимитед | Способ получения макролидных соединений |
| EP0240274A3 (en) * | 1986-04-03 | 1990-03-14 | Merck & Co. Inc. | Avermectins as growth promotant agents |
| JPS6333341A (ja) * | 1986-07-28 | 1988-02-13 | Seitetsu Kagaku Co Ltd | 配糖体の処理方法 |
| IN167980B (da) * | 1987-01-23 | 1991-01-19 | Pfizer | |
| US4895837A (en) * | 1988-01-29 | 1990-01-23 | Merck & Co., Inc. | Avermectin derivatives |
| US5387395A (en) * | 1992-07-06 | 1995-02-07 | Beckman Instruments, Inc. | Fluid distribution manifold |
| DE69310539T2 (de) * | 1992-11-20 | 1998-01-15 | British Tech Group | Bildrekonstruktion |
| US5380838A (en) * | 1993-10-08 | 1995-01-10 | Merck & Co. Inc. | Stable solvates of avermectin compounds |
| WO1997046204A2 (en) | 1996-06-05 | 1997-12-11 | Ashmont Holdings Limited | Injectable compositions |
| AU5261301A (en) | 2000-04-27 | 2001-11-12 | Sankyo Co | 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests |
| CR6574A (es) | 2001-02-27 | 2004-10-28 | Syngenta Participations Ag | Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas |
| EG23124A (en) | 2001-02-27 | 2004-04-28 | Syngenta Participations Ag | Avermectins substituted in the 4-position having pesticidal properties |
| AR036486A1 (es) | 2001-08-28 | 2004-09-15 | Syngenta Participations Ag | Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion |
| AR040073A1 (es) | 2002-05-07 | 2005-03-16 | Syngenta Participations Ag | Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas |
| US7001889B2 (en) | 2002-06-21 | 2006-02-21 | Merial Limited | Anthelmintic oral homogeneous veterinary pastes |
| GB0302308D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties |
| GB0302310D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties |
| GB0320176D0 (en) | 2003-08-28 | 2003-10-01 | Syngenta Participations Ag | Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties |
| DE102007007750A1 (de) | 2006-08-17 | 2008-02-21 | Bayer Cropscience Ag | Avermectinderivate |
| JP2010006703A (ja) * | 2006-11-07 | 2010-01-14 | Hokko Chem Ind Co Ltd | アベルメクチンモノ配糖体誘導体 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4914624A (da) * | 1972-06-08 | 1974-02-08 | ||
| JPS5645890B2 (da) * | 1973-05-29 | 1981-10-29 | ||
| SE434277B (sv) * | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
-
1978
- 1978-09-20 NZ NZ188459A patent/NZ188459A/xx unknown
- 1978-09-22 AU AU40089/78A patent/AU519570B2/en not_active Expired
- 1978-09-29 IT IT51320/78A patent/IT1157353B/it active
- 1978-09-29 EP EP78300435A patent/EP0001688B1/en not_active Expired
- 1978-09-29 DE DE7878300435T patent/DE2861286D1/de not_active Expired
- 1978-10-02 DK DK434478A patent/DK152049C/da not_active IP Right Cessation
- 1978-10-02 IE IE1964/78A patent/IE47570B1/en not_active IP Right Cessation
- 1978-10-03 OA OA56623A patent/OA06063A/xx unknown
- 1978-10-03 JP JP12128378A patent/JPS5461197A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| OA06063A (fr) | 1981-06-30 |
| NZ188459A (en) | 1982-09-07 |
| EP0001688A1 (en) | 1979-05-02 |
| IT7851320A0 (it) | 1978-09-29 |
| DE2861286D1 (en) | 1982-01-14 |
| AU519570B2 (en) | 1981-12-10 |
| AU4008978A (en) | 1980-03-27 |
| IE47570B1 (en) | 1984-05-02 |
| JPS5461197A (en) | 1979-05-17 |
| JPS6254113B2 (da) | 1987-11-13 |
| IT1157353B (it) | 1987-02-11 |
| DK152049B (da) | 1988-01-25 |
| IE781964L (en) | 1979-04-03 |
| DK434478A (da) | 1979-04-04 |
| EP0001688B1 (en) | 1981-11-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |