DK149893C - Analogifremgangsmaade til fremstilling af thiazolderivater eller farmaceutisk acceptable salte deraf - Google Patents
Analogifremgangsmaade til fremstilling af thiazolderivater eller farmaceutisk acceptable salte derafInfo
- Publication number
- DK149893C DK149893C DK452273A DK452273A DK149893C DK 149893 C DK149893 C DK 149893C DK 452273 A DK452273 A DK 452273A DK 452273 A DK452273 A DK 452273A DK 149893 C DK149893 C DK 149893C
- Authority
- DK
- Denmark
- Prior art keywords
- thiazold
- analogue
- derivatives
- preparation
- acceptable salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8257472 | 1972-08-17 | ||
JP47082574A JPS5238559B2 (xx) | 1972-08-17 | 1972-08-17 | |
JP48039354A JPS49125359A (xx) | 1973-04-05 | 1973-04-05 | |
JP3935473 | 1973-04-05 | ||
ZA00741280A ZA741280B (en) | 1972-08-17 | 1974-02-26 | Thiazole derivatives |
ZA7401280 | 1974-02-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
DK149893B DK149893B (da) | 1986-10-20 |
DK149893C true DK149893C (da) | 1987-04-21 |
Family
ID=27290112
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK452273A DK149893C (da) | 1972-08-17 | 1973-08-16 | Analogifremgangsmaade til fremstilling af thiazolderivater eller farmaceutisk acceptable salte deraf |
Country Status (10)
Country | Link |
---|---|
US (1) | US3932400A (xx) |
CA (1) | CA991640A (xx) |
CH (1) | CH581640A5 (xx) |
DE (1) | DE2341753C2 (xx) |
DK (1) | DK149893C (xx) |
FR (1) | FR2196162B1 (xx) |
GB (1) | GB1435139A (xx) |
NL (1) | NL179733C (xx) |
SE (1) | SE421615B (xx) |
ZA (1) | ZA741280B (xx) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4001421A (en) * | 1971-10-27 | 1977-01-04 | Syntex (U.S.A.) Inc. | Thiazole cardiovascular agents |
US4119718A (en) * | 1977-05-02 | 1978-10-10 | Merck & Co., Inc. | 3-Amino-2-oxy-propoxy-substituted isothiazoles |
US4260609A (en) * | 1977-06-01 | 1981-04-07 | Merck & Co., Inc. | Di- and tri- substituted thiazoles |
US4259341A (en) * | 1977-06-01 | 1981-03-31 | Merck & Co., Inc. | Di- and tri-substituted thiazoles |
US4396625A (en) * | 1980-05-13 | 1983-08-02 | Sumitomo Chemical Company, Limited | Treatment of glaucoma or ocular hypertension and ophthalmic composition |
US4670450A (en) * | 1985-11-13 | 1987-06-02 | Merrell Dow Pharmaceuticals Inc. | Cardiotonic thiazolones |
ES2362998T3 (es) | 2002-08-19 | 2011-07-18 | Pfizer Inc. | Terapia de combinación para enfermedades hiperproliferativas. |
GEP20084406B (en) * | 2003-05-30 | 2008-06-25 | Ranbaxy Lab Ltd | Substituted pyrrole derivatives and their use as hmg-co inhibitors |
US20050037063A1 (en) * | 2003-07-21 | 2005-02-17 | Bolton Anthony E. | Combined therapies |
US20060063803A1 (en) * | 2004-09-23 | 2006-03-23 | Pfizer Inc | 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds |
AU2005308575A1 (en) * | 2004-11-23 | 2006-06-01 | Warner-Lambert Company Llc | 7-(2h-pyrazol-3-yl)-3, 5-dihyroxy-heptanoic acid derivatives as HMG Co-A reductase inhibitors for the treatment of lipidemia |
GT200600381A (es) | 2005-08-25 | 2007-03-28 | Compuestos organicos | |
US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
AU2006313430B2 (en) * | 2005-11-08 | 2012-09-06 | Ranbaxy Laboratories Limited | Process for (3R,5R)-7-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4- [(4-hydroxy methyl phenyl amino) carbonyl]-pyrrol-1-yl]-3, 5-dihydroxy-heptanoic acid hemi calcium salt |
WO2007086980A2 (en) * | 2005-11-10 | 2007-08-02 | Duke University | Methods of determining the risk of developing coronary artery disease |
US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
CA2636077C (en) * | 2006-01-18 | 2012-01-03 | Amgen Inc. | Thiazole compounds as protein kinase b (pkb) inhibitors |
US8383660B2 (en) | 2006-03-10 | 2013-02-26 | Pfizer Inc. | Dibenzyl amine compounds and derivatives |
US7919506B2 (en) | 2006-03-10 | 2011-04-05 | Pfizer Inc. | Dibenzyl amine compounds and derivatives |
AR059838A1 (es) * | 2006-03-14 | 2008-04-30 | Ranbaxy Lab Ltd | Formulaciones para dosis estabilizantes de estatina |
CN101494980A (zh) * | 2006-07-14 | 2009-07-29 | 兰贝克赛实验室有限公司 | HMG-CoA还原酶抑制剂的多晶型形式及其应用 |
US8404896B2 (en) | 2006-12-01 | 2013-03-26 | Bristol-Myers Squibb Company | N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
WO2009011871A2 (en) * | 2007-07-17 | 2009-01-22 | Amgen Inc. | Thiadiazole modulators of pkb |
AU2014255381A1 (en) | 2013-04-17 | 2015-10-08 | Pfizer Inc. | N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases |
WO2016055901A1 (en) | 2014-10-08 | 2016-04-14 | Pfizer Inc. | Substituted amide compounds |
CN104530033B (zh) * | 2014-12-26 | 2017-07-07 | 江西百神药业股份有限公司 | 一种盐酸阿罗洛尔的制备工艺新方法 |
CN105646472A (zh) * | 2016-02-29 | 2016-06-08 | 山东齐都药业有限公司 | 一种盐酸阿罗洛尔的制备方法 |
MX2021008533A (es) | 2019-01-18 | 2021-08-19 | Astrazeneca Ab | Inhibidores de la pcsk9 y metodos de uso de los mismos. |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA599475A (en) * | 1960-06-07 | W. Harman Marion | Aminoethylthiazoles | |
US2221147A (en) * | 1938-11-18 | 1940-11-12 | Goodrich Co B F | Preparation of aminated esters of sulphydryl compounds |
US3228952A (en) * | 1962-06-27 | 1966-01-11 | Dow Chemical Co | Thiazole thioethers |
US3158623A (en) * | 1963-03-01 | 1964-11-24 | Abbott Lab | 5-nitro-2-furylthioamide |
BE790569A (fr) * | 1971-10-27 | 1973-04-26 | Syntex Corp | Agents cardiovasculaires a base de thiazoles |
-
1973
- 1973-08-14 GB GB3950573A patent/GB1435139A/en not_active Expired
- 1973-08-15 NL NLAANVRAGE7311248,A patent/NL179733C/xx not_active IP Right Cessation
- 1973-08-16 FR FR7329860A patent/FR2196162B1/fr not_active Expired
- 1973-08-16 DK DK452273A patent/DK149893C/da not_active IP Right Cessation
- 1973-08-16 US US05/389,517 patent/US3932400A/en not_active Expired - Lifetime
- 1973-08-16 CH CH1182373A patent/CH581640A5/xx not_active IP Right Cessation
- 1973-08-16 CA CA178,970A patent/CA991640A/en not_active Expired
- 1973-08-16 SE SE7311181A patent/SE421615B/xx unknown
- 1973-08-17 DE DE2341753A patent/DE2341753C2/de not_active Expired
-
1974
- 1974-02-26 ZA ZA00741280A patent/ZA741280B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
NL179733C (nl) | 1986-11-03 |
ZA741280B (en) | 1975-03-26 |
CA991640A (en) | 1976-06-22 |
DK149893B (da) | 1986-10-20 |
NL7311248A (xx) | 1974-02-19 |
US3932400A (en) | 1976-01-13 |
GB1435139A (en) | 1976-05-12 |
AU5928173A (en) | 1975-02-20 |
DE2341753C2 (de) | 1982-12-09 |
SE421615B (sv) | 1982-01-18 |
FR2196162A1 (xx) | 1974-03-15 |
FR2196162B1 (xx) | 1977-01-28 |
NL179733B (nl) | 1986-06-02 |
CH581640A5 (xx) | 1976-11-15 |
DE2341753A1 (de) | 1974-02-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUP | Patent expired |