DK148036C - METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS. - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS.

Info

Publication number
DK148036C
DK148036C DK51878A DK51878A DK148036C DK 148036 C DK148036 C DK 148036C DK 51878 A DK51878 A DK 51878A DK 51878 A DK51878 A DK 51878A DK 148036 C DK148036 C DK 148036C
Authority
DK
Denmark
Prior art keywords
epimere
analogue
amino
preparation
acid addition
Prior art date
Application number
DK51878A
Other languages
Danish (da)
Other versions
DK148036B (en
DK51878A (en
Inventor
Frank Christian Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/856,479 external-priority patent/US4150220A/en
Application filed by Pfizer filed Critical Pfizer
Publication of DK51878A publication Critical patent/DK51878A/en
Publication of DK148036B publication Critical patent/DK148036B/en
Application granted granted Critical
Publication of DK148036C publication Critical patent/DK148036C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
DK51878A 1977-02-04 1978-02-03 METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS. DK148036C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US76548077A 1977-02-04 1977-02-04
US76548077 1977-02-04
US85647977 1977-12-01
US05/856,479 US4150220A (en) 1977-02-04 1977-12-01 Semi-synthetic 4"-erythromycin A derivatives

Publications (3)

Publication Number Publication Date
DK51878A DK51878A (en) 1978-08-05
DK148036B DK148036B (en) 1985-02-11
DK148036C true DK148036C (en) 1985-07-15

Family

ID=27117613

Family Applications (1)

Application Number Title Priority Date Filing Date
DK51878A DK148036C (en) 1977-02-04 1978-02-03 METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS.

Country Status (30)

Country Link
JP (1) JPS5827798B2 (en)
AR (1) AR222147A1 (en)
AU (1) AU501298B1 (en)
BG (2) BG33159A3 (en)
CA (1) CA1106367A (en)
CH (1) CH628906A5 (en)
CS (1) CS221801B2 (en)
DD (1) DD140048A5 (en)
DE (1) DE2804507C2 (en)
DK (1) DK148036C (en)
ES (2) ES466057A1 (en)
FI (1) FI780354A (en)
FR (2) FR2379550A1 (en)
GB (2) GB1585315A (en)
GR (1) GR68691B (en)
HU (1) HU182559B (en)
IE (1) IE46661B1 (en)
IL (2) IL53968A0 (en)
IT (1) IT1094209B (en)
LU (1) LU79004A1 (en)
NL (1) NL176174C (en)
NO (2) NO146472C (en)
NZ (1) NZ186385A (en)
PH (2) PH14421A (en)
PL (1) PL116228B1 (en)
PT (1) PT67568B (en)
RO (4) RO79687A7 (en)
SE (2) SE445223B (en)
SU (1) SU927122A3 (en)
YU (3) YU40913B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4382085A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
HN1998000074A (en) * 1997-06-11 1999-01-08 Pfizer Prod Inc DERIVATIVES FROM MACROLIDES C-4 SUBSTITUTED
US6407074B1 (en) 1997-06-11 2002-06-18 Pfizer Inc C-4″-substituted macrolide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

Also Published As

Publication number Publication date
YU40913B (en) 1986-08-31
FR2379550A1 (en) 1978-09-01
BG33159A3 (en) 1982-12-15
AR222147A1 (en) 1981-04-30
NO146472B (en) 1982-06-28
ES466057A1 (en) 1978-10-01
IE46661B1 (en) 1983-08-24
FI780354A (en) 1978-08-05
YU227983A (en) 1984-04-30
IE780239L (en) 1978-08-04
RO77345A (en) 1981-08-17
NO780389L (en) 1978-08-07
DE2804507C2 (en) 1982-11-04
IL61997A0 (en) 1981-02-27
GB1585316A (en) 1981-02-25
PH16675A (en) 1983-12-13
PT67568B (en) 1979-06-18
AU501298B1 (en) 1979-06-14
RO79686A7 (en) 1982-08-17
CS221801B2 (en) 1983-04-29
JPS5827798B2 (en) 1983-06-11
NL176174B (en) 1984-10-01
DE2804507A1 (en) 1978-08-10
SE8300870D0 (en) 1983-02-16
IT1094209B (en) 1985-07-26
NL7801262A (en) 1978-08-08
YU26583A (en) 1984-02-29
DD140048A5 (en) 1980-02-06
SE8300870L (en) 1983-02-16
FR2379550B1 (en) 1980-07-04
ES472429A1 (en) 1979-04-01
NZ186385A (en) 1980-10-08
NO146472C (en) 1982-10-06
GR68691B (en) 1982-02-01
DK148036B (en) 1985-02-11
SE445223B (en) 1986-06-09
JPS53101337A (en) 1978-09-04
IT7820005A0 (en) 1978-02-03
NO811913L (en) 1978-08-07
SE457086B (en) 1988-11-28
NL176174C (en) 1985-03-01
RO79687A7 (en) 1982-08-17
NO150484C (en) 1984-10-24
GB1585315A (en) 1981-02-25
HU182559B (en) 1984-02-28
PL204428A1 (en) 1979-06-04
RO81622B (en) 1983-04-30
IL53968A0 (en) 1978-04-30
PL116228B1 (en) 1981-05-30
LU79004A1 (en) 1979-09-06
NO150484B (en) 1984-07-16
DK51878A (en) 1978-08-05
CH628906A5 (en) 1982-03-31
YU7378A (en) 1983-04-30
RO81622A (en) 1983-04-29
BG32718A3 (en) 1982-09-15
SE7800270L (en) 1978-08-05
SU927122A3 (en) 1982-05-07
PT67568A (en) 1978-02-01
CA1106367A (en) 1981-08-04
FR2385735B1 (en) 1980-10-24
PH14421A (en) 1981-07-10
YU40798B (en) 1986-06-30
FR2385735A1 (en) 1978-10-27
YU40799B (en) 1986-06-30

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