DK145577C - Analogifremgangsmaade til fremstilling af s-triazolo(4,3-a)-(1,4)-benzodiazepiner eller 5n-oxyder eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af s-triazolo(4,3-a)-(1,4)-benzodiazepiner eller 5n-oxyder eller syreadditionssalte deraf

Info

Publication number
DK145577C
DK145577C DK583669A DK583669A DK145577C DK 145577 C DK145577 C DK 145577C DK 583669 A DK583669 A DK 583669A DK 583669 A DK583669 A DK 583669A DK 145577 C DK145577 C DK 145577C
Authority
DK
Denmark
Prior art keywords
oxydes
benzodiazepines
triazolo
analogue
preparation
Prior art date
Application number
DK583669A
Other languages
Danish (da)
English (en)
Other versions
DK145577B (da
Inventor
K Meguro
Y Kuwada
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP9292968A external-priority patent/JPS4843754B1/ja
Priority claimed from JP9518768A external-priority patent/JPS4916436B1/ja
Priority claimed from JP1070269A external-priority patent/JPS4920596B1/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DK145577B publication Critical patent/DK145577B/da
Application granted granted Critical
Publication of DK145577C publication Critical patent/DK145577C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK583669A 1968-11-05 1969-11-05 Analogifremgangsmaade til fremstilling af s-triazolo(4,3-a)-(1,4)-benzodiazepiner eller 5n-oxyder eller syreadditionssalte deraf DK145577C (da)

Applications Claiming Priority (14)

Application Number Priority Date Filing Date Title
JP8081368 1968-11-05
JP8081368 1968-11-05
JP9292968A JPS4843754B1 (cg-RX-API-DMAC7.html) 1968-12-17 1968-12-17
JP9292868 1968-12-17
JP9293168 1968-12-17
JP9293068 1968-12-17
JP9292868 1968-12-17
JP9293068 1968-12-17
JP9293168 1968-12-17
JP9292968 1968-12-17
JP9518768A JPS4916436B1 (cg-RX-API-DMAC7.html) 1968-12-25 1968-12-25
JP9518768 1968-12-25
JP1070269A JPS4920596B1 (cg-RX-API-DMAC7.html) 1969-02-13 1969-02-13
JP1070269 1969-02-13

Publications (2)

Publication Number Publication Date
DK145577B DK145577B (da) 1982-12-13
DK145577C true DK145577C (da) 1983-05-16

Family

ID=27563558

Family Applications (1)

Application Number Title Priority Date Filing Date
DK583669A DK145577C (da) 1968-11-05 1969-11-05 Analogifremgangsmaade til fremstilling af s-triazolo(4,3-a)-(1,4)-benzodiazepiner eller 5n-oxyder eller syreadditionssalte deraf

Country Status (8)

Country Link
CH (1) CH532065A (cg-RX-API-DMAC7.html)
DK (1) DK145577C (cg-RX-API-DMAC7.html)
FI (1) FI50981C (cg-RX-API-DMAC7.html)
MY (1) MY7600024A (cg-RX-API-DMAC7.html)
NL (1) NL157601C (cg-RX-API-DMAC7.html)
NO (1) NO126325B (cg-RX-API-DMAC7.html)
PH (1) PH9315A (cg-RX-API-DMAC7.html)
YU (1) YU36178B (cg-RX-API-DMAC7.html)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE758921A (fr) * 1969-11-15 1971-04-16 Takeda Chemical Industries Ltd Derives de benzodiazepine
BE759099A (fr) * 1969-11-18 1971-04-30 Takeda Chemical Industries Ltd Procede de fabrication de composes heterocycliques
JPS494470B1 (cg-RX-API-DMAC7.html) * 1970-08-26 1974-02-01
JPS4932874B1 (cg-RX-API-DMAC7.html) * 1970-12-11 1974-09-03
US4250094A (en) * 1971-04-28 1981-02-10 The Upjohn Company 1-(Aminoalkyl) substituted-6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
US4902794A (en) * 1971-04-28 1990-02-20 The Upjohn Company Triazolo-benzodiazepines
US4141902A (en) * 1971-04-28 1979-02-27 The Upjohn Company 1-Halomethyl-6-phenyl-4H-s-[4,3-a][1,4]benzodiazepines
US3856802A (en) * 1971-05-10 1974-12-24 Upjohn Co 1,6-DISUBSTITUTED-4H-5-{8 4,3-a{9 BENZODIAZEPINES
US3870793A (en) * 1971-08-09 1975-03-11 Upjohn Co Animal feed and process
DE2356369C2 (de) * 1972-11-24 1984-08-23 The Upjohn Co., Kalamazoo, Mich. Pharmazeutisches Präparat, enthaltend eine oder mehrere Benzodiazepinverbindungen
US3864328A (en) * 1973-10-19 1975-02-04 Hoffmann La Roche 2-hydrazino benzodiazepine derivatives
JPS5747916B2 (cg-RX-API-DMAC7.html) 1974-05-13 1982-10-13
US4018788A (en) * 1975-06-16 1977-04-19 The Upjohn Company 6-(O-Halophenyl)-1-methyl-4H-s-triazolo[4,3-a][1,4]-benzodiazepine

Also Published As

Publication number Publication date
NL157601B (nl) 1978-08-15
YU275369A (en) 1981-06-30
FI50981B (cg-RX-API-DMAC7.html) 1976-05-31
DK145577B (da) 1982-12-13
MY7600024A (en) 1976-12-31
YU36178B (en) 1982-02-25
NL157601C (nl) 1982-04-16
FI50981C (fi) 1976-09-10
NO126325B (cg-RX-API-DMAC7.html) 1973-01-22
CH532065A (de) 1972-12-31
NL6916543A (cg-RX-API-DMAC7.html) 1970-05-08
PH9315A (en) 1975-08-22

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