DK144376C - Analogifremgangsmaade til fremstilling af bis-penicillanoyloxy-alkaner eller salte deraf - Google Patents

Analogifremgangsmaade til fremstilling af bis-penicillanoyloxy-alkaner eller salte deraf

Info

Publication number
DK144376C
DK144376C DK162177A DK162177A DK144376C DK 144376 C DK144376 C DK 144376C DK 162177 A DK162177 A DK 162177A DK 162177 A DK162177 A DK 162177A DK 144376 C DK144376 C DK 144376C
Authority
DK
Denmark
Prior art keywords
penicillanoyloxy
alkanes
analogue
salts
preparing bis
Prior art date
Application number
DK162177A
Other languages
Danish (da)
English (en)
Other versions
DK162177A (da
DK144376B (da
Inventor
K Hansen
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of DK162177A publication Critical patent/DK162177A/da
Publication of DK144376B publication Critical patent/DK144376B/da
Application granted granted Critical
Publication of DK144376C publication Critical patent/DK144376C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/20Spiro-condensed ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/06Seven-membered rings having the hetero atoms in positions 1 and 4 not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/06Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals
    • C07D295/067Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals with the ring nitrogen atoms and the substituents attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/194Radicals derived from thio- or thiono carboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK162177A 1976-04-15 1977-04-13 Analogifremgangsmaade til fremstilling af bis-penicillanoyloxy-alkaner eller salte deraf DK144376C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB15746/76A GB1579931A (en) 1976-04-15 1976-04-15 Bis-penicillanoyl-oxy-alkanes
GB1574676 1976-04-15

Publications (3)

Publication Number Publication Date
DK162177A DK162177A (da) 1977-10-16
DK144376B DK144376B (da) 1982-03-01
DK144376C true DK144376C (da) 1982-08-02

Family

ID=10064756

Family Applications (1)

Application Number Title Priority Date Filing Date
DK162177A DK144376C (da) 1976-04-15 1977-04-13 Analogifremgangsmaade til fremstilling af bis-penicillanoyloxy-alkaner eller salte deraf

Country Status (24)

Country Link
US (1) US4181659A (xx)
JP (1) JPS52128391A (xx)
AR (1) AR218870A1 (xx)
AT (1) AT353960B (xx)
AU (1) AU510825B2 (xx)
BE (1) BE853607A (xx)
CA (1) CA1112239A (xx)
DE (1) DE2716172C2 (xx)
DK (1) DK144376C (xx)
ES (1) ES457829A1 (xx)
FI (1) FI63759C (xx)
FR (1) FR2348217A1 (xx)
GB (1) GB1579931A (xx)
GR (1) GR63089B (xx)
IE (1) IE44809B1 (xx)
IT (1) IT1116735B (xx)
LU (1) LU77135A1 (xx)
NL (1) NL7704085A (xx)
NZ (1) NZ183756A (xx)
PH (1) PH14046A (xx)
PT (1) PT66434B (xx)
SE (1) SE425490B (xx)
YU (1) YU94277A (xx)
ZA (1) ZA771935B (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4407751A (en) * 1979-02-13 1983-10-04 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) Processes for preparing β-lactams
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
DE3051044C2 (xx) * 1979-06-19 1989-03-30 Leo Pharmaceutical Products Ltd. A/S (Loevens Kemiske Fabrik Produktionsaktieselskab), Ballerup, Dk
US4340539A (en) * 1980-01-21 1982-07-20 Bristol-Myers Company Derivatives of 6-bromo penicillanic acid
US4323499A (en) * 1981-01-05 1982-04-06 Pfizer Inc. 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE758782A (fr) * 1969-11-11 1971-05-10 Leo Pharm Prod Ltd Nouveaux derives d'acide 6-amidino penicillanique leur procede de preparation et leurs applications comme antibiotiques
US3957764A (en) * 1969-11-11 1976-05-18 Lovens Kemiske Fabrik Produktionsaktieselskab 6-aminopenicillanic acid derivatives
GB1303491A (xx) * 1970-03-24 1973-01-17
US3755588A (en) * 1970-11-04 1973-08-28 Leo Pharm Prod Ltd Penicillanic acid in dosage unit form
GB1335718A (en) * 1971-05-05 1973-10-31 Leo Pharm Prod Ltd Penicillin esters salts thereof and methods for their preparation
GB1405886A (en) * 1971-11-01 1975-09-10 Astra Laekemedel Ab Synergistic compositions comprising penicillin and cephalosporin antibiotics
GB1427139A (en) * 1972-03-13 1976-03-10 Astra Laekemedel Ab Penicillins

Also Published As

Publication number Publication date
SE7704311L (sv) 1977-10-16
JPS52128391A (en) 1977-10-27
SE425490B (sv) 1982-10-04
FR2348217A1 (fr) 1977-11-10
IE44809L (en) 1977-10-15
DK162177A (da) 1977-10-16
FR2348217B1 (xx) 1980-04-25
NL7704085A (nl) 1977-10-18
DE2716172C2 (de) 1985-09-05
PT66434B (en) 1978-09-20
US4181659A (en) 1980-01-01
PH14046A (en) 1980-12-29
AR218870A1 (es) 1980-07-15
ZA771935B (en) 1978-02-22
NZ183756A (en) 1978-12-18
AU2428577A (en) 1978-10-19
PT66434A (en) 1977-05-01
FI63759C (fi) 1983-08-10
GR63089B (en) 1979-08-11
ATA240677A (de) 1979-05-15
IT1116735B (it) 1986-02-10
GB1579931A (en) 1980-11-26
YU94277A (en) 1982-10-31
FI771183A (xx) 1977-10-16
AT353960B (de) 1979-12-10
ES457829A1 (es) 1978-03-01
IE44809B1 (en) 1982-04-07
FI63759B (fi) 1983-04-29
LU77135A1 (xx) 1977-08-12
JPS6129959B2 (xx) 1986-07-10
AU510825B2 (en) 1980-07-17
DK144376B (da) 1982-03-01
DE2716172A1 (de) 1977-10-27
BE853607A (fr) 1977-08-01
CA1112239A (en) 1981-11-10

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