DK139944B - Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser. - Google Patents
Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser.Info
- Publication number
- DK139944B DK139944B DK127372AA DK127372A DK139944B DK 139944 B DK139944 B DK 139944B DK 127372A A DK127372A A DK 127372AA DK 127372 A DK127372 A DK 127372A DK 139944 B DK139944 B DK 139944B
- Authority
- DK
- Denmark
- Prior art keywords
- isomers
- separation
- optically active
- chemical compounds
- certain chemical
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- SYSQUGFVNFXIIT-UHFFFAOYSA-N n-[4-(1,3-benzoxazol-2-yl)phenyl]-4-nitrobenzenesulfonamide Chemical class C1=CC([N+](=O)[O-])=CC=C1S(=O)(=O)NC1=CC=C(C=2OC3=CC=CC=C3N=2)C=C1 SYSQUGFVNFXIIT-UHFFFAOYSA-N 0.000 title 1
- 238000000926 separation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
- C07F9/6574—Esters of oxyacids of phosphorus
- C07F9/65744—Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
- Braiding, Manufacturing Of Bobbin-Net Or Lace, And Manufacturing Of Nets By Knotting (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT49167/71A IT951631B (it) | 1971-03-18 | 1971-03-18 | Composti utili per la separazione di isomeri ottici geometrici e strutturali e relativo procedimen to di sintesi |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK139944B true DK139944B (da) | 1979-05-21 |
| DK139944C DK139944C (Direct) | 1979-10-22 |
Family
ID=11269830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK127372AA DK139944B (da) | 1971-03-18 | 1972-03-17 | Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US3848030A (Direct) |
| JP (1) | JPS5547013B1 (Direct) |
| AU (1) | AU462431B2 (Direct) |
| BE (1) | BE780887A (Direct) |
| CA (1) | CA961500A (Direct) |
| CH (1) | CH576921A5 (Direct) |
| DE (1) | DE2212660C3 (Direct) |
| DK (1) | DK139944B (Direct) |
| ES (1) | ES400862A1 (Direct) |
| FR (1) | FR2129741A5 (Direct) |
| GB (1) | GB1360946A (Direct) |
| IL (1) | IL38860A (Direct) |
| IT (1) | IT951631B (Direct) |
| NL (1) | NL7203574A (Direct) |
| NO (1) | NO136357C (Direct) |
| PH (1) | PH10768A (Direct) |
| SE (1) | SE409323B (Direct) |
| ZA (1) | ZA721297B (Direct) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4143028A (en) * | 1977-12-05 | 1979-03-06 | Ciba-Geigy Corporation | Alkylated 1,1'-biphenyl-2,2'-diyl phosphonites and stabilized compositions |
| US5288914A (en) * | 1984-08-27 | 1994-02-22 | The Dow Chemical Company | Poly(arylcyclobutenes) |
| NL8403224A (nl) * | 1984-10-24 | 1986-05-16 | Oce Andeno Bv | Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen. |
| DE3940765A1 (de) * | 1989-12-09 | 1991-06-13 | Hoechst Ag | Verfahren zur herstellung reiner cyclischer phosphorsaeurediarylester |
| JPH10503752A (ja) * | 1994-05-16 | 1998-04-07 | メリル・フアーマシユウテイカルズ・インコーポレイテツド | ラセミ形α−〔4−(1,1−ジメチルエチル)フェニル〕−4−(ヒドロキシジフェニルメチル)−1−ピペリジンブタノールおよび誘導体化合物の光学分割に有用な方法およびジアステレオマー塩 |
| JP4725757B2 (ja) * | 1999-03-24 | 2011-07-13 | 東ソー株式会社 | ビナフトールリン酸誘導体及びその利用 |
| US6274745B1 (en) | 1999-03-24 | 2001-08-14 | Tosoh Corporation | Binaphthol monophosphoric acid derivative and its use |
| ATE320420T1 (de) | 1999-10-22 | 2006-04-15 | Takeda Pharmaceutical | Verfahren zur herstellung von optisch aktiven naphthalinderivaten und darin eingesetzte optische resolver |
| WO2001034557A1 (en) * | 1999-11-10 | 2001-05-17 | Takeda Chemical Industries, Ltd. | Process for the production of optically active cyclic enaminone derivatives |
| US6391926B2 (en) | 2000-03-13 | 2002-05-21 | Tosoh Corporation | Optically active phosphate derivative |
| WO2003005954A2 (en) | 2001-07-09 | 2003-01-23 | Zonagen, Inc. | Methods and materials for the treatment of testosterone deficiency in men |
| CN100410234C (zh) * | 2003-04-25 | 2008-08-13 | 东亚合成株式会社 | 利用手性布朗斯台德酸的不对称合成用催化剂和使用该催化剂的不对称合成方法 |
| US7229557B2 (en) * | 2004-02-04 | 2007-06-12 | Konec, Inc. | Method to separate stereoisomers |
| EP2486032A4 (en) * | 2009-10-09 | 2013-03-27 | Hetero Research Foundation | RACEMATSPALTUNG SUBSTITUTED 2- (2-PYRIDINYLMETHYLSULFINYL) -1H-BENZIMIDAZOLE |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| US20150202167A1 (en) | 2012-08-21 | 2015-07-23 | Repros Therapeutics Inc. | Trans-Clomiphene Formulations and Uses Thereof |
| CN104994877A (zh) | 2012-11-02 | 2015-10-21 | 利普生物药剂公司 | 用于癌症治疗的反式-克罗米芬 |
| WO2015138340A1 (en) * | 2014-03-11 | 2015-09-17 | Repros Therapeutics Inc. | Clomiphene synthesis using a single solvent |
| RU2020120156A (ru) | 2014-07-24 | 2020-07-03 | Эспен Парк Фармасьютикалз, Инк. | Лечение приливов и потери костной ткани, вызванных андрогенной депривационной терапией с применением цис-кломифена |
| EP3015453B1 (en) | 2014-10-28 | 2016-10-12 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Process for the preparation of Clomiphene |
| EP3015454A1 (en) * | 2014-10-28 | 2016-05-04 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Stable solid form of trans-Clomiphene citrate |
| WO2017182097A1 (en) | 2016-04-22 | 2017-10-26 | F.I.S. - Fabbrica Italiana Sintetici S.P.A. | Process for the preparation of enclomiphene citrate having needle shaped crystal habit. |
| EP3681491A4 (en) | 2017-09-11 | 2021-06-30 | Atossa Therapeutics, Inc. | Methods for making and using endoxifen |
| FR3082842A1 (fr) * | 2018-06-21 | 2019-12-27 | Veru Inc. | Polymorphe de cis-clomiphene (zuclomiphene) et procedes d'utilisation de celui-ci |
| US12201591B2 (en) | 2019-07-03 | 2025-01-21 | Atossa Therapeutics, Inc. | Sustained release compositions of endoxifen |
| CA3098725A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Zuclpomiphene salts and crystalline forms thereof |
| CA3098552A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Processes for the preparation of zuclomiphene and intermediates thereof |
| CA3105944A1 (en) | 2020-01-22 | 2021-07-22 | Apotex Inc. | Crystalline forms of zuclomiphene citrate |
| EP3907213A1 (en) | 2020-05-04 | 2021-11-10 | Pcas | Processes for the production of isomerically pure or enriched cis-clomiphene |
| US11578025B2 (en) | 2020-10-19 | 2023-02-14 | Apotex Inc. | Processes for the preparation of zuclomiphene intermediates |
-
1971
- 1971-03-18 IT IT49167/71A patent/IT951631B/it active
-
1972
- 1972-02-28 ZA ZA721297A patent/ZA721297B/xx unknown
- 1972-02-29 IL IL38860A patent/IL38860A/xx unknown
- 1972-03-03 AU AU39611/72A patent/AU462431B2/en not_active Expired
- 1972-03-03 PH PH13312A patent/PH10768A/en unknown
- 1972-03-09 GB GB1104172A patent/GB1360946A/en not_active Expired
- 1972-03-09 CA CA136,671A patent/CA961500A/en not_active Expired
- 1972-03-10 US US00233793A patent/US3848030A/en not_active Expired - Lifetime
- 1972-03-15 SE SE7203303A patent/SE409323B/xx unknown
- 1972-03-16 DE DE2212660A patent/DE2212660C3/de not_active Expired
- 1972-03-17 JP JP2661472A patent/JPS5547013B1/ja active Pending
- 1972-03-17 BE BE780887A patent/BE780887A/xx unknown
- 1972-03-17 FR FR7209350A patent/FR2129741A5/fr not_active Expired
- 1972-03-17 ES ES400862A patent/ES400862A1/es not_active Expired
- 1972-03-17 CH CH395572A patent/CH576921A5/xx not_active IP Right Cessation
- 1972-03-17 NO NO880/72A patent/NO136357C/no unknown
- 1972-03-17 NL NL7203574A patent/NL7203574A/xx not_active Application Discontinuation
- 1972-03-17 DK DK127372AA patent/DK139944B/da unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL7203574A (Direct) | 1972-09-20 |
| SE409323B (sv) | 1979-08-13 |
| IL38860A0 (en) | 1972-04-27 |
| ES400862A1 (es) | 1976-04-16 |
| CH576921A5 (Direct) | 1976-06-30 |
| DE2212660A1 (de) | 1972-09-28 |
| NO136357C (no) | 1977-08-24 |
| FR2129741A5 (Direct) | 1972-10-27 |
| CA961500A (en) | 1975-01-21 |
| ZA721297B (en) | 1973-03-28 |
| DE2212660C3 (de) | 1981-09-24 |
| NO136357B (Direct) | 1977-05-16 |
| IL38860A (en) | 1975-06-25 |
| GB1360946A (en) | 1974-07-24 |
| IT951631B (it) | 1973-07-10 |
| DE2212660B2 (de) | 1980-07-10 |
| US3848030A (en) | 1974-11-12 |
| DK139944C (Direct) | 1979-10-22 |
| PH10768A (en) | 1977-09-05 |
| AU462431B2 (en) | 1975-06-09 |
| AU3961172A (en) | 1973-09-06 |
| JPS5547013B1 (Direct) | 1980-11-27 |
| BE780887A (fr) | 1972-07-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK139944B (da) | Optisk aktive syrer til anvendelse ved adskillelse af isomere af visse kemiske forbindelser. | |
| DK138419B (da) | Fremgangsmåde til fremstilling af 1alfa-hydroxycholecalciferol. | |
| DK133974B (da) | Fremgangsmåde til fremstilling af optisk aktive alkylchrysanthemater. | |
| DK133828B (da) | Fremgangsmåde til fremstilling af zeaxanthin. | |
| DK135584B (da) | Analogifremgangsmåde til fremstilling af substituerede phenyl-2-pyrrolidinoner eller de cis- og trans-diastereoisomere eller optisk aktive isomere deraf. | |
| DK129291B (da) | Fremgangsmåde til fremstilling af et kimfattigt, flydedygtigt pancreatinpræparat. | |
| DK129987B (da) | Analogifremgangsmåde til fremstilling af guanidiner. | |
| DK135799B (da) | Fremgangsmåde til fremstilling af ethambutol. | |
| DK127119B (da) | Analogifremgangsmåde til fremstilling af 6-amino-9-benzylpurin-forbindelser. | |
| DK133470B (da) | Fremgangsmåde til fremstilling af 3alfa-hydroxy-5alfa-steroider. | |
| DK130582B (da) | Analogifremgangsmåde til fremstilling af racemiske blandinger eller optisk aktive isomere af 5-cyclohexyl-1-indancarboxylsyreforbindelser. | |
| DK134225B (da) | Fremgangsmåde til kontinuerlig fremstilling af opløsninger af organiske peroxider. | |
| DK129573B (da) | Analogifremgangsmåde til fremstilling af 4-(4-biphenylyl)-1-butanol. | |
| DK139582B (da) | Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive benzocycloheptaisoquinolin-forbindelser eller syreadditionssalte deraf. | |
| DK138790B (da) | Fremgangsmåde til fremstilling af phenylethanolaminforbindelser. | |
| DK138650B (da) | Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive penicilliner. | |
| DK130959B (da) | Analogifremgangsmåde til fremstilling af benzamidoacetohydroxamsyrer. | |
| DK140045B (da) | Fremgangsmåde ved membranseparering. | |
| DK139384B (da) | Fremgangsmåde til spaltning af dl-allethrolon i de optisk aktive antipoder. | |
| DK129794B (da) | Analogifremgangsmåde til fremstilling af N-acyl-3-(piperazinoethyl)-pyrazoler. | |
| DK125324B (da) | Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive sulfamoylpyrimidiner. | |
| DK126780B (da) | Fremgangsmåde til fremstilling af flavon-7-oxyacetater. | |
| DK135312B (da) | Fremgangsmåde til fremstilling af optisk aktiv dihydrochrysanthemolacton. | |
| DK123912B (da) | Fremgangsmåde til fremstilling af et granulat, der indeholder et olieagtigt eller flydende, terapeutisk anvendeligt glucofuranosid. | |
| DK130985B (da) | Fremgangsmåde til fremstilling af methanthionophosphonsyreestre. |