DK138076B - Analogifremgangsmåde til fremstilling af indolderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af indolderivater eller syreadditionssalte deraf.

Info

Publication number
DK138076B
DK138076B DK80874AA DK80874A DK138076B DK 138076 B DK138076 B DK 138076B DK 80874A A DK80874A A DK 80874AA DK 80874 A DK80874 A DK 80874A DK 138076 B DK138076 B DK 138076B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
indole derivatives
analogous process
Prior art date
Application number
DK80874AA
Other languages
Danish (da)
English (en)
Other versions
DK138076C (fr
Inventor
Marcel Descamps
Henri Inion
Original Assignee
Labaz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Labaz filed Critical Labaz
Publication of DK138076B publication Critical patent/DK138076B/da
Application granted granted Critical
Publication of DK138076C publication Critical patent/DK138076C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
DK80874AA 1973-02-16 1974-02-15 Analogifremgangsmåde til fremstilling af indolderivater eller syreadditionssalte deraf. DK138076B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB786673A GB1436771A (en) 1973-02-16 1973-02-16 Indole derivatives and process for preparing the same

Publications (2)

Publication Number Publication Date
DK138076B true DK138076B (da) 1978-07-10
DK138076C DK138076C (fr) 1978-11-27

Family

ID=9841293

Family Applications (1)

Application Number Title Priority Date Filing Date
DK80874AA DK138076B (da) 1973-02-16 1974-02-15 Analogifremgangsmåde til fremstilling af indolderivater eller syreadditionssalte deraf.

Country Status (23)

Country Link
US (1) US3946029A (fr)
JP (1) JPS5058076A (fr)
AR (1) AR202639A1 (fr)
AT (1) AT330776B (fr)
BE (1) BE810759A (fr)
CA (1) CA1003835A (fr)
CH (1) CH580073A5 (fr)
DE (1) DE2407465A1 (fr)
DK (1) DK138076B (fr)
ES (1) ES423288A1 (fr)
FI (1) FI58123C (fr)
FR (1) FR2218098B1 (fr)
GB (1) GB1436771A (fr)
HU (1) HU166731B (fr)
IE (1) IE40378B1 (fr)
IN (1) IN139121B (fr)
NL (1) NL7401955A (fr)
NO (1) NO140424C (fr)
OA (1) OA04687A (fr)
SE (1) SE390536B (fr)
SU (1) SU543343A3 (fr)
YU (1) YU36722B (fr)
ZA (1) ZA74701B (fr)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2334358A1 (fr) * 1975-12-12 1977-07-08 Sogeras Nouveaux medicaments derives de l'indole
ZA825413B (en) * 1981-08-26 1983-06-29 Pfizer Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them
JPS60142981A (ja) * 1983-12-28 1985-07-29 Yoshitomi Pharmaceut Ind Ltd ３−インド−ルカルボキサミド誘導体
US4581354A (en) * 1984-08-06 1986-04-08 Sterling Drug Inc. 3-arylcarbonyl- and 3-cycloalkylcarbonyl-1-aminoalkyl-1H-indoles, compositions and use
US5013732A (en) * 1984-08-06 1991-05-07 Sterling Drug Inc. 3-arylcarbonyl- and 3-cycloalkyl-carbonyl-1-aminoalkyl-1H-indoles
US4634776A (en) * 1984-08-06 1987-01-06 Sterling Drug, Inc. 3-arylcarbonyl-and 3-cycloalkylcarbonyl-1-aminoalkyl-1H-indoles
USRE32761E (en) * 1984-08-06 1988-10-04 Sterling Drug Inc. 3-arylcarbonyl and 3-cycloalkylcarbonyl-1-aminoalkyl-1H-indoles, compositions and use
US4978664A (en) * 1984-08-06 1990-12-18 Sterling Drug Inc. 3-arylcarbonyl- and 3-cycloalkyl-carbonyl-1-aminoalkyl-1H-indole pharmaceutical compositions
PH23498A (en) * 1984-08-06 1989-08-16 Sterling Drug Inc 3-carbonyl-1-aminoalkyl-1h-indoles,composition and use thereof
US4690943A (en) * 1984-09-19 1987-09-01 Pfizer Inc. Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds
US4840950A (en) * 1987-02-11 1989-06-20 Sterling Drug Inc. 4-arylcarbonyl-1-[(4-morpholinyl)-lower-alkyl]-1H-indoles
US5068234A (en) * 1990-02-26 1991-11-26 Sterling Drug Inc. 3-arylcarbonyl-1-(c-attached-n-heteryl)-1h-indoles
US5081122A (en) * 1990-03-05 1992-01-14 Sterling Drug Inc. Antiglaucoma compositions containing 4-arylcarbonyl-1-(4-morpholinyl)-lower-alkyl)-1H-indoles and method of use thereof
US4973587A (en) * 1990-03-08 1990-11-27 Sterling Drug Inc. 3-arylcarbonyl-1-aminoalkyl-1H-indole-containing antiglaucoma method
CA2036307C (fr) * 1990-03-08 2002-07-09 Susan Jean Ward Compositions anti-glaucome, a base de 3-arylcarbonyl-1-aminoalkyl-1h-indole; methode d'utilisation
US5013837A (en) * 1990-03-08 1991-05-07 Sterling Drug Inc. 3-Arylcarbonyl-1H-indole-containing compounds
US6342611B1 (en) * 1997-10-10 2002-01-29 Cytovia, Inc. Fluorogenic or fluorescent reporter molecules and their applications for whole-cell fluorescence screening assays for capsases and other enzymes and the use thereof
ATE247097T1 (de) * 1998-05-04 2003-08-15 Univ Connecticut Analgetische und immunomodulierende cannabinoiden
US7589220B2 (en) * 1998-06-09 2009-09-15 University Of Connecticut Inhibitors of the anandamide transporter
US7897598B2 (en) * 1998-06-09 2011-03-01 Alexandros Makriyannis Inhibitors of the anandamide transporter
US7161016B1 (en) 1998-11-24 2007-01-09 University Of Connecticut Cannabimimetic lipid amides as useful medications
US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
US6943266B1 (en) * 1999-10-18 2005-09-13 University Of Connecticut Bicyclic cannabinoid agonists for the cannabinoid receptor
US8084467B2 (en) * 1999-10-18 2011-12-27 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
US7119108B1 (en) 1999-10-18 2006-10-10 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US6900236B1 (en) * 1999-10-18 2005-05-31 University Of Connecticut Cannabimimetic indole derivatives
US7741365B2 (en) * 1999-10-18 2010-06-22 University Of Connecticut Peripheral cannabinoid receptor (CB2) selective ligands
US7329651B2 (en) * 2001-01-26 2008-02-12 University Of Connecticut Cannabimimetic ligands
JP2005503998A (ja) * 2001-01-29 2005-02-10 ユニバーシティ オブ コネチカット 受容体選択性のカンナビミメティックアミノアルキルインドール
JP4312594B2 (ja) * 2001-07-13 2009-08-12 ユニバーシティ オブ コネチカット 新規な二環式及び三環式カンナビノイド
US7666867B2 (en) * 2001-10-26 2010-02-23 University Of Connecticut Heteroindanes: a new class of potent cannabimimetic ligands
EP1998766A2 (fr) * 2005-12-16 2008-12-10 Ironwood Pharmaceuticals, Inc. Composes indole utiles
WO2007112322A2 (fr) * 2006-03-28 2007-10-04 Allergan, Inc. Composés d'indole présentant une activité biologique agoniste et/ou antagoniste vis-à-vis du récepteur de la sphingosine-1-phosphate (s1p)
JP5406716B2 (ja) 2006-08-07 2014-02-05 アイアンウッド ファーマシューティカルズ インコーポレイテッド インドール化合物
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen
CN113480530A (zh) * 2016-12-26 2021-10-08 阿里根公司 芳香烃受体调节剂
US11459322B2 (en) 2017-11-20 2022-10-04 Ariagen, Inc. Indole compounds and their use
MX2021012543A (es) 2019-04-15 2021-12-10 Ariagen Inc Compuestos de indoles quirales y su uso.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1068259B (fr) * 1954-04-28 1959-11-05
US3557142A (en) * 1968-02-20 1971-01-19 Sterling Drug Inc 4,5,6,7-tetrahydro-indole-lower-alkanoic acids and esters
US3686213A (en) * 1970-08-28 1972-08-22 American Cyanamid Co Substituted aminoethyl indoles

Also Published As

Publication number Publication date
CA1003835A (en) 1977-01-18
AR202639A1 (es) 1975-06-30
ZA74701B (en) 1974-12-24
IE40378L (en) 1974-08-16
FR2218098B1 (fr) 1978-03-24
FR2218098A1 (fr) 1974-09-13
FI58123C (fi) 1980-12-10
NO140424B (no) 1979-05-21
DE2407465A1 (de) 1974-08-22
HU166731B (fr) 1975-05-28
NL7401955A (fr) 1974-08-20
AU6536374A (en) 1975-08-14
US3946029A (en) 1976-03-23
SE390536B (sv) 1976-12-27
IN139121B (fr) 1976-05-08
NO140424C (no) 1979-08-29
YU36722B (en) 1984-08-31
IE40378B1 (en) 1979-05-23
AT330776B (de) 1976-07-26
NO740516L (no) 1974-08-19
OA04687A (fr) 1980-07-31
FI58123B (fi) 1980-08-29
YU39474A (en) 1982-02-25
DK138076C (fr) 1978-11-27
SU543343A3 (ru) 1977-01-15
ATA119174A (de) 1975-10-15
BE810759A (fr) 1974-08-08
CH580073A5 (fr) 1976-09-30
JPS5058076A (fr) 1975-05-20
ES423288A1 (es) 1976-04-16
GB1436771A (en) 1976-05-26

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