DK128738B - Analogifremgangsmåde til fremstilling af cardenolid- eller bufadienolid-3-[2',3'-didesoxyglycosider]. - Google Patents

Analogifremgangsmåde til fremstilling af cardenolid- eller bufadienolid-3-[2',3'-didesoxyglycosider].

Info

Publication number
DK128738B
DK128738B DK445070AA DK445070A DK128738B DK 128738 B DK128738 B DK 128738B DK 445070A A DK445070A A DK 445070AA DK 445070 A DK445070 A DK 445070A DK 128738 B DK128738 B DK 128738B
Authority
DK
Denmark
Prior art keywords
dideoxyglycosides
bufadienolide
cardenolide
preparation
analogous process
Prior art date
Application number
DK445070AA
Other languages
Danish (da)
English (en)
Inventor
U Stache
W Fritsch
W Haede
K Radscheit
E Lindner
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691943903 external-priority patent/DE1943903B2/de
Priority claimed from DE1943901A external-priority patent/DE1943901C3/de
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK128738B publication Critical patent/DK128738B/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J19/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 by a lactone ring
DK445070AA 1969-08-29 1970-08-28 Analogifremgangsmåde til fremstilling af cardenolid- eller bufadienolid-3-[2',3'-didesoxyglycosider]. DK128738B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19691943903 DE1943903B2 (de) 1969-08-29 1969-08-29 Verfahren zur Herstellung von Cardenolid- und Bufadienolid-3- [2'J' didesoxy-2'3-oxidoglykosiden], sowie Cxtivao&a-^rß' -didesoxy-2'3' -oxido-glykoside]
DE1943901A DE1943901C3 (de) 1969-08-29 1969-08-29 Cardenolid-3-[2', 3' - didesoxyglykoside] und Verfahren zu ihrer Herstellung, sowie Verwendung dieser Verbindungen zur Bekämpfung von Herzkrankheiten

Publications (1)

Publication Number Publication Date
DK128738B true DK128738B (da) 1974-06-24

Family

ID=25757845

Family Applications (2)

Application Number Title Priority Date Filing Date
DK445070AA DK128738B (da) 1969-08-29 1970-08-28 Analogifremgangsmåde til fremstilling af cardenolid- eller bufadienolid-3-[2',3'-didesoxyglycosider].
DK37072AA DK127421B (da) 1969-08-29 1972-01-27 Fremgangsmåde til fremstilling af cardenolid-3[2',3'-didesoxyglycosider].

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK37072AA DK127421B (da) 1969-08-29 1972-01-27 Fremgangsmåde til fremstilling af cardenolid-3[2',3'-didesoxyglycosider].

Country Status (16)

Country Link
US (1) US3838146A (es)
JP (2) JPS5248983B1 (es)
BE (1) BE755537A (es)
BG (2) BG18864A3 (es)
CA (1) CA923491A (es)
CH (2) CH537377A (es)
DK (2) DK128738B (es)
ES (1) ES383115A1 (es)
FI (1) FI49161C (es)
FR (1) FR2068530B1 (es)
GB (1) GB1323775A (es)
IL (1) IL35113A (es)
NL (1) NL7012422A (es)
OA (1) OA03653A (es)
PL (1) PL80915B1 (es)
SE (2) SE368570B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2237144A1 (de) * 1972-07-28 1974-02-14 Hoechst Ag Herzwirksame anhydrotalomethyloside und verfahren zu ihrer herstellung
DE2254060A1 (de) * 1972-11-04 1974-05-16 Hoechst Ag Cardenolid-3-eckige klammer auf 4'-amino-2',3',4'-tridesoxy-glykoside eckige klammer zu und verfahren zu ihrer herstellung
DE2256912C2 (de) * 1972-11-20 1984-04-05 Hoechst Ag, 6230 Frankfurt Digoxigenin-3-[2',3'-didesoxy-glykoside], Verfahren zu ihrer Herstellung und deren Verwendung
US5496806A (en) * 1990-01-23 1996-03-05 R. Erich Klemke Glycoside compounds and production and use thereof
CN103328038A (zh) 2010-12-01 2013-09-25 史拜诺莫度雷森公司 向神经解剖结构直接递送药剂

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1768164A1 (de) * 1968-04-06 1971-10-14 Hoechst Ag Tridesoxypyranoside und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
JPS538697B1 (es) 1978-03-31
DK127421B (da) 1973-11-05
FI49161C (fi) 1975-04-10
FR2068530B1 (es) 1973-08-10
OA03653A (fr) 1971-12-24
SE383521B (sv) 1976-03-15
FR2068530A1 (es) 1971-08-27
IL35113A (en) 1975-06-25
NL7012422A (es) 1971-03-02
BG18864A3 (es) 1975-03-20
CH537377A (de) 1973-07-13
BG20578A3 (es) 1975-12-05
GB1323775A (en) 1973-07-18
IL35113A0 (en) 1970-10-30
BE755537A (fr) 1971-03-01
CA923491A (en) 1973-03-27
CH537375A (de) 1973-05-31
PL80915B1 (es) 1975-08-30
US3838146A (en) 1974-09-24
SE368570B (es) 1974-07-08
JPS5248983B1 (es) 1977-12-14
FI49161B (es) 1974-12-31
ES383115A1 (es) 1972-12-16

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