DK127332B - Analogifremgangsmåde til fremstilling af terapeutisk virksomme 1-substituerede 2[1H]-quinazolinoner. - Google Patents

Analogifremgangsmåde til fremstilling af terapeutisk virksomme 1-substituerede 2[1H]-quinazolinoner.

Info

Publication number
DK127332B
DK127332B DK603267A DK603267A DK127332B DK 127332 B DK127332 B DK 127332B DK 603267 A DK603267 A DK 603267A DK 603267 A DK603267 A DK 603267A DK 127332 B DK127332 B DK 127332B
Authority
DK
Denmark
Prior art keywords
quinazolinones
substituted
preparation
therapeutically effective
analogous process
Prior art date
Application number
DK603267A
Other languages
English (en)
Inventor
A Allais
J Meier
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK127332B publication Critical patent/DK127332B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • C07D239/82Oxygen atoms with an aryl radical attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
DK603267A 1966-12-02 1967-12-01 Analogifremgangsmåde til fremstilling af terapeutisk virksomme 1-substituerede 2[1H]-quinazolinoner. DK127332B (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR85985A FR6001M (da) 1966-12-02 1966-12-02
FR97203A FR1520743A (fr) 1966-12-02 1967-03-02 Nouvelles quinazolinones substituées et procédé de préparation
FR106810A FR6158M (da) 1966-12-02 1967-05-18
FR125422 1967-10-23

Publications (1)

Publication Number Publication Date
DK127332B true DK127332B (da) 1973-10-22

Family

ID=27444746

Family Applications (1)

Application Number Title Priority Date Filing Date
DK603267A DK127332B (da) 1966-12-02 1967-12-01 Analogifremgangsmåde til fremstilling af terapeutisk virksomme 1-substituerede 2[1H]-quinazolinoner.

Country Status (7)

Country Link
CH (1) CH482685A (da)
DE (1) DE1695656B2 (da)
DK (1) DK127332B (da)
FR (3) FR6001M (da)
GB (1) GB1181570A (da)
IL (1) IL28991A (da)
NL (1) NL6716429A (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923803A (en) * 1968-07-18 1975-12-02 Sumitomo Chemical Co 2(1H)-Quinozalinones and process therefor
DE1932402C3 (de) * 1969-06-26 1981-09-03 Sandoz-Patent-GmbH, 7850 Lörrach 1-Isopropyl-4-phenyl-3,4-dihydro-2(1H)chinazolinonderivate und deren Weiterverarbeitung zu 1-Isopropyl-4-phenyl-2(1H)chinazolinonen
DE2118315C3 (de) * 1970-04-20 1975-04-03 Sumitomo Chemical Co., Ltd., Osaka (Japan) 2-(1H)-Chinazolinonderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
US3764600A (en) * 1970-10-06 1973-10-09 Sandoz Ag 1-substituted-quinazoline-2(1h)-thiones
US3925549A (en) * 1970-10-06 1975-12-09 Sandoz Ag 1-Substituted-quinazoline-2(1H)-thiones in the treatment of inflammation
US4071516A (en) 1976-08-20 1978-01-31 Sandoz, Inc. 4-(Acyloxyphenyl)-quinazolin-2(1H)-ones
AR038658A1 (es) 2001-06-15 2005-01-26 Novartis Ag Derivados de 4-aril-2(1h) quinazolinona y 4-aril-quinazolina 2-sustituidas, un proceso para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la preparacion de un medicamento
GB0230015D0 (en) 2002-12-23 2003-01-29 Novartis Ag Organic compounds
RU2629947C2 (ru) * 2012-04-10 2017-09-05 Аннцзи Фармасьютикал Ко., Лтд. Ингибиторы деацетилаз гистонов (hdacs)

Also Published As

Publication number Publication date
DE1695656B2 (de) 1974-06-06
GB1181570A (en) 1970-02-18
DE1695656A1 (de) 1972-04-13
FR1520743A (fr) 1968-04-12
IL28991A (en) 1972-11-28
FR6001M (da) 1968-04-29
FR6158M (da) 1968-07-01
NL6716429A (da) 1968-06-04
CH482685A (fr) 1969-12-15
DE1695656C3 (da) 1979-12-06

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Legal Events

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PBP Patent lapsed