DK121708B - Analogifremgangsmåde til fremstilling af terapeutisk virksomme 22-aza-cholestanderivater. - Google Patents
Analogifremgangsmåde til fremstilling af terapeutisk virksomme 22-aza-cholestanderivater.Info
- Publication number
- DK121708B DK121708B DK144564AA DK144564A DK121708B DK 121708 B DK121708 B DK 121708B DK 144564A A DK144564A A DK 144564AA DK 144564 A DK144564 A DK 144564A DK 121708 B DK121708 B DK 121708B
- Authority
- DK
- Denmark
- Prior art keywords
- aza
- preparation
- therapeutically effective
- cholesterol derivatives
- analogous process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0055—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J21/00—Catalysts comprising the elements, oxides, or hydroxides of magnesium, boron, aluminium, carbon, silicon, titanium, zirconium, or hafnium
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of only two carbon atoms, e.g. pregnane derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DEM56198A DE1294961B (de) | 1963-03-21 | 1963-03-21 | Verfahren zur Herstellung von 22-Azacholestanderivaten und deren Saeureadditionssalzen |
| DEM0056329 | 1963-04-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK121708B true DK121708B (da) | 1971-11-22 |
Family
ID=25987371
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK144564AA DK121708B (da) | 1963-03-21 | 1964-03-20 | Analogifremgangsmåde til fremstilling af terapeutisk virksomme 22-aza-cholestanderivater. |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US3326758A (da) |
| BR (2) | BR6457766D0 (da) |
| DE (2) | DE1294961B (da) |
| DK (1) | DK121708B (da) |
| NL (2) | NL6401648A (da) |
| SE (2) | SE334356B (da) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4125544A (en) * | 1977-06-09 | 1978-11-14 | G. D. Searle | 20/22/23/24-Oxa-7-oxocholesterols and esters thereof |
| WO1987002367A2 (en) * | 1985-10-18 | 1987-04-23 | The Upjohn Company | Cyclic hydrocarbons with an aminoalkyl sidechain |
| US5274089A (en) * | 1985-10-18 | 1993-12-28 | The Upjohn Company | Cyclic hydrocarbons with an aminoalkyl sidechain |
| AU2002211863A1 (en) * | 2000-10-06 | 2002-04-15 | Xenoport, Inc. | Bile-acid derived compounds for providing sustained systemic concentrations of drugs after oral administration |
| EP1361847A2 (en) * | 2000-10-06 | 2003-11-19 | Xenoport, Inc. | Bile-acid conjugates for providing sustained systemic concentrations of drugs |
| WO2002028411A1 (en) * | 2000-10-06 | 2002-04-11 | Xenoport, Inc. | Compounds for sustained release of orally delivered drugs |
| WO2006104883A1 (en) * | 2005-03-28 | 2006-10-05 | Shell Internationale Research Maatschappij B.V. | Formation of heteroatom containing derivatives of paraffins |
| US20090270655A1 (en) * | 2005-03-28 | 2009-10-29 | Howard Lam-Ho Fong | Conversion of Alkylhalides Into Alcohol Alkoxylates |
| WO2006104909A2 (en) * | 2005-03-28 | 2006-10-05 | Shell Internationale Research Maatschappij B.V. | Catalytic distillation process for primary haloalkanes |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3013008A (en) * | 1961-01-09 | 1961-12-12 | Searle & Co | N-substituted 20-aminopregnan-3-ols, esters thereof, and deta-derivatives corresponding |
| US3038912A (en) * | 1961-07-21 | 1962-06-12 | Searle & Co | 20(bets)-[(monoalkylamino)methyl]pregn-5-en-3beta-ols, esters corresponding and intermediates thereto |
| US3084156A (en) * | 1961-11-30 | 1963-04-02 | Searle & Co | 17beta-[n-(aminoalkyl)amino]androstan-3-ols, 5-dehydro derivatives corresponding, and esters thereof |
| US3097200A (en) * | 1962-01-03 | 1963-07-09 | Syntex Corp | 17-aminoandrostanes |
| US3144471A (en) * | 1963-01-04 | 1964-08-11 | Upjohn Co | 25-azacholesterol nu-oxide and derivatives |
-
1963
- 1963-03-21 DE DEM56198A patent/DE1294961B/de active Pending
- 1963-04-01 DE DE19631468254 patent/DE1468254A1/de active Pending
-
1964
- 1964-02-21 NL NL6401648A patent/NL6401648A/xx unknown
- 1964-03-13 NL NL6402671A patent/NL6402671A/xx unknown
- 1964-03-20 SE SE03451/64A patent/SE334356B/xx unknown
- 1964-03-20 DK DK144564AA patent/DK121708B/da unknown
- 1964-03-20 BR BR157766/64A patent/BR6457766D0/pt unknown
- 1964-03-23 US US354158A patent/US3326758A/en not_active Expired - Lifetime
- 1964-03-26 SE SE03836/64A patent/SE347506B/xx unknown
- 1964-04-02 BR BR158037/64A patent/BR6458037D0/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR6457766D0 (pt) | 1973-07-17 |
| US3326758A (en) | 1967-06-20 |
| DE1468254A1 (de) | 1969-01-09 |
| NL6401648A (da) | 1964-09-22 |
| DE1294961B (de) | 1969-08-21 |
| NL6402671A (da) | 1964-10-02 |
| SE347506B (da) | 1972-08-07 |
| SE334356B (da) | 1971-04-26 |
| BR6458037D0 (pt) | 1973-09-20 |
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