DK122581A - ISOXAZOLDE DERIVATIVES OF THEIR PREPARATION AND USE - Google Patents

ISOXAZOLDE DERIVATIVES OF THEIR PREPARATION AND USE

Info

Publication number
DK122581A
DK122581A DK122581A DK122581A DK122581A DK 122581 A DK122581 A DK 122581A DK 122581 A DK122581 A DK 122581A DK 122581 A DK122581 A DK 122581A DK 122581 A DK122581 A DK 122581A
Authority
DK
Denmark
Prior art keywords
isoxazolde
derivatives
preparation
isoxazolde derivatives
Prior art date
Application number
DK122581A
Other languages
Danish (da)
Other versions
DK151012B (en
DK151012C (en
Inventor
R Bognar
I P Ferenczik
F Sztaricskai
Z Gyoergydeak
J Szegi
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of DK122581A publication Critical patent/DK122581A/en
Publication of DK151012B publication Critical patent/DK151012B/en
Application granted granted Critical
Publication of DK151012C publication Critical patent/DK151012C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK122581A 1980-03-19 1981-03-18 ANALOGY PROCEDURE FOR PREPARING 3-METHYL-4-HALOGEN-5-AMINOOXYMETHYL-ISOXAZOLES OR ANY ACID ADDITION SALT DK151012C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU63780 1980-03-19
HU8080637A HU180567B (en) 1980-03-19 1980-03-19 Method for producing derivatives of isooxazole

Publications (3)

Publication Number Publication Date
DK122581A true DK122581A (en) 1981-09-20
DK151012B DK151012B (en) 1987-10-12
DK151012C DK151012C (en) 1988-07-04

Family

ID=10950573

Family Applications (3)

Application Number Title Priority Date Filing Date
DK122581A DK151012C (en) 1980-03-19 1981-03-18 ANALOGY PROCEDURE FOR PREPARING 3-METHYL-4-HALOGEN-5-AMINOOXYMETHYL-ISOXAZOLES OR ANY ACID ADDITION SALT
DK023087A DK151959C (en) 1980-03-19 1987-01-16 METHOD OF ANALOGY FOR THE PREPARATION OF 3-METHYL-4-HALOGENISOXAZOL-5-YL-METHYLENOXYGUANIDINE OR PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS.
DK023187A DK153549C (en) 1980-03-19 1987-01-16 METHOD OF ANALOGUE FOR THE PREPARATION OF 3-METHYL-4-HALOGEN-5-BROMETHYLAMINOMETHYLISOXAZOLES OR PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS.

Family Applications After (2)

Application Number Title Priority Date Filing Date
DK023087A DK151959C (en) 1980-03-19 1987-01-16 METHOD OF ANALOGY FOR THE PREPARATION OF 3-METHYL-4-HALOGENISOXAZOL-5-YL-METHYLENOXYGUANIDINE OR PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS.
DK023187A DK153549C (en) 1980-03-19 1987-01-16 METHOD OF ANALOGUE FOR THE PREPARATION OF 3-METHYL-4-HALOGEN-5-BROMETHYLAMINOMETHYLISOXAZOLES OR PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS.

Country Status (15)

Country Link
JP (1) JPS56158774A (en)
BE (1) BE887954A (en)
CA (1) CA1163631A (en)
CH (1) CH646157A5 (en)
DE (1) DE3110817A1 (en)
DK (3) DK151012C (en)
ES (3) ES501095A0 (en)
FI (1) FI70011C (en)
FR (1) FR2478634A1 (en)
GB (1) GB2075009B (en)
HU (1) HU180567B (en)
IT (1) IT1211010B (en)
SE (1) SE454695B (en)
SU (3) SU1053750A3 (en)
YU (1) YU42560B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1138764C (en) * 1997-04-21 2004-02-18 住友制药株式会社 Isoxazole derivatives
US6100260A (en) * 1997-04-21 2000-08-08 Sumitomo Pharmaceutical Company, Limited Isoxazole derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL302496A (en) * 1962-12-22
US3808221A (en) * 1971-04-14 1974-04-30 Hoffmann La Roche Antiandrogenic n-(3,5-dilower alkyl-4-heterocyclic)methyl)phthalimides

Also Published As

Publication number Publication date
SU1158044A3 (en) 1985-05-23
DK151959B (en) 1988-01-18
DK151012B (en) 1987-10-12
JPS56158774A (en) 1981-12-07
DK153549C (en) 1988-12-05
FR2478634B1 (en) 1983-11-10
CH646157A5 (en) 1984-11-15
YU42560B (en) 1988-10-31
FI70011B (en) 1986-01-31
HU180567B (en) 1983-03-28
ES8401758A1 (en) 1984-01-01
ES8302674A1 (en) 1983-02-16
DK23187A (en) 1987-01-16
DK153549B (en) 1988-07-25
ES511895A0 (en) 1983-05-01
GB2075009A (en) 1981-11-11
DK23087A (en) 1987-01-16
DE3110817A1 (en) 1982-03-04
SU1053750A3 (en) 1983-11-07
ES511894A0 (en) 1984-01-01
SE8101703L (en) 1981-09-20
DK151959C (en) 1988-07-11
DK151012C (en) 1988-07-04
ES501095A0 (en) 1983-02-16
SU1152518A3 (en) 1985-04-23
FR2478634A1 (en) 1981-09-25
SE454695B (en) 1988-05-24
YU68981A (en) 1983-10-31
IT8120395A0 (en) 1981-03-18
FI70011C (en) 1986-09-12
IT1211010B (en) 1989-09-29
CA1163631A (en) 1984-03-13
FI810838L (en) 1981-09-20
ES8305340A1 (en) 1983-05-01
BE887954A (en) 1981-09-16
GB2075009B (en) 1983-11-30

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Legal Events

Date Code Title Description
PBP Patent lapsed