DK121369B - Fremgangsmåde til fremstilling af 3-oxo-Δ<4>-steroider, 3-oxo-Δ<5(10)>-steroider eller enolethere deraf. - Google Patents

Fremgangsmåde til fremstilling af 3-oxo-Δ<4>-steroider, 3-oxo-Δ<5(10)>-steroider eller enolethere deraf.

Info

Publication number
DK121369B
DK121369B DK375361AA DK375361A DK121369B DK 121369 B DK121369 B DK 121369B DK 375361A A DK375361A A DK 375361AA DK 375361 A DK375361 A DK 375361A DK 121369 B DK121369 B DK 121369B
Authority
DK
Denmark
Prior art keywords
steroids
oxo
preparation
enol ethers
enol
Prior art date
Application number
DK375361AA
Other languages
Danish (da)
English (en)
Inventor
G Hughes
H Smith
Original Assignee
H Smith
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H Smith filed Critical H Smith
Publication of DK121369B publication Critical patent/DK121369B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/008Ketals at position 17
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J75/00Processes for the preparation of steroids in general

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK375361AA 1960-09-22 1961-09-21 Fremgangsmåde til fremstilling af 3-oxo-Δ<4>-steroider, 3-oxo-Δ<5(10)>-steroider eller enolethere deraf. DK121369B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB32670/60A GB1010053A (en) 1960-09-22 1960-09-22 13-alkyl 5,10-ethylenic steroid 3-ketones and their enol ethers

Publications (1)

Publication Number Publication Date
DK121369B true DK121369B (da) 1971-10-11

Family

ID=10342246

Family Applications (2)

Application Number Title Priority Date Filing Date
DK375361AA DK121369B (da) 1960-09-22 1961-09-21 Fremgangsmåde til fremstilling af 3-oxo-Δ<4>-steroider, 3-oxo-Δ<5(10)>-steroider eller enolethere deraf.
DK283471AA DK125991B (da) 1960-09-22 1971-06-10 Enolethere af 3-oxo-Δ<4>- eller 3-oxo-Δ<5(10)>- steroider til anvendelse som mellemprodukter ved syntesen af 3-oxo-Δ<4>- eller 3-oxo-Δ<5(10)>-steroider.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK283471AA DK125991B (da) 1960-09-22 1971-06-10 Enolethere af 3-oxo-Δ<4>- eller 3-oxo-Δ<5(10)>- steroider til anvendelse som mellemprodukter ved syntesen af 3-oxo-Δ<4>- eller 3-oxo-Δ<5(10)>-steroider.

Country Status (8)

Country Link
AT (2) AT268544B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (3) CH427785A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (2) DE1443124A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (2) DK121369B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR1393968A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1010053A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1061739B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (3) SE307787B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2012219096A1 (en) 2011-02-17 2013-08-29 Lupin Limited An improved process for preparation of levonorgestrel

Also Published As

Publication number Publication date
AT282083B (de) 1970-06-10
DK125991B (da) 1973-05-28
GB1010053A (en) 1965-11-17
SE307787B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1969-01-20
CH430706A (de) 1967-02-28
CH427785A (de) 1967-01-15
FR1393968A (fr) 1965-04-02
CH421096A (de) 1966-09-30
SE334878B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1971-05-10
AT268544B (de) 1969-02-10
DE1443124A1 (de) 1968-10-24
DE1793659A1 (de) 1972-01-13
DE1793659B2 (de) 1974-08-15
IT1061739B (it) 1983-04-30
SE354064B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1973-02-26
DE1793659C3 (de) 1975-03-27

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