DK115916B - Process for the preparation of 1- (2'-deoxy-D-ribofuranosyl) -5-fluoro-cytosines or 4-N-p-toluoyl derivatives thereof. - Google Patents

Process for the preparation of 1- (2'-deoxy-D-ribofuranosyl) -5-fluoro-cytosines or 4-N-p-toluoyl derivatives thereof.

Info

Publication number
DK115916B
DK115916B DK206163A DK206163A DK115916B DK 115916 B DK115916 B DK 115916B DK 206163 A DK206163 A DK 206163A DK 206163 A DK206163 A DK 206163A DK 115916 B DK115916 B DK 115916B
Authority
DK
Denmark
Prior art keywords
ribofuranosyl
cytosines
toluoyl
deoxy
fluoro
Prior art date
Application number
DK206163A
Other languages
Danish (da)
Inventor
R Duschinsky
M Hoffer
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK115916B publication Critical patent/DK115916B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
DK206163A 1962-05-01 1963-05-01 Process for the preparation of 1- (2'-deoxy-D-ribofuranosyl) -5-fluoro-cytosines or 4-N-p-toluoyl derivatives thereof. DK115916B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19143862A 1962-05-01 1962-05-01

Publications (1)

Publication Number Publication Date
DK115916B true DK115916B (en) 1969-11-24

Family

ID=22705512

Family Applications (1)

Application Number Title Priority Date Filing Date
DK206163A DK115916B (en) 1962-05-01 1963-05-01 Process for the preparation of 1- (2'-deoxy-D-ribofuranosyl) -5-fluoro-cytosines or 4-N-p-toluoyl derivatives thereof.

Country Status (6)

Country Link
BR (1) BR6348745D0 (en)
CH (1) CH421973A (en)
DK (1) DK115916B (en)
ES (1) ES287587A1 (en)
FR (1) FR1514917A (en)
GB (3) GB989456A (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA106889C2 (en) * 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі N1-ACYL-5-FLORPYRIMIDINONE DERIVATIVES
CN110003118A (en) 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 The method for preparing carboxylic ester derivative
EP3689142A1 (en) 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
EP2945634A4 (en) 2012-12-28 2016-05-25 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxamides derivatives
PL2953463T3 (en) 2012-12-31 2022-01-03 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides

Also Published As

Publication number Publication date
GB989455A (en) 1965-04-22
GB989456A (en) 1965-04-22
CH421973A (en) 1966-10-15
ES287587A1 (en) 1963-11-01
BR6348745D0 (en) 1973-07-03
FR1514917A (en) 1968-03-01
GB1002278A (en) 1965-08-25

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