DK112589B - Fremgangsmåde til fremstilling af 2,3,5,6-tetrahydroimidazo[2,1-b]thiazoler eller syreadditionssalte deraf. - Google Patents
Fremgangsmåde til fremstilling af 2,3,5,6-tetrahydroimidazo[2,1-b]thiazoler eller syreadditionssalte deraf.Info
- Publication number
- DK112589B DK112589B DK638166AA DK638166A DK112589B DK 112589 B DK112589 B DK 112589B DK 638166A A DK638166A A DK 638166AA DK 638166 A DK638166 A DK 638166A DK 112589 B DK112589 B DK 112589B
- Authority
- DK
- Denmark
- Prior art keywords
- tetrahydroimidazo
- thiazoles
- preparation
- acid addition
- addition salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/18—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36663864A | 1964-05-11 | 1964-05-11 | |
| US38723164A | 1964-08-03 | 1964-08-03 | |
| US40125164A | 1964-10-02 | 1964-10-02 | |
| US446408A US3274209A (en) | 1964-05-11 | 1965-04-07 | Certain 6-substituted-imidazo[2, 1-b] thiazole compounds |
| US553595A US3364112A (en) | 1964-05-11 | 1966-03-21 | Compositions and methods employing certain 6-substituted-imidazo(2, 1-b) thiazoles as anthelmintics |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK112589B true DK112589B (da) | 1968-12-30 |
Family
ID=27541299
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK237665AA DK122888B (da) | 1964-05-11 | 1965-05-11 | Fremgangsmåde til fremstilling af imidazo[2,1-b]thiazoler eller syreadditionssalte deraf. |
| DK638266AA DK113148B (da) | 1964-05-11 | 1966-12-09 | Fremgangsmåde til fremstilling af 5,6-dihydro-imidazo[2,1-b]thiazoler eller syreadditionssalte deraf. |
| DK638166AA DK112589B (da) | 1964-05-11 | 1966-12-09 | Fremgangsmåde til fremstilling af 2,3,5,6-tetrahydroimidazo[2,1-b]thiazoler eller syreadditionssalte deraf. |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK237665AA DK122888B (da) | 1964-05-11 | 1965-05-11 | Fremgangsmåde til fremstilling af imidazo[2,1-b]thiazoler eller syreadditionssalte deraf. |
| DK638266AA DK113148B (da) | 1964-05-11 | 1966-12-09 | Fremgangsmåde til fremstilling af 5,6-dihydro-imidazo[2,1-b]thiazoler eller syreadditionssalte deraf. |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US3274209A (da) |
| BE (1) | BE663591A (da) |
| BR (1) | BR6569567D0 (da) |
| CH (2) | CH463513A (da) |
| CS (3) | CS158182B2 (da) |
| DE (1) | DE1545995C3 (da) |
| DK (3) | DK122888B (da) |
| ES (1) | ES312813A1 (da) |
| FI (1) | FI47193C (da) |
| FR (1) | FR4705M (da) |
| GB (1) | GB1043489A (da) |
| IL (1) | IL23501A (da) |
| IT (1) | IT1053975B (da) |
| MY (1) | MY6900207A (da) |
| NL (2) | NL6505806A (da) |
| NO (1) | NO117369B (da) |
| SE (2) | SE353095B (da) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4059588A (en) * | 1965-07-19 | 1977-11-22 | Ici Australia Limited | Process for preparing 6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole |
| NL129632C (da) * | 1965-12-10 | |||
| US3673206A (en) * | 1969-04-02 | 1972-06-27 | American Cyanamid Co | RACEMIZATION OF d({30 ) 6-PHENYL-2,3,5,6-TETRAHYDROIMIDAZO {8 2,1-b{9 Thiazole |
| ZA704419B (en) * | 1969-07-21 | 1971-04-28 | Ici Australia Ltd | Injectable aqueous solutions of tetramisole |
| GB1287674A (en) * | 1969-07-21 | 1972-09-06 | Ici Australia Ltd | Injectable compositions |
| BR6915163D0 (pt) * | 1969-12-15 | 1973-05-31 | Cyanamid Co American | Processo quimico |
| US3673205A (en) * | 1970-03-25 | 1972-06-27 | American Cyanamid Co | 6-(m-AMINO AND SUBSTITUTED-AMINO PHENYL)-2,3,5,6-TETRAHYDRO{8 2,1-b{9 THIAZOLES AND METHOD OF USE |
| US3878222A (en) * | 1972-03-13 | 1975-04-15 | American Cyanamid Co | Methods of preparing substituted imidazothiazolium compounds |
| US3852458A (en) * | 1972-08-11 | 1974-12-03 | Janssen Pharmaceutica Nv | Antidepressive activity of tetramisole |
| DE2340633C2 (de) * | 1972-08-17 | 1985-09-05 | Janssen Pharmaceutica, N.V., Beerse | Pharmazeutische Verwendung von 2,3,5,6-Tetrahydro-6-phenylimidazo[2,1-b]thiazol |
| DE2340632C2 (de) * | 1972-08-17 | 1985-09-05 | Janssen Pharmaceutica, N.V., Beerse | Verwendung von 2,3,5,6-Tetrahydro-6-phenylimidazo[2,1-b]thiazol oder von dessen Salzen bei der unterstützenden Behandlung zur Rückbildung und Linderung von Neoplasmen |
| IE38848B1 (en) * | 1973-02-23 | 1978-06-07 | Fisons Ltd | Anthelmintic method and composition |
| US3860718A (en) * | 1973-09-20 | 1975-01-14 | Pfizer | IMIDAZO (2,1-b) THIAZOLE AND THIAZOLO (3,2-a) BENZIMIDAZOLE QUATERNARY SALTS HYPOGLYCEMIC AGENTS |
| US4042583A (en) * | 1973-09-20 | 1977-08-16 | Pfizer Inc. | Imidazo[2,1-b]thiazole and thiazolo[3,2-a]-benzimidazole quaternary salts as hypoglycemic agents and growth promotants |
| GB1541321A (en) * | 1976-03-10 | 1979-02-28 | Metabio | 2,3-dihydroimidazo(2,1-b)thiazole derivatives and process for their preparation |
| GB1516938A (en) * | 1976-05-01 | 1978-07-05 | Pfizer Ltd | Halopyridylamides of m-aminotetramisole and their use as anthelmintics |
| US4263311A (en) * | 1976-09-27 | 1981-04-21 | Smithkline Corporation | 5,6-Phenyl-2,3-dihydroimidazo [2,1-b] thiazoles |
| GB1533347A (en) * | 1976-10-22 | 1978-11-22 | Pfizer Ltd | Anthelmintic compounds |
| US4150141A (en) * | 1977-06-28 | 1979-04-17 | Johnson & Johnson | Treatment for scabies |
| LU77703A1 (de) * | 1977-07-07 | 1979-03-26 | Ciba Geigy Ag | Verfahren zur herstellung von bicyclischen thia-diaza-verbindungen |
| US4104400A (en) * | 1977-07-08 | 1978-08-01 | E. R. Squibb & Sons, Inc. | Imidazo(2,1-b)thiazole derivatives, compositions containing same, and method of treating helminthiasis |
| US4153706A (en) * | 1978-02-13 | 1979-05-08 | Smithkline Corporation | 6-Hydroxy-5,6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazoles |
| US4153678A (en) * | 1978-07-17 | 1979-05-08 | American Cyanamid Company | Levamisole effervescent tablets |
| CA1131226A (en) * | 1978-09-28 | 1982-09-07 | Tomohiko Munakata | Heterocyclic compounds |
| PL221188A1 (da) * | 1979-01-05 | 1980-12-01 | Ciba Geigy Ag | |
| DE3162522D1 (en) * | 1980-09-04 | 1984-04-12 | Janssen Pharmaceutica Nv | A new method of preparing 3-(2-hydroxy-2-arylethyl)-2-iminothiazolidines |
| CA1194791A (en) * | 1981-05-08 | 1985-10-08 | John M. Ballany | Parasiticidal pour-on compositions |
| US4376769A (en) * | 1981-06-19 | 1983-03-15 | Schering Corporation | Substituted imidazo thiazoles thiazines, thiazepines and thiazocines |
| AU1611383A (en) * | 1982-07-02 | 1984-01-05 | Robert Young & Company Limited | Pesticidal formulation with cypermethrin |
| ZW24186A1 (en) * | 1985-12-12 | 1987-07-08 | Smithkline Beckman Corp | Inhibition of the 5-lipoxygenase pathway |
| US5527915A (en) * | 1989-11-24 | 1996-06-18 | Janssen Pharmaceutica N.V. | Immunostimulating 6-aryl-5,6-dihydroimidazo[2,1-beta]thiazole derivatives |
| US5212192A (en) * | 1989-11-24 | 1993-05-18 | Janssen Pharmaceutica N.V. | Immunostimulating 6-aryl-5,6-dihydroimidazo[2,1-b]thiazole derivatives |
| US5516647A (en) * | 1993-11-05 | 1996-05-14 | Abbott Laboratories | Compounds useful as alkaline phosphatase inhibitors and therapeutic agents |
| JP2001302635A (ja) * | 2000-04-21 | 2001-10-31 | Suntory Ltd | 新規複素環化合物 |
| US8067382B2 (en) * | 2002-01-08 | 2011-11-29 | Merial Limited | Anthelmintic composition |
| GB201909771D0 (en) * | 2019-07-08 | 2019-08-21 | Governing Council Of The Univ Of Toronto | Imidazothiazole compounds and methods for treating plant nematode infections |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2775538A (en) * | 1951-06-04 | 1956-12-25 | Boskamp Arthur | Stabilized hexylresorcinol therapeutic agent containing castor oil |
| US2799617A (en) * | 1953-10-21 | 1957-07-16 | British Drug Houses Ltd | Piperazine adipate compositions and treatment of helminth infections therewith |
| US2969369A (en) * | 1959-10-23 | 1961-01-24 | Searle & Co | Derivatives of 3-phenyl-5, 6-dihydroimidazo-[2. 1-b] thiazoles |
| US3147273A (en) * | 1963-05-02 | 1964-09-01 | Upjohn Co | Certain 2h-isothiazolo [4, 5-b] indol-3 (4h)-one 1-oxide compounds and their preparation |
-
0
- NL NL131034D patent/NL131034C/xx active
-
1965
- 1965-04-07 US US446408A patent/US3274209A/en not_active Expired - Lifetime
- 1965-04-29 CH CH435267A patent/CH463513A/fr unknown
- 1965-04-29 CH CH604765A patent/CH440285A/fr unknown
- 1965-05-03 GB GB18479/65A patent/GB1043489A/en not_active Expired
- 1965-05-03 DE DE1545995A patent/DE1545995C3/de not_active Expired
- 1965-05-07 NL NL6505806A patent/NL6505806A/xx unknown
- 1965-05-07 BE BE663591D patent/BE663591A/xx unknown
- 1965-05-10 IT IT10267/65A patent/IT1053975B/it active
- 1965-05-10 NO NO65158028A patent/NO117369B/no unknown
- 1965-05-10 SE SE16780/69A patent/SE353095B/xx unknown
- 1965-05-10 CS CS399772*1A patent/CS158182B2/cs unknown
- 1965-05-10 CS CS304965A patent/CS158180B2/cs unknown
- 1965-05-10 CS CS284970*1A patent/CS158181B2/cs unknown
- 1965-05-10 IL IL23501A patent/IL23501A/xx unknown
- 1965-05-10 SE SE6092/65A patent/SE321237B/xx unknown
- 1965-05-10 FI FI651133A patent/FI47193C/fi active
- 1965-05-11 BR BR169567/65A patent/BR6569567D0/pt unknown
- 1965-05-11 ES ES0312813A patent/ES312813A1/es not_active Expired
- 1965-05-11 DK DK237665AA patent/DK122888B/da unknown
- 1965-08-04 FR FR27243A patent/FR4705M/fr not_active Expired
-
1966
- 1966-03-21 US US553595A patent/US3364112A/en not_active Expired - Lifetime
- 1966-12-09 DK DK638266AA patent/DK113148B/da unknown
- 1966-12-09 DK DK638166AA patent/DK112589B/da unknown
-
1969
- 1969-12-31 MY MY1969207A patent/MY6900207A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US3364112A (en) | 1968-01-16 |
| IL23501A (en) | 1968-11-27 |
| FI47193B (da) | 1973-07-02 |
| GB1043489A (en) | 1966-09-21 |
| FI47193C (fi) | 1973-10-10 |
| CH463513A (fr) | 1968-10-15 |
| CH440285A (fr) | 1967-07-31 |
| BE663591A (da) | 1965-11-08 |
| IT1053975B (it) | 1981-10-10 |
| CS158180B2 (da) | 1974-10-15 |
| DE1545995C3 (de) | 1973-11-22 |
| DE1545995B2 (de) | 1973-04-26 |
| US3274209A (en) | 1966-09-20 |
| DK122888B (da) | 1972-04-24 |
| SE321237B (da) | 1970-03-02 |
| CS158181B2 (da) | 1974-10-15 |
| ES312813A1 (es) | 1966-02-16 |
| DK113148B (da) | 1969-02-24 |
| DE1545995A1 (de) | 1969-11-13 |
| NL131034C (da) | |
| CS158182B2 (da) | 1974-10-15 |
| MY6900207A (en) | 1969-12-31 |
| NL6505806A (da) | 1965-11-12 |
| FR4705M (da) | 1966-12-26 |
| NO117369B (da) | 1969-08-04 |
| SE353095B (da) | 1973-01-22 |
| BR6569567D0 (pt) | 1973-08-02 |
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