DK0826663T3 - Alkynylaminosyrederivater og deres anvendelse som farmaceutiske forbindelser - Google Patents

Alkynylaminosyrederivater og deres anvendelse som farmaceutiske forbindelser

Info

Publication number
DK0826663T3
DK0826663T3 DK97306421T DK97306421T DK0826663T3 DK 0826663 T3 DK0826663 T3 DK 0826663T3 DK 97306421 T DK97306421 T DK 97306421T DK 97306421 T DK97306421 T DK 97306421T DK 0826663 T3 DK0826663 T3 DK 0826663T3
Authority
DK
Denmark
Prior art keywords
pharmaceutical compounds
alkynylamino
acid derivatives
phenyl
alkenyl
Prior art date
Application number
DK97306421T
Other languages
Danish (da)
English (en)
Inventor
Stephen Richard Baker
Estaban Almudena Rubio
John Goldsworthy
Tercero Concepcion Pedregal
Original Assignee
Lilly Sa
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Sa, Lilly Co Eli filed Critical Lilly Sa
Application granted granted Critical
Publication of DK0826663T3 publication Critical patent/DK0826663T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/30Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK97306421T 1996-08-27 1997-08-22 Alkynylaminosyrederivater og deres anvendelse som farmaceutiske forbindelser DK0826663T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9617822.3A GB9617822D0 (en) 1996-08-27 1996-08-27 Pharmaceutical compounds

Publications (1)

Publication Number Publication Date
DK0826663T3 true DK0826663T3 (da) 2001-11-19

Family

ID=10798951

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97306421T DK0826663T3 (da) 1996-08-27 1997-08-22 Alkynylaminosyrederivater og deres anvendelse som farmaceutiske forbindelser

Country Status (10)

Country Link
US (1) US5906985A (es)
EP (1) EP0826663B1 (es)
JP (1) JPH1087585A (es)
AT (1) ATE207879T1 (es)
CA (1) CA2213893A1 (es)
DE (1) DE69707793T2 (es)
DK (1) DK0826663T3 (es)
ES (1) ES2163103T3 (es)
GB (1) GB9617822D0 (es)
PT (1) PT826663E (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959356A (en) * 1975-03-18 1976-05-25 Richardson-Merrell Inc. Acetylene derivatives of amino acids
US4190586A (en) * 1977-07-01 1980-02-26 Merrell Toraude Et Compagnie α-Acetylenic derivatives of α-amino acids
EP0326766B1 (en) * 1988-02-05 1992-06-17 Merrell Dow Pharmaceuticals Inc. 5-substituted ornithine derivatives
FR2645858B1 (fr) * 1989-04-18 1991-06-14 Roussel Uclaf Nouveaux derives insatures de l'acide 2,6-diamino heptanedioique, leur procede de preparation et leur application comme medicaments
DE3917836A1 (de) * 1989-06-01 1990-12-20 Hoechst Ag (alpha)-trifluormethyl-substituierte aminosaeuren mit acetylenfunktion, verfahren zu deren herstellung und deren verwendung
GB9324872D0 (en) * 1993-12-03 1994-01-19 Univ Pasteur Pharmaceutical compounds
GB9325368D0 (en) * 1993-12-10 1994-02-16 Univ Bristol Organic compounds

Also Published As

Publication number Publication date
US5906985A (en) 1999-05-25
ATE207879T1 (de) 2001-11-15
GB9617822D0 (en) 1996-10-09
DE69707793D1 (de) 2001-12-06
PT826663E (pt) 2002-03-28
ES2163103T3 (es) 2002-01-16
EP0826663B1 (en) 2001-10-31
CA2213893A1 (en) 1998-02-27
JPH1087585A (ja) 1998-04-07
EP0826663A3 (en) 1999-03-03
DE69707793T2 (de) 2002-07-04
EP0826663A2 (en) 1998-03-04

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