DK0801655T3 - Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika - Google Patents

Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Info

Publication number
DK0801655T3
DK0801655T3 DK96903955T DK96903955T DK0801655T3 DK 0801655 T3 DK0801655 T3 DK 0801655T3 DK 96903955 T DK96903955 T DK 96903955T DK 96903955 T DK96903955 T DK 96903955T DK 0801655 T3 DK0801655 T3 DK 0801655T3
Authority
DK
Denmark
Prior art keywords
pct
antibiotics
basic
derivatives
sec
Prior art date
Application number
DK96903955T
Other languages
English (en)
Inventor
Sergio Lociuro
Pierfausto Seneci
Ermenegildo Restelli
Romeo Ciabatti
Original Assignee
Biosearch Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa
Application granted granted Critical
Publication of DK0801655T3 publication Critical patent/DK0801655T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK96903955T 1995-02-07 1996-02-01 Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika DK0801655T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP95101597 1995-02-07
PCT/EP1996/000407 WO1996024607A1 (en) 1995-02-07 1996-02-01 Basic proline-amide derivatives of ge 2270 and ge 2270-like antibiotics

Publications (1)

Publication Number Publication Date
DK0801655T3 true DK0801655T3 (da) 1999-02-08

Family

ID=8218961

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96903955T DK0801655T3 (da) 1995-02-07 1996-02-01 Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Country Status (12)

Country Link
US (1) US6143739A (da)
EP (1) EP0801655B1 (da)
JP (1) JP2825667B2 (da)
KR (1) KR100381688B1 (da)
AT (1) ATE165101T1 (da)
AU (1) AU693995B2 (da)
CA (1) CA2212372A1 (da)
DE (1) DE69600244T2 (da)
DK (1) DK0801655T3 (da)
ES (1) ES2115424T3 (da)
SI (1) SI0801655T1 (da)
WO (1) WO1996024607A1 (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2161344T3 (es) * 1995-02-07 2001-12-01 Biosearch Italia Spa Derivados oxazolin-amidicos basicos de los antibioticos ge2270 y similares.
DK0801655T3 (da) * 1995-02-07 1999-02-08 Biosearch Italia Spa Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika
ATE231163T1 (de) * 1996-02-14 2003-02-15 Biosearch Italia Spa Derivate des antibiotisch wirkenden faktors ge2270
EP1180513A4 (en) * 1999-04-28 2002-07-10 Takeda Chemical Industries Ltd CYCLIC AMID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND USE THEREOF
KR20050026401A (ko) * 2002-06-17 2005-03-15 비큐론 파마세티컬스 인코포레이티드 여드름 치료를 위한 ge 2270 인자 a3의 아미드유도체의 용도
US7119061B2 (en) * 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
KR101173310B1 (ko) * 2002-11-18 2012-08-10 비큐론 파마세티컬스 인코포레이티드 박테리아 감염 치료를 위한 달바반신 투여 방법
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US8288606B2 (en) * 2005-03-08 2012-10-16 Ineos Usa Llc Propylene polymer catalyst donor component
PE20080103A1 (es) * 2006-05-31 2008-04-03 Novartis Ag AMINOTIAZOLES COMO MODULADORES DEL FACTOR DE ELONGACION EF-Tu
MX2009006745A (es) * 2006-12-20 2009-08-19 Novartis Ag Macrociclos de amino-tiazol, su uso como compuestos anti-bacterianos y procesos para su produccion.
CN101945866B (zh) 2007-12-12 2013-06-19 诺瓦提斯公司 氨基噻唑化合物及其用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5202241A (en) * 1988-09-09 1993-04-13 Gruppo Lepetit S.P.A. Antibiotic GE 2270
ES2066914T3 (es) * 1989-07-04 1995-03-16 Lepetit Spa Factores a1, a2, a3 y h del antibiotico ge 2270.
DE69108972T2 (de) * 1990-03-08 1995-10-19 Lepetit Spa Antibiotika GE 2270 Faktoren B1, B2, C1, D1, D2, E und T.
IL100572A (en) * 1991-01-03 1997-01-10 Lepetit Spa Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
DE69224497T2 (de) * 1991-08-30 1998-07-02 Biosearch Italia Spa Faktor C2a des Antibiotikums CE 2270
ES2161344T3 (es) * 1995-02-07 2001-12-01 Biosearch Italia Spa Derivados oxazolin-amidicos basicos de los antibioticos ge2270 y similares.
DK0801655T3 (da) * 1995-02-07 1999-02-08 Biosearch Italia Spa Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika
ATE231163T1 (de) * 1996-02-14 2003-02-15 Biosearch Italia Spa Derivate des antibiotisch wirkenden faktors ge2270

Also Published As

Publication number Publication date
JPH10504040A (ja) 1998-04-14
ES2115424T3 (es) 1998-06-16
KR100381688B1 (ko) 2003-12-11
DE69600244T2 (de) 1998-10-01
SI0801655T1 (en) 1998-08-31
AU693995B2 (en) 1998-07-09
EP0801655A1 (en) 1997-10-22
US6143739A (en) 2000-11-07
ATE165101T1 (de) 1998-05-15
DE69600244D1 (de) 1998-05-20
EP0801655B1 (en) 1998-04-15
WO1996024607A1 (en) 1996-08-15
JP2825667B2 (ja) 1998-11-18
AU4785896A (en) 1996-08-27
CA2212372A1 (en) 1996-08-15
KR19980701996A (ko) 1998-06-25

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