DK0712408T3 - Tropyl-7-azaindol-3-ylcarboxyamider som antihostemiddel - Google Patents

Tropyl-7-azaindol-3-ylcarboxyamider som antihostemiddel

Info

Publication number
DK0712408T3
DK0712408T3 DK94921777T DK94921777T DK0712408T3 DK 0712408 T3 DK0712408 T3 DK 0712408T3 DK 94921777 T DK94921777 T DK 94921777T DK 94921777 T DK94921777 T DK 94921777T DK 0712408 T3 DK0712408 T3 DK 0712408T3
Authority
DK
Denmark
Prior art keywords
azaindol
pct
ylcarboxyamides
tropyl
cough agent
Prior art date
Application number
DK94921777T
Other languages
English (en)
Inventor
Gabriella Melillo
Marco Mantovanini
Luisa Daffonchio
Original Assignee
Dompe Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dompe Spa filed Critical Dompe Spa
Application granted granted Critical
Publication of DK0712408T3 publication Critical patent/DK0712408T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
DK94921777T 1993-08-05 1994-08-04 Tropyl-7-azaindol-3-ylcarboxyamider som antihostemiddel DK0712408T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT93MI001780A IT1265057B1 (it) 1993-08-05 1993-08-05 Tropil 7-azaindolil-3-carbossiamidi
PCT/IB1994/000234 WO1995004742A1 (en) 1993-08-05 1994-08-04 Tropyl 7-azaindol-3-ylcarboxyamides as antitussive agent

Publications (1)

Publication Number Publication Date
DK0712408T3 true DK0712408T3 (da) 1999-07-12

Family

ID=11366781

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94921777T DK0712408T3 (da) 1993-08-05 1994-08-04 Tropyl-7-azaindol-3-ylcarboxyamider som antihostemiddel

Country Status (12)

Country Link
US (1) US5750536A (da)
EP (1) EP0712408B1 (da)
AT (1) ATE172735T1 (da)
AU (1) AU683524B2 (da)
CA (1) CA2172616C (da)
DE (1) DE69414256T2 (da)
DK (1) DK0712408T3 (da)
ES (1) ES2126766T3 (da)
HK (1) HK1011359A1 (da)
IT (1) IT1265057B1 (da)
WO (1) WO1995004742A1 (da)
ZA (1) ZA945817B (da)

Families Citing this family (31)

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Publication number Priority date Publication date Assignee Title
IT1303123B1 (it) 1998-10-13 2000-10-30 Rotta Research Lab Derivati basici di benz(e)isoindol-1-oni e pirrolo(3,4-c)chinolin-1-oni ad attivita' 5ht3 antagonista, loro preparazione ed
US6476034B2 (en) 2000-02-22 2002-11-05 Bristol-Myers Squibb Company Antiviral azaindole derivatives
US20040110785A1 (en) 2001-02-02 2004-06-10 Tao Wang Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
US20030207910A1 (en) 2001-02-02 2003-11-06 Tao Wang Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
US6825201B2 (en) 2001-04-25 2004-11-30 Bristol-Myers Squibb Company Indole, azaindole and related heterocyclic amidopiperazine derivatives
AR036040A1 (es) * 2001-06-12 2004-08-04 Upjohn Co Compuestos de heteroarilo multiciclicos sustituidos con quinuclidinas y composiciones farmaceuticas que los contienen
CA2462453C (en) 2001-10-02 2009-07-28 Pharmacia & Upjohn Company Azabicyclic-substituted fused-heteroaryl compounds for the treatment of disease
WO2003028724A1 (en) * 2001-10-04 2003-04-10 Smithkline Beecham Corporation Chk1 kinase inhibitors
US20030236277A1 (en) 2002-02-14 2003-12-25 Kadow John F. Indole, azaindole and related heterocyclic pyrrolidine derivatives
US6894042B2 (en) 2002-02-19 2005-05-17 Pharmacia & Upjohn Company Azabicyclic compounds for the treatment of disease
CA2476681A1 (en) 2002-02-19 2003-08-28 Bruce N. Rogers Fused bicyclic-n-bridged-heteroaromatic carboxamides for the treatment of disease
US7037913B2 (en) 2002-05-01 2006-05-02 Bristol-Myers Squibb Company Bicyclo 4.4.0 antiviral derivatives
US7348337B2 (en) 2002-05-28 2008-03-25 Bristol-Myers Squibb Company Indole, azaindole and related heterocyclic 4-alkenyl piperidine amides
US6900206B2 (en) 2002-06-20 2005-05-31 Bristol-Myers Squibb Company Indole, azaindole and related heterocyclic sulfonylureido piperazine derivatives
CA2503786A1 (en) * 2002-11-01 2004-05-13 Pharmacia & Upjohn Company Llc Compounds having both alpha7 nicotinic agonist activity and 5ht, antagonist activity for treatment of cns diseases
US20050075364A1 (en) 2003-07-01 2005-04-07 Kap-Sun Yeung Indole, azaindole and related heterocyclic N-substituted piperazine derivatives
US20050124623A1 (en) 2003-11-26 2005-06-09 Bender John A. Diazaindole-dicarbonyl-piperazinyl antiviral agents
SI1696920T1 (sl) 2003-12-19 2015-02-27 Plexxikon Inc. Spojine in postopki za razvoj modulatorjev ret
ATE487716T1 (de) * 2004-04-22 2010-11-15 Memory Pharm Corp Indole, 1h-indazole, 1,2-benzisoxazole, 1,2- benzoisothiazole, deren herstellung und verwendungen
US7498342B2 (en) 2004-06-17 2009-03-03 Plexxikon, Inc. Compounds modulating c-kit activity
US20060100432A1 (en) 2004-11-09 2006-05-11 Matiskella John D Crystalline materials of 1-(4-benzoyl-piperazin-1-yl)-2-[4-methoxy-7-(3-methyl-[1,2,4]triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-ethane-1,2-dione
PE20071159A1 (es) * 2005-10-31 2007-11-30 Schering Corp Derivados de tropano 3-monosustituido como ligandos de receptores de nociceptina
US7851476B2 (en) 2005-12-14 2010-12-14 Bristol-Myers Squibb Company Crystalline forms of 1-benzoyl-4-[2-[4-methoxy-7-(3-methyl-1H-1,2,4-triazol-1-YL)-1-[(phosphonooxy)methyl]-1H-pyrrolo[2,3-C]pyridin-3-YL]-1,2-dioxoethyl]-piperazine
US7807671B2 (en) 2006-04-25 2010-10-05 Bristol-Myers Squibb Company Diketo-piperazine and piperidine derivatives as antiviral agents
WO2008063888A2 (en) 2006-11-22 2008-05-29 Plexxikon, Inc. Compounds modulating c-fms and/or c-kit activity and uses therefor
US20100190777A1 (en) 2007-07-17 2010-07-29 Plexxikon Inc. Compounds and methods for kinase modulation, and indications therefor
MX2011008303A (es) 2009-04-03 2011-11-29 Plexxikon Inc Composiciones del acido propano-1-sulfonico {3-[5-(4-cloro-fenil)- 1h-pirrolo [2,3-b]-piridina-3-carbonil]-2,4-difluoro-fenil}-amida y el uso de las mismas.
AU2010315126B2 (en) 2009-11-06 2015-06-25 Plexxikon, Inc. Compounds and methods for kinase modulation, and indications therefor
AU2012214762B2 (en) 2011-02-07 2015-08-13 Plexxikon Inc. Compounds and methods for kinase modulation, and indications therefor
TWI558702B (zh) 2011-02-21 2016-11-21 普雷辛肯公司 醫藥活性物質的固態形式
US9150570B2 (en) 2012-05-31 2015-10-06 Plexxikon Inc. Synthesis of heterocyclic compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0421681A (ja) * 1990-05-14 1992-01-24 Fujisawa Pharmaceut Co Ltd ピロロピリジン誘導体
US5260303A (en) * 1991-03-07 1993-11-09 G. D. Searle & Co. Imidazopyridines as serotonergic 5-HT3 antagonists
IT1255467B (it) * 1992-07-29 1995-11-02 Dompe Farmaceutici Spa Ammidi acriliche farmacologicamente attive
JPH09221681A (ja) * 1996-02-16 1997-08-26 Mitsui Petrochem Ind Ltd プラスチックの油化方法

Also Published As

Publication number Publication date
AU1318295A (en) 1995-02-28
US5750536A (en) 1998-05-12
DE69414256D1 (de) 1998-12-03
CA2172616A1 (en) 1995-02-16
AU683524B2 (en) 1997-11-13
HK1011359A1 (en) 1999-07-09
EP0712408A1 (en) 1996-05-22
DE69414256T2 (de) 1999-06-02
ATE172735T1 (de) 1998-11-15
ZA945817B (en) 1995-03-10
IT1265057B1 (it) 1996-10-28
ITMI931780A0 (it) 1993-08-05
EP0712408B1 (en) 1998-10-28
ITMI931780A1 (it) 1995-02-05
WO1995004742A1 (en) 1995-02-16
CA2172616C (en) 2001-05-29
ES2126766T3 (es) 1999-04-01

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