DK0548824T3 - Nye tricycliske steroidanaloge - Google Patents
Nye tricycliske steroidanalogeInfo
- Publication number
- DK0548824T3 DK0548824T3 DK92121556.2T DK92121556T DK0548824T3 DK 0548824 T3 DK0548824 T3 DK 0548824T3 DK 92121556 T DK92121556 T DK 92121556T DK 0548824 T3 DK0548824 T3 DK 0548824T3
- Authority
- DK
- Denmark
- Prior art keywords
- fluoroalkyl
- carbonyl
- alkyl
- different
- same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
- C07C69/716—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
- C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
- C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
- C07C2603/16—Benz[e]indenes; Hydrogenated benz[e]indenes
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/811,208 US5206415A (en) | 1991-12-20 | 1991-12-20 | Tricyclic steroid analogs |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0548824T3 true DK0548824T3 (da) | 1996-02-19 |
Family
ID=25205887
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK92121556.2T DK0548824T3 (da) | 1991-12-20 | 1992-12-18 | Nye tricycliske steroidanaloge |
Country Status (7)
Country | Link |
---|---|
US (3) | US5206415A (de) |
EP (1) | EP0548824B1 (de) |
JP (1) | JP3238962B2 (de) |
AT (1) | ATE133654T1 (de) |
CA (1) | CA2085819A1 (de) |
DE (1) | DE69208068T2 (de) |
DK (1) | DK0548824T3 (de) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5434274A (en) * | 1991-12-20 | 1995-07-18 | Washington University | Benz(epsilon)indene compounds |
US5696199A (en) * | 1995-12-07 | 1997-12-09 | Minnesota Mining And Manufacturing Company | Pressure-sensitive adhesive polyacrylate polymer and method of making |
US6787530B1 (en) | 1996-08-23 | 2004-09-07 | Monash University | Use of pregnane-diones as analgesic agents |
CA2330611A1 (en) | 1998-05-22 | 1999-12-02 | The Board Of Trustees Of The Leland Stanford Junior University | Bifunctional molecules and therapies based thereon |
WO1999066915A2 (en) | 1998-06-23 | 1999-12-29 | Southern Illinois University At Carbondale | Therapeutic applications of estrogenic carboxylic acids |
US6653471B2 (en) | 2000-08-07 | 2003-11-25 | Neurogen Corporation | Heterocyclic compounds as ligands of the GABAA receptor |
US20020072509A1 (en) * | 2000-10-11 | 2002-06-13 | Stein Donald Gerald | Methods for the treatment of a traumatic central nervous system injury |
AR031473A1 (es) * | 2000-11-20 | 2003-09-24 | Lundbeck & Co As H | Intensificadores de gaba en el tratamiento de enfermedades relacionadas con una reducida actividad neuroesteroide |
US20030037354A1 (en) * | 2001-08-02 | 2003-02-20 | Ornitz David M. | Animal model with disrupted Fgf14 gene |
US7473687B2 (en) * | 2005-03-24 | 2009-01-06 | Emory University | Methods for the treatment of a traumatic central nervous system injury |
JP5295755B2 (ja) | 2005-03-24 | 2013-09-18 | エモリー ユニバーシティー | プロゲステロンによる外傷性脳損傷の治療のための投薬レジメン |
EP1889198B1 (de) | 2005-04-28 | 2014-11-26 | Proteus Digital Health, Inc. | Pharma-informatiksystem |
JP2009508494A (ja) | 2005-09-16 | 2009-03-05 | ラプトール ファーマシューティカル インコーポレイテッド | Crを含むタンパク質に対して特異的な受容体−結合タンパク質(rap)変異体を含む組成物およびその使用 |
DK3395372T3 (da) | 2009-02-20 | 2022-04-19 | Enhanx Biopharm Inc | System til afgivelse af glutathion-baseret medikament |
EP2427178B1 (de) | 2009-05-06 | 2023-01-04 | Laboratory Skin Care, Inc. | Dermale freisetzungszusammensetzung mit wirkstoff-calciumphosphat-partikelkomplexen und anwendungsverfahren |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2830075A (en) * | 1954-05-10 | 1958-04-08 | Farinacci Nicholas Thomas | 2-alpha-carbonylated 8, 13-dimethyl polyhydrophenanthrene compounds and preparation thereof |
US2830325A (en) * | 1956-05-10 | 1958-04-15 | Davol Rubber Co | Mold for forming open-ended bulbs |
US3293284A (en) * | 1964-08-07 | 1966-12-20 | Searle & Co | 1, 2-seco-alpha-nor-5 alpha-androstane-1, 2, 17 beta-triols, 17-alkylated-1, 2-seco-alpha-nor-5 alpha-androstane-1, 2, 17 beta-triols and esters thereof |
US3281431A (en) * | 1964-09-28 | 1966-10-25 | Searle & Co | 17-oxygenated-2-thia-5alpha-androstanes and derivatives thereof |
FR1526962A (fr) * | 1967-01-06 | 1968-05-31 | Roussel Uclaf | Nouveau procédé de préparation d'un composé gonatriénique et produits en résultant |
IL32496A (en) * | 1968-07-24 | 1973-06-29 | Roussel Uclaf | 1-oxa-a-nor-androstanes |
US3821288A (en) * | 1971-07-01 | 1974-06-28 | Syntex Inc | 16,17-seco-a-nor steroids |
GB2068363A (en) * | 1980-01-30 | 1981-08-12 | Sarabhai Ambalal Ets | Substituted Benzhydrindanes |
US4874891A (en) * | 1986-05-01 | 1989-10-17 | Washington University | Open "D" ring hormone analogs |
AU609927B2 (en) * | 1987-08-25 | 1991-05-09 | Kelvin W. Gee | Compositions and methods for alleviating stress, anxiety and seizure activity |
-
1991
- 1991-12-20 US US07/811,208 patent/US5206415A/en not_active Expired - Lifetime
-
1992
- 1992-12-18 JP JP33897092A patent/JP3238962B2/ja not_active Expired - Fee Related
- 1992-12-18 EP EP92121556A patent/EP0548824B1/de not_active Expired - Lifetime
- 1992-12-18 CA CA002085819A patent/CA2085819A1/en not_active Abandoned
- 1992-12-18 DE DE69208068T patent/DE69208068T2/de not_active Expired - Fee Related
- 1992-12-18 DK DK92121556.2T patent/DK0548824T3/da active
- 1992-12-18 AT AT92121556T patent/ATE133654T1/de not_active IP Right Cessation
-
1993
- 1993-01-14 US US08/004,768 patent/US5292906A/en not_active Expired - Lifetime
- 1993-10-15 US US08/136,150 patent/US5344826A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP0548824A1 (de) | 1993-06-30 |
EP0548824B1 (de) | 1996-01-31 |
US5292906A (en) | 1994-03-08 |
JP3238962B2 (ja) | 2001-12-17 |
DE69208068T2 (de) | 1996-05-30 |
ATE133654T1 (de) | 1996-02-15 |
US5344826A (en) | 1994-09-06 |
JPH05306257A (ja) | 1993-11-19 |
DE69208068D1 (de) | 1996-03-14 |
US5206415A (en) | 1993-04-27 |
CA2085819A1 (en) | 1993-06-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK0548824T3 (da) | Nye tricycliske steroidanaloge | |
EP0515514A4 (en) | 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents | |
ES479134A1 (es) | Un procedimiento para la preparacion de un derivado de car- boestirilo. | |
HUP0002682A1 (hu) | VLA-4 által közvetített leukocita adhéziót gátló dipeptidszármazékok | |
SE8704599D0 (sv) | Teobrominderivat | |
RO82370B (ro) | Procedeu pentru prepararea unor derivati de 9-aminodibenzopiran | |
DE69430636T2 (de) | Neue imidazol-derivate und verfahren zu deren herstellung | |
JPS5472248A (en) | Light stabilizer for synthetic resin | |
DK0488513T3 (da) | Anvendelse af dioxabicyclo(3.3.0)octanderivater til fremstilling af et medikament til inhibering af cholesterolmetabolismen | |
ES8306474A1 (es) | Derivados de encefalina. | |
ATE140700T1 (de) | Flüssigkristalline verbindung, diese enthaltende flüssigkristalline zusammensetzung und diese zusammensetzung verwendende vorrichtung | |
DK0601191T3 (da) | Hidtil ukendt tetracyklisk forbindelse | |
UA43338C2 (uk) | Похідні бензолу | |
GR900100035A (el) | Παράγωγα υδροξυαλκανοκαρβονικού οξέος, η παρασευή και η χρησιμοπποίηση τους. | |
ATE72247T1 (de) | Estran- und androstan-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende praeparate. | |
EP0630893A4 (de) | N,n'-disubstituierte amidderivate. | |
ATE94526T1 (de) | Verbindung, verfahren und verwendung. | |
AR247737A1 (es) | Un procedimiento para la fabricacion de compuestos. | |
ES2138052T3 (es) | Derivados de ciclopropano y agentes antiviricos que los contienen. | |
IL132225A0 (en) | Chelating agents | |
GB1515161A (en) | Selenium labelled nucleotides | |
JPS52124642A (en) | Elevator | |
ES2170802T3 (es) | Carboxamidas biciclicas como ligandos de los receptores 5-ht1a. | |
TW216417B (en) | Carboxylic acid derivative having retinoid type pharmacological activities | |
ATE1008T1 (de) | Isomerisation von 3-azabi cyclo(3.1.0)hexan-derivaten. |