DK0548790T3 - (1S)-hydroxyalkyloxapenem-3-carboxylsyrer og deres anvendelse som betalactamasehæmmere - Google Patents

(1S)-hydroxyalkyloxapenem-3-carboxylsyrer og deres anvendelse som betalactamasehæmmere

Info

Publication number
DK0548790T3
DK0548790T3 DK92121455.7T DK92121455T DK0548790T3 DK 0548790 T3 DK0548790 T3 DK 0548790T3 DK 92121455 T DK92121455 T DK 92121455T DK 0548790 T3 DK0548790 T3 DK 0548790T3
Authority
DK
Denmark
Prior art keywords
compounds
carboxylic acids
lactamase inhibitors
beta
hydroxyalkyloxapenem
Prior art date
Application number
DK92121455.7T
Other languages
English (en)
Inventor
Hans Rudolf Prof Dr Pfaendler
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK0548790T3 publication Critical patent/DK0548790T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK92121455.7T 1991-12-20 1992-12-17 (1S)-hydroxyalkyloxapenem-3-carboxylsyrer og deres anvendelse som betalactamasehæmmere DK0548790T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4142423A DE4142423A1 (de) 1991-12-20 1991-12-20 ((ls)-hydroxyalkyl)oxapenem-3-carbonsaeuren und ihre verwendung als betalactamasehemmer

Publications (1)

Publication Number Publication Date
DK0548790T3 true DK0548790T3 (da) 1996-06-03

Family

ID=6447783

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92121455.7T DK0548790T3 (da) 1991-12-20 1992-12-17 (1S)-hydroxyalkyloxapenem-3-carboxylsyrer og deres anvendelse som betalactamasehæmmere

Country Status (7)

Country Link
EP (1) EP0548790B1 (da)
JP (1) JPH05194528A (da)
AT (1) ATE137503T1 (da)
CA (1) CA2085834A1 (da)
DE (2) DE4142423A1 (da)
DK (1) DK0548790T3 (da)
ES (1) ES2087421T3 (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1199077A1 (en) * 2000-10-19 2002-04-24 Amura Limited Stable compositions of oxapenem-3-carboxylic acids by Co-lyophilisation with pharmaceutical carriers
GB2369358A (en) * 2000-10-19 2002-05-29 Amura Ltd Oxapenems and pharmaceutical compositions thereof
JP4283535B2 (ja) * 2000-10-19 2009-06-24 アムラ リミティド オキサペネム−３−カルボン酸を含有する医薬組成物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3725375A1 (de) * 1987-07-31 1989-02-09 Bayer Ag Stabile oxapenem-3-carbonsaeuren
DE3833693A1 (de) * 1988-10-04 1990-04-05 Bayer Ag Stabile oxapenem-3-carbonsaeuren und ihre verwendung als ss-lactamasehemmer
DE4027928A1 (de) * 1990-09-04 1992-03-05 Bayer Ag Neue 2-tert.substituierte methyl-oxapenem-3-carbonsaeuren und -ester, verfahren zu ihrer herstellung und ihre verwendung

Also Published As

Publication number Publication date
CA2085834A1 (en) 1993-06-21
ES2087421T3 (es) 1996-07-16
JPH05194528A (ja) 1993-08-03
DE4142423A1 (de) 1993-06-24
ATE137503T1 (de) 1996-05-15
EP0548790A1 (de) 1993-06-30
EP0548790B1 (de) 1996-05-01
DE59206181D1 (de) 1996-06-05

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