DE69923718D1 - Ppar-alpha und ppar-gamma-hemmer - Google Patents
Ppar-alpha und ppar-gamma-hemmerInfo
- Publication number
- DE69923718D1 DE69923718D1 DE69923718T DE69923718T DE69923718D1 DE 69923718 D1 DE69923718 D1 DE 69923718D1 DE 69923718 T DE69923718 T DE 69923718T DE 69923718 T DE69923718 T DE 69923718T DE 69923718 D1 DE69923718 D1 DE 69923718D1
- Authority
- DE
- Germany
- Prior art keywords
- ppar
- gamma
- alpha
- medicinal drug
- fatty acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Diabetes (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/JP1999/005217 WO2001021181A1 (fr) | 1999-09-24 | 1999-09-24 | INHIBITEURS DE PPARα ET PPAR$g(g) |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69923718D1 true DE69923718D1 (de) | 2005-03-17 |
DE69923718T2 DE69923718T2 (de) | 2006-01-12 |
Family
ID=14236796
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69923718T Expired - Lifetime DE69923718T2 (de) | 1999-09-24 | 1999-09-24 | Ppar-alpha und ppar-gamma-hemmer |
Country Status (7)
Country | Link |
---|---|
US (1) | US6762171B1 (de) |
EP (1) | EP1214939B1 (de) |
AT (1) | ATE288757T1 (de) |
AU (1) | AU5759499A (de) |
CA (1) | CA2383140C (de) |
DE (1) | DE69923718T2 (de) |
WO (1) | WO2001021181A1 (de) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2003514855A (ja) * | 1999-10-13 | 2003-04-22 | チャコン,マルコ,エー. | カロリー制限の効果を模倣した治療的介入 |
EP1911462A3 (de) | 2001-01-26 | 2011-11-30 | Schering Corporation | Zusammensetzungen enthaltend einen Sterolabsorptionshemmer |
US20030104975A1 (en) * | 2001-06-14 | 2003-06-05 | Johan Auwerx | Cofactor-based screening method for nuclear receptor modulators and related modulators |
CA2576993C (en) * | 2004-08-12 | 2013-09-24 | Amgen Inc. | Bisaryl-sulfonamides |
CA2666670A1 (en) * | 2006-10-20 | 2008-05-02 | Dow Global Technologies Inc. | Uses of water-soluble cellulose derivatives for preventing or treating metabolic syndrome |
WO2012027331A1 (en) | 2010-08-27 | 2012-03-01 | Ironwood Pharmaceuticals, Inc. | Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders |
WO2014037834A2 (en) * | 2012-09-08 | 2014-03-13 | Mahesh Kandula | Compositions and methods for the treatment of inflammation and lipid disorders |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0482097B1 (de) * | 1989-07-11 | 2001-06-06 | Genentech, Inc. | Oberflächenaktive zusammensetzungen und verfahren |
EP0788353A1 (de) * | 1995-09-18 | 1997-08-13 | Ligand Pharmaceuticals, Inc. | Ppar gamma antagonisten zur behandlung der fettleibigkeit |
AU7493198A (en) * | 1997-05-15 | 1998-12-08 | Geoffrey J Schmidt | Method of reducing immunological tolerance to malignancy |
-
1999
- 1999-09-24 DE DE69923718T patent/DE69923718T2/de not_active Expired - Lifetime
- 1999-09-24 AT AT99944810T patent/ATE288757T1/de not_active IP Right Cessation
- 1999-09-24 CA CA002383140A patent/CA2383140C/en not_active Expired - Fee Related
- 1999-09-24 US US10/070,439 patent/US6762171B1/en not_active Expired - Fee Related
- 1999-09-24 EP EP99944810A patent/EP1214939B1/de not_active Expired - Lifetime
- 1999-09-24 WO PCT/JP1999/005217 patent/WO2001021181A1/ja active IP Right Grant
- 1999-09-24 AU AU57594/99A patent/AU5759499A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1214939B1 (de) | 2005-02-09 |
CA2383140C (en) | 2007-12-04 |
AU5759499A (en) | 2001-04-24 |
ATE288757T1 (de) | 2005-02-15 |
EP1214939A4 (de) | 2003-10-01 |
DE69923718T2 (de) | 2006-01-12 |
US6762171B1 (en) | 2004-07-13 |
EP1214939A1 (de) | 2002-06-19 |
WO2001021181A1 (fr) | 2001-03-29 |
CA2383140A1 (en) | 2001-03-29 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR0207910A (pt) | HidantÈnios e sua utilização no tratamento do diabetes | |
CY1108823T1 (el) | Παραγωγα 2-υδροξυ-3-ετεροαρυλινδολης ως αναστολεις της gsk3 | |
AU8355998A (en) | Medicinal compositions with cholesterol-lowering effect | |
NZ515705A (en) | Substituted phenylpropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor (PPAR) alpha | |
BR0111438A (pt) | Análogos de ácido barbitúrico como agentes terapeuticos | |
KR950703953A (ko) | 2-아미노-6-n-프로필아미노-4, 5, 6, 7-테트라하이드로벤조티아졸(프라미펙솔)의 항우울제로서의 용도(Use of 2-amino-6-n-propylamino-4, 5, 6, 7-tetrahydrobenzothiazole (pramipexol)as an antidepressant drug) | |
AR013079A1 (es) | Derivados sustituidos de tetrahidrofurano-3-onas, de tetrahidropirano-3- onas y tetrahidrotiofen-3-onas, un procedimiento para su preparacion unacomposicion farmaceutica de un medicamento util como inhibidores de proteasas e intermediarios | |
ZA874812B (en) | Drug | |
BR0012610A (pt) | Novo derivado de difenilpiperidina | |
BR0107628A (pt) | l,2-diarilbenzimidazóis para tratamento de doenças que estão associadas a uma ativação microglial | |
DE69923718D1 (de) | Ppar-alpha und ppar-gamma-hemmer | |
PT1150686E (pt) | Matriz directamente compressivel para libertacao controlada de doses diarias unitarias de claritromicina | |
EP1284265A4 (de) | Benzothiophenderivate und deren medizinische verwendungen | |
HUP0203884A2 (hu) | Kristályos oximinoalkánsav-származékok és cukorbaj elleni alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények | |
LV10267A (lv) | Savienojums arstniecibas lidzeklis panemiens savienojuma iegusanai | |
AR035006A1 (es) | Derivado de naftiridin-dibenzo[a,d]ciclohepteno-10-acetico, composicion farmaceutica, y el uso de dicho derivado para la fabricacion de un medicamento. | |
FR2387221A1 (fr) | Derives du benzimidazole utilisables comme substances actives de medicaments veterinaires | |
FR2701260B1 (fr) | Dérivés de 2-[4-(4-azolylbutyl)-1-pipérazinyl]-5-hydroxypyrimidine, leur préparation et leur application en tant que médicaments. | |
FR2363324A1 (fr) | Solutions aqueuses ou hydroalcooliques stables d'essences parfumees ou de medicaments solubles dans l'huile | |
FR2376661A1 (fr) | Medicaments anthelminthiques renfermant comme substances actives des anilinomethylene-malononitriles | |
BR0015781A (pt) | Composição farmacêutica para tratamento de doenças associadas à diminuição de massa óssea | |
FR2361110A1 (fr) | Medicaments anthelminthiques renfermant une association synergique de substances actives | |
BRPI0413101A (pt) | compostos de sulfonamida derivado de benzoxazinona, sua preparação e uso como medicamentos | |
FI964303A (fi) | Keuhkosydänvian hoitamiseen tarkoitettu aine | |
HUP0202893A2 (hu) | Szubsztituált benziltiazolidin-2,4-dion-származékok és ezeket tartalmazó gyógyászati készítmények |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition |