DE69713098T2 - Verfahren zur monoacylierung von hydroxytaxanen - Google Patents

Verfahren zur monoacylierung von hydroxytaxanen

Info

Publication number
DE69713098T2
DE69713098T2 DE69713098T DE69713098T DE69713098T2 DE 69713098 T2 DE69713098 T2 DE 69713098T2 DE 69713098 T DE69713098 T DE 69713098T DE 69713098 T DE69713098 T DE 69713098T DE 69713098 T2 DE69713098 T2 DE 69713098T2
Authority
DE
Germany
Prior art keywords
hydroxytaxans
monoacylating
monoacylating hydroxytaxans
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69713098T
Other languages
English (en)
Other versions
DE69713098D1 (de
Inventor
Eric Didier
Pascal Pecquet
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Publication of DE69713098D1 publication Critical patent/DE69713098D1/de
Application granted granted Critical
Publication of DE69713098T2 publication Critical patent/DE69713098T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE69713098T 1996-07-09 1997-07-04 Verfahren zur monoacylierung von hydroxytaxanen Expired - Fee Related DE69713098T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9608505A FR2750989B1 (fr) 1996-07-09 1996-07-09 Procede de monoacylation d'hydroxy taxanes
PCT/FR1997/001201 WO1998001435A1 (fr) 1996-07-09 1997-07-04 Procede de monoacylation d'hydroxy taxanes

Publications (2)

Publication Number Publication Date
DE69713098D1 DE69713098D1 (de) 2002-07-11
DE69713098T2 true DE69713098T2 (de) 2002-11-28

Family

ID=9493827

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69713098T Expired - Fee Related DE69713098T2 (de) 1996-07-09 1997-07-04 Verfahren zur monoacylierung von hydroxytaxanen

Country Status (20)

Country Link
US (1) US6127555A (de)
EP (1) EP0912536B1 (de)
JP (1) JP2000514082A (de)
AR (1) AR007834A1 (de)
AT (1) ATE218559T1 (de)
AU (1) AU3546997A (de)
CA (1) CA2259278A1 (de)
CO (1) CO4890872A1 (de)
DE (1) DE69713098T2 (de)
DK (1) DK0912536T3 (de)
ES (1) ES2177988T3 (de)
FR (1) FR2750989B1 (de)
IN (1) IN188980B (de)
MA (1) MA24258A1 (de)
PE (1) PE69499A1 (de)
PT (1) PT912536E (de)
TN (1) TNSN97118A1 (de)
UY (1) UY24609A1 (de)
WO (1) WO1998001435A1 (de)
ZA (1) ZA976071B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
US5750736A (en) * 1996-07-11 1998-05-12 Napro Biotherapeutics, Inc. Method for acylating 10-deacetylbaccatin III selectively at the c-10 position
US7288665B1 (en) 1997-08-18 2007-10-30 Florida State University Process for selective derivatization of taxanes

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2698871B1 (fr) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2702212B1 (fr) * 1993-03-02 1995-04-07 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2718135B1 (fr) * 1994-04-05 1996-04-26 Rhone Poulenc Rorer Sa Procédé de préparation d'hydroxy-7 taxanes.
FR2721023B1 (fr) * 1994-06-09 1996-07-12 Rhone Poulenc Rorer Sa Nouveaux Taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
ES2177988T3 (es) 2002-12-16
MA24258A1 (fr) 1998-04-01
FR2750989B1 (fr) 1998-09-25
DE69713098D1 (de) 2002-07-11
JP2000514082A (ja) 2000-10-24
AU3546997A (en) 1998-02-02
DK0912536T3 (da) 2002-09-16
FR2750989A1 (fr) 1998-01-16
PE69499A1 (es) 1999-10-15
US6127555A (en) 2000-10-03
CA2259278A1 (fr) 1998-01-15
PT912536E (pt) 2002-11-29
AR007834A1 (es) 1999-11-24
ATE218559T1 (de) 2002-06-15
TNSN97118A1 (fr) 2005-03-15
ZA976071B (en) 1998-02-02
CO4890872A1 (es) 2000-02-28
EP0912536B1 (de) 2002-06-05
UY24609A1 (es) 2001-08-27
EP0912536A1 (de) 1999-05-06
IN188980B (de) 2002-11-30
WO1998001435A1 (fr) 1998-01-15

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee