DE69317122D1 - Verfahren zur herstellung von triazolonderivaten - Google Patents
Verfahren zur herstellung von triazolonderivatenInfo
- Publication number
- DE69317122D1 DE69317122D1 DE69317122T DE69317122T DE69317122D1 DE 69317122 D1 DE69317122 D1 DE 69317122D1 DE 69317122 T DE69317122 T DE 69317122T DE 69317122 T DE69317122 T DE 69317122T DE 69317122 D1 DE69317122 D1 DE 69317122D1
- Authority
- DE
- Germany
- Prior art keywords
- pct
- date
- alkyl
- producing
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- FFSJPOPLSWBGQY-UHFFFAOYSA-N triazol-4-one Chemical class O=C1C=NN=N1 FFSJPOPLSWBGQY-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000003118 aryl group Chemical group 0.000 abstract 2
- -1 1,2,4-triazol-3-one compound Chemical group 0.000 abstract 1
- 150000007933 aliphatic carboxylic acids Chemical class 0.000 abstract 1
- WPYMKLBDIGXBTP-UHFFFAOYSA-N benzoic acid Chemical compound OC(=O)C1=CC=CC=C1 WPYMKLBDIGXBTP-UHFFFAOYSA-N 0.000 abstract 1
- KXDHJXZQYSOELW-UHFFFAOYSA-N carbonic acid monoamide Natural products NC(O)=O KXDHJXZQYSOELW-UHFFFAOYSA-N 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- KJAMZCVTJDTESW-UHFFFAOYSA-N tiracizine Chemical compound C1CC2=CC=CC=C2N(C(=O)CN(C)C)C2=CC(NC(=O)OCC)=CC=C21 KJAMZCVTJDTESW-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI922604A IT1256387B (it) | 1992-11-13 | 1992-11-13 | Procedimento per preparare triazoloni |
| PCT/EP1993/003119 WO1994011357A1 (en) | 1992-11-13 | 1993-11-06 | Process for the preparation of triazolone compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69317122D1 true DE69317122D1 (de) | 1998-04-02 |
| DE69317122T2 DE69317122T2 (de) | 1998-09-24 |
Family
ID=11364287
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69317122T Expired - Lifetime DE69317122T2 (de) | 1992-11-13 | 1993-11-06 | Verfahren zur herstellung von triazolonderivaten |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US5767275A (de) |
| EP (1) | EP0668857B1 (de) |
| AT (1) | ATE163414T1 (de) |
| AU (1) | AU5464394A (de) |
| DE (1) | DE69317122T2 (de) |
| DK (1) | DK0668857T3 (de) |
| ES (1) | ES2115916T3 (de) |
| IT (1) | IT1256387B (de) |
| WO (1) | WO1994011357A1 (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5625064A (en) * | 1995-04-19 | 1997-04-29 | Schering Corporation | Process for the preparation of triazolones |
| CA2182241C (en) * | 1996-07-29 | 2002-09-17 | Bo Lei | Methods for the manufacture of nefazodone |
| DE19816882A1 (de) * | 1998-04-17 | 1999-10-21 | Boehringer Ingelheim Pharma | Triazolone mit neuroprotektiver Wirkung |
| ES2152860B1 (es) * | 1998-10-23 | 2001-08-16 | Finaf 92 Sa | Forma cristalina de la nefazodona y procedimiento para su preparacion. |
| ES2262515T3 (es) | 1999-04-09 | 2006-12-01 | Sepracor Inc. | R-hidroxinefazodona. |
| JP2002541192A (ja) | 1999-04-09 | 2002-12-03 | セプラコール， インク． | Ｓ−ヒドロキシネファゾドン |
| WO2013134562A1 (en) | 2012-03-09 | 2013-09-12 | Inception 2, Inc. | Triazolone compounds and uses thereof |
| EP2935228B9 (de) | 2012-12-20 | 2017-12-06 | Inception 2, Inc. | Triazolonverbindungen und verwendungen davon |
| CA2921420A1 (en) | 2013-09-06 | 2015-03-12 | Inception 2, Inc. | Triazolone compounds and uses thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1545646B1 (de) * | 1965-12-15 | 1969-09-18 | Boehringer Sohn Ingelheim | 1,3-Dimethyl-4-(2',4'-dichlorphenyl)-1,2,4-triazolon-(5) und Verfahren zu dessen Herstellung |
| IT1052119B (it) * | 1972-10-16 | 1981-06-20 | Sigma Tau Ind Farmaceuti | Derivati del triazolinone e procedimento per la loro preparazione |
| US4338317A (en) * | 1981-03-16 | 1982-07-06 | Mead Johnson & Company | Phenoxyethyl-1,2,4,-triazol-3-one antidepressants |
| US4596884A (en) * | 1983-11-30 | 1986-06-24 | Bristol-Myers Company | 4-(2-phenoxyethyl)-1,2,4-triazolone process intermediates |
| US5094683A (en) * | 1988-05-09 | 1992-03-10 | Bayer Aktiengesellschaft | Sulphonylaminocarbonyltriazolinones |
-
1992
- 1992-11-13 IT ITMI922604A patent/IT1256387B/it active IP Right Grant
-
1993
- 1993-11-06 EP EP94900112A patent/EP0668857B1/de not_active Expired - Lifetime
- 1993-11-06 AU AU54643/94A patent/AU5464394A/en not_active Abandoned
- 1993-11-06 DE DE69317122T patent/DE69317122T2/de not_active Expired - Lifetime
- 1993-11-06 ES ES94900112T patent/ES2115916T3/es not_active Expired - Lifetime
- 1993-11-06 AT AT94900112T patent/ATE163414T1/de active
- 1993-11-06 US US08/424,477 patent/US5767275A/en not_active Expired - Lifetime
- 1993-11-06 WO PCT/EP1993/003119 patent/WO1994011357A1/en active IP Right Grant
- 1993-11-06 DK DK94900112T patent/DK0668857T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| IT1256387B (it) | 1995-12-04 |
| AU5464394A (en) | 1994-06-08 |
| ITMI922604A0 (it) | 1992-11-13 |
| ES2115916T3 (es) | 1998-07-01 |
| ATE163414T1 (de) | 1998-03-15 |
| US5767275A (en) | 1998-06-16 |
| EP0668857A1 (de) | 1995-08-30 |
| DK0668857T3 (da) | 1998-12-07 |
| ITMI922604A1 (it) | 1994-05-13 |
| WO1994011357A1 (en) | 1994-05-26 |
| DE69317122T2 (de) | 1998-09-24 |
| EP0668857B1 (de) | 1998-02-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |