DE68920493D1 - Verfahren zur Herstellung von Derivaten von 2'-Deoxy-beta-cytidin und Salze davon. - Google Patents

Verfahren zur Herstellung von Derivaten von 2'-Deoxy-beta-cytidin und Salze davon.

Info

Publication number
DE68920493D1
DE68920493D1 DE68920493T DE68920493T DE68920493D1 DE 68920493 D1 DE68920493 D1 DE 68920493D1 DE 68920493 T DE68920493 T DE 68920493T DE 68920493 T DE68920493 T DE 68920493T DE 68920493 D1 DE68920493 D1 DE 68920493D1
Authority
DE
Germany
Prior art keywords
cytidine
deoxy
beta
derivatives
salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE68920493T
Other languages
English (en)
Other versions
DE68920493T2 (de
Inventor
Hiroshi Life Science Kawakami
Hajime Life Science Matsushita
Nobuhiro C O Tokyo La Mizutani
Toshimi C O Tokyo La Takiguchi
Kazuo C O Tokyo Laborator Itoh
Yoshitake C O Tokyo Labor Naoi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
YUKI GOSEI YAKUHIN KOGYO KK
Japan Tobacco Inc
Original Assignee
YUKI GOSEI YAKUHIN KOGYO KK
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by YUKI GOSEI YAKUHIN KOGYO KK, Japan Tobacco Inc filed Critical YUKI GOSEI YAKUHIN KOGYO KK
Publication of DE68920493D1 publication Critical patent/DE68920493D1/de
Application granted granted Critical
Publication of DE68920493T2 publication Critical patent/DE68920493T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE68920493T 1988-07-05 1989-07-05 Verfahren zur Herstellung von Derivaten von 2'-Deoxy-beta-cytidin und Salze davon. Expired - Fee Related DE68920493T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP63166062A JPH0217198A (ja) 1988-07-05 1988-07-05 2’−デオキシ−β−シチジン誘導体およびその塩の製造法

Publications (2)

Publication Number Publication Date
DE68920493D1 true DE68920493D1 (de) 1995-02-23
DE68920493T2 DE68920493T2 (de) 1995-05-18

Family

ID=15824268

Family Applications (1)

Application Number Title Priority Date Filing Date
DE68920493T Expired - Fee Related DE68920493T2 (de) 1988-07-05 1989-07-05 Verfahren zur Herstellung von Derivaten von 2'-Deoxy-beta-cytidin und Salze davon.

Country Status (3)

Country Link
EP (1) EP0350293B1 (de)
JP (1) JPH0217198A (de)
DE (1) DE68920493T2 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0217199A (ja) * 1988-07-05 1990-01-22 Japan Tobacco Inc 2’−デオキシ−β−アデノシンの製造方法
JPH02289595A (ja) * 1989-02-22 1990-11-29 Yuki Gosei Kogyo Co Ltd 2’―デオキシ―5―トリフルオロメチル―β―ウリジンの製造方法
AU659008B2 (en) * 1992-06-22 1995-05-04 Eli Lilly And Company Stereoselective anion glycosylation process

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
GB1601020A (en) * 1978-04-24 1981-10-21 Stichting Grega Vzw 2'-deoxy-5 (2-halogenovinyl)-uridines
US4782142A (en) * 1982-01-05 1988-11-01 The Research Foundation Of State University Of New York Novel 5-substituted 2-pyrimidinone nucleosides and methods of use
CA1301166C (en) * 1987-07-21 1992-05-19 John Nicholas Freskos Process for preparing 2-deoxynucleosides

Also Published As

Publication number Publication date
EP0350293A3 (en) 1990-12-27
EP0350293A2 (de) 1990-01-10
DE68920493T2 (de) 1995-05-18
JPH0217198A (ja) 1990-01-22
EP0350293B1 (de) 1995-01-11

Similar Documents

Publication Publication Date Title
DE3887625T2 (de) Verfahren zur Herstellung von 1,1,1-Trifluorodichlorethan und von 1,1,1,2-Tetrafluorchlorethan.
DE68910145D1 (de) Verfahren zur Herstellung von Azolylmethyl-cyclopentanol-Derivaten.
DE68927703D1 (de) Verfahren zur Herstellung von 2,3-Dimethylbutenen
DE68927949T2 (de) 3,9-Diphosphaspiroundecane und Verfahren zur Herstellung von 3,9-Diphosphaspiroundecanen
DE68928619T2 (de) Verfahren zur Herstellung von mono-N-alkylierten Polyazamacrocyclen
DE68912160D1 (de) Verfahren zur Herstellung von beta-Lactamderivaten.
DE68925711D1 (de) Verfahren zur Herstellung von Alkadienolen
DE68925831D1 (de) Verfahren zur Herstellung von Cyanopyridinen
ATE76636T1 (de) Verfahren zur herstellung von benzoesaeure und ihren salzen.
DE69019052T2 (de) Verfahren zur Herstellung von 2'Deoxy-5-trifluoromethyl-ss-uridin.
DE69322127T2 (de) Verfahren zur Herstellung von Peptidderivaten und ihrer Salze
DE68915067T2 (de) Verfahren zur Herstellung von 2'-Deoxy-beta-adenosin.
DE69207051D1 (de) Substituierte Acetoxyazetidinonderivate und Verfahren zur Herstellung von 4-Acyloxyazetidinonderivate
DE68923159D1 (de) Verfahren zur Herstellung von 1,4-Dihydropyridin-Derivaten.
DE68920493T2 (de) Verfahren zur Herstellung von Derivaten von 2'-Deoxy-beta-cytidin und Salze davon.
DE68924093D1 (de) Verfahren zur Herstellung von 3-Exomethylencepham-Derivaten.
DE69217616D1 (de) Verfahren zur Herstellung von (S)-1-Phenyl-1,3-Propanediol und Derivaten
DE69012430D1 (de) Verfahren zur Herstellung von Sulfoniumverbindungen und Methylthiophenylderivaten.
DE68915904D1 (de) Verfahren zur Herstellung von Para-bromphenoxyacetaldehyd-dialkylacetal-Derivaten.
DE68922900T2 (de) Verfahren zur Herstellung von 2'-Deoxy-beta-adenosin.
DE68920755T2 (de) Verfahren zur Herstellung von alpha-Aspartyl-phenylalaninderivaten.
DE59209848D1 (de) Verfahren zur Herstellung von 2,4,5-Triamino-6-halogenopyrimidinen und 2-Amino-6-halogenopurinen
DE59201322D1 (de) Verfahren zur Herstellung von 3'-Aminopropyl-2-chlorethylsulfon-semisulfat.
DD279881A1 (de) Verfahren zur herstellung von 3,18-dihydroxy-9,13-epoxylabdanderivaten
DE68913685D1 (de) Verfahren zur Herstellung von 2,2'-Bis-defla2-oxazolin.

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee