DE60327220D1 - Benzolsulfonamide und verfahren zu ihrer herstellung - Google Patents

Benzolsulfonamide und verfahren zu ihrer herstellung

Info

Publication number
DE60327220D1
DE60327220D1 DE60327220T DE60327220T DE60327220D1 DE 60327220 D1 DE60327220 D1 DE 60327220D1 DE 60327220 T DE60327220 T DE 60327220T DE 60327220 T DE60327220 T DE 60327220T DE 60327220 D1 DE60327220 D1 DE 60327220D1
Authority
DE
Germany
Prior art keywords
formula
methoxy
benzyl
benzenesulphonamide
propyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60327220T
Other languages
English (en)
Inventor
Tibor Gizur
Jozsef Toerley
Elemer Fogassy
Jozsef Balint
Gabriella Egri
Adam Demeter
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richter Gedeon Nyrt
Original Assignee
Richter Gedeon Nyrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Nyrt filed Critical Richter Gedeon Nyrt
Application granted granted Critical
Publication of DE60327220D1 publication Critical patent/DE60327220D1/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE60327220T 2002-09-09 2003-09-08 Benzolsulfonamide und verfahren zu ihrer herstellung Expired - Fee Related DE60327220D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU0202963A HU225505B1 (en) 2002-09-09 2002-09-09 Process for the preparation of r-(-)-tamsulosin hydrochloride and novel intermediates
PCT/HU2003/000071 WO2004022532A1 (en) 2002-09-09 2003-09-08 Benzenesulphonamides and process for their preparation

Publications (1)

Publication Number Publication Date
DE60327220D1 true DE60327220D1 (de) 2009-05-28

Family

ID=89980754

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60327220T Expired - Fee Related DE60327220D1 (de) 2002-09-09 2003-09-08 Benzolsulfonamide und verfahren zu ihrer herstellung

Country Status (6)

Country Link
EP (1) EP1539684B1 (de)
AT (1) ATE428689T1 (de)
AU (1) AU2003263378A1 (de)
DE (1) DE60327220D1 (de)
HU (1) HU225505B1 (de)
WO (1) WO2004022532A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100545148C (zh) 2004-08-16 2009-09-30 神隆新加坡私人有限公司 一种抗良性前列腺肥大药物坦索罗辛之合成方法
US8273918B2 (en) 2005-09-12 2012-09-25 Avrobindo Pharma Ltd. Process for preparing tamsulosin hydrochloride

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1429306A (fr) * 1964-11-23 1966-02-25 Soc Ind Fab Antibiotiques Sifa Nouvelles benzylamines substituées et leurs sels, et procédé de préparation
US3860647A (en) * 1973-08-20 1975-01-14 Smithkline Corp {60 -Aminomethyl-4-hydroxy-3-sulfamyl-benzyl alcohols and 4-hydroxy-3-sulfamyl phenethylamines
JPH066565B2 (ja) * 1986-07-21 1994-01-26 山之内製薬株式会社 光学活性なベンゼンスルホンアミド誘導体の製造法
JP4342101B2 (ja) * 1998-02-27 2009-10-14 キッセイ薬品工業株式会社 インドール誘導体および当該誘導体を含有する医薬品組成物
JP2000029901A (ja) * 1998-07-14 2000-01-28 Canon Inc 画像検索装置及び方法

Also Published As

Publication number Publication date
HU0202963D0 (de) 2002-10-28
HU225505B1 (en) 2007-01-29
ATE428689T1 (de) 2009-05-15
AU2003263378A1 (en) 2004-03-29
EP1539684B1 (de) 2009-04-15
EP1539684A1 (de) 2005-06-15
WO2004022532A1 (en) 2004-03-18
HUP0202963A2 (hu) 2004-10-28

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee