DE60126831D1 - Benz(g)indole und deren verwendung als spla2 inhibitoren - Google Patents
Benz(g)indole und deren verwendung als spla2 inhibitorenInfo
- Publication number
- DE60126831D1 DE60126831D1 DE60126831T DE60126831T DE60126831D1 DE 60126831 D1 DE60126831 D1 DE 60126831D1 DE 60126831 T DE60126831 T DE 60126831T DE 60126831 T DE60126831 T DE 60126831T DE 60126831 D1 DE60126831 D1 DE 60126831D1
- Authority
- DE
- Germany
- Prior art keywords
- benz
- indole
- spla2 inhibitors
- compounds
- spla2
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/58—[b]- or [c]-condensed
- C07D209/60—Naphtho [b] pyrroles; Hydrogenated naphtho [b] pyrroles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25629400P | 2000-12-18 | 2000-12-18 | |
PCT/US2001/043182 WO2002057231A2 (en) | 2000-12-18 | 2001-12-06 | Benz(g) indoles and their use as spla2 inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
DE60126831D1 true DE60126831D1 (de) | 2007-04-05 |
Family
ID=22971699
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60126831T Expired - Lifetime DE60126831D1 (de) | 2000-12-18 | 2001-12-06 | Benz(g)indole und deren verwendung als spla2 inhibitoren |
Country Status (8)
Country | Link |
---|---|
US (1) | US6916840B2 (de) |
EP (1) | EP1358156B1 (de) |
JP (1) | JP2004520363A (de) |
AT (1) | ATE354567T1 (de) |
AU (1) | AU2002245019A1 (de) |
CA (1) | CA2431506A1 (de) |
DE (1) | DE60126831D1 (de) |
WO (1) | WO2002057231A2 (de) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2424521A4 (de) | 2009-04-29 | 2015-03-04 | Amarin Pharmaceuticals Ie Ltd | Pharmazeutische zusammensetzungen mit epa und einem kardiovaskulären mittel sowie verwendungsverfahren dafür |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL109311A0 (en) * | 1993-04-16 | 1994-07-31 | Lilly Co Eli | 1H-indole-3-acetamide sPla2 inhibitors |
CN1067054C (zh) | 1994-04-01 | 2001-06-13 | 伊莱利利公司 | 1H-吲哚-3-乙醛酰胺sPLA2抑制剂 |
AU2373600A (en) | 1998-12-22 | 2000-07-12 | Eli Lilly And Company | Novel spla2 inhibitors |
-
2001
- 2001-12-06 CA CA002431506A patent/CA2431506A1/en not_active Abandoned
- 2001-12-06 WO PCT/US2001/043182 patent/WO2002057231A2/en active IP Right Grant
- 2001-12-06 AT AT01993161T patent/ATE354567T1/de not_active IP Right Cessation
- 2001-12-06 EP EP01993161A patent/EP1358156B1/de not_active Expired - Lifetime
- 2001-12-06 AU AU2002245019A patent/AU2002245019A1/en not_active Abandoned
- 2001-12-06 JP JP2002557912A patent/JP2004520363A/ja active Pending
- 2001-12-06 US US10/450,860 patent/US6916840B2/en not_active Expired - Fee Related
- 2001-12-06 DE DE60126831T patent/DE60126831D1/de not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP1358156B1 (de) | 2007-02-21 |
CA2431506A1 (en) | 2002-07-25 |
US20040063967A1 (en) | 2004-04-01 |
JP2004520363A (ja) | 2004-07-08 |
AU2002245019A1 (en) | 2002-07-30 |
US6916840B2 (en) | 2005-07-12 |
WO2002057231A3 (en) | 2003-01-09 |
WO2002057231A2 (en) | 2002-07-25 |
EP1358156A2 (de) | 2003-11-05 |
ATE354567T1 (de) | 2007-03-15 |
WO2002057231A8 (en) | 2003-11-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE540923T1 (de) | Ää3-(2-amino-1,2-dioxoethyl)-2-ethyl-1- (phenylmethyl)-11h-indol-4-ylüoxyüessigsäure methyl ester als spla2 inhibitor | |
ATE246501T1 (de) | Pyrrole als spla2 inhibitoren | |
ATE326963T1 (de) | Indolverbindungen als spla2 inhibitoren | |
WO2002050030A8 (en) | Cycloalkylfused [g]-indole compounds as spla2-inhibitors in the treatment of inflammatory diseases | |
ATE234850T1 (de) | Phenylglyoxamide als spla2-inhibitoren | |
ATE312817T1 (de) | Cyclohept'bö indolderivate als spla2-inhibitoren | |
DE60032774D1 (de) | Spla2 inhibitoren | |
DE60126831D1 (de) | Benz(g)indole und deren verwendung als spla2 inhibitoren | |
WO2002012249A3 (en) | Substituted pyrrole compounds and their use as spla2 inhibitors | |
DE60032254D1 (de) | Hydroxyfunktionelle amid-1h-indolderivate aktiv als spla2 inhibitoren | |
DE69910432D1 (de) | Substituierte pyrroloindole | |
WO2002050028A8 (en) | Substituted benzoindoles as spla2 inhibitors | |
WO2001049662A3 (en) | Carbazole derivatives as inhibitors of spla2 | |
ATE329905T1 (de) | Tetracyclische derivate als spla2 inhibitoren |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8332 | No legal effect for de |