ATE354567T1 - Benz(g)indole und deren verwendung als spla2 inhibitoren - Google Patents

Benz(g)indole und deren verwendung als spla2 inhibitoren

Info

Publication number
ATE354567T1
ATE354567T1 AT01993161T AT01993161T ATE354567T1 AT E354567 T1 ATE354567 T1 AT E354567T1 AT 01993161 T AT01993161 T AT 01993161T AT 01993161 T AT01993161 T AT 01993161T AT E354567 T1 ATE354567 T1 AT E354567T1
Authority
AT
Austria
Prior art keywords
benz
indole
spla2 inhibitors
compounds
spla2
Prior art date
Application number
AT01993161T
Other languages
English (en)
Inventor
Douglas Wade Beight
Michael Dean Kinnick
Ho-Shen Lin
John Michael Junior Morin
Michael Enrico Richett
Daniel Jon Sall
Jason Scott Sawyer
Edward C R Smith
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of ATE354567T1 publication Critical patent/ATE354567T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/58—[b]- or [c]-condensed
    • C07D209/60—Naphtho [b] pyrroles; Hydrogenated naphtho [b] pyrroles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT01993161T 2000-12-18 2001-12-06 Benz(g)indole und deren verwendung als spla2 inhibitoren ATE354567T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25629400P 2000-12-18 2000-12-18

Publications (1)

Publication Number Publication Date
ATE354567T1 true ATE354567T1 (de) 2007-03-15

Family

ID=22971699

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01993161T ATE354567T1 (de) 2000-12-18 2001-12-06 Benz(g)indole und deren verwendung als spla2 inhibitoren

Country Status (8)

Country Link
US (1) US6916840B2 (de)
EP (1) EP1358156B1 (de)
JP (1) JP2004520363A (de)
AT (1) ATE354567T1 (de)
AU (1) AU2002245019A1 (de)
CA (1) CA2431506A1 (de)
DE (1) DE60126831D1 (de)
WO (1) WO2002057231A2 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2424521A4 (de) 2009-04-29 2015-03-04 Amarin Pharmaceuticals Ie Ltd Pharmazeutische zusammensetzungen mit epa und einem kardiovaskulären mittel sowie verwendungsverfahren dafür

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL109311A0 (en) * 1993-04-16 1994-07-31 Lilly Co Eli 1H-indole-3-acetamide sPla2 inhibitors
CO4370099A1 (es) * 1994-04-01 1996-10-07 Lilly Co Eli 1H-INDOL-3-GLIOXILAMIDAS INHIBIDORAS DE sPLA2
US6391908B1 (en) 1998-12-22 2002-05-21 Eli Lilly And Company Oxime amide indole type sPLA2 inhibitors

Also Published As

Publication number Publication date
WO2002057231A3 (en) 2003-01-09
EP1358156A2 (de) 2003-11-05
WO2002057231A8 (en) 2003-11-13
WO2002057231A2 (en) 2002-07-25
DE60126831D1 (de) 2007-04-05
US20040063967A1 (en) 2004-04-01
CA2431506A1 (en) 2002-07-25
JP2004520363A (ja) 2004-07-08
US6916840B2 (en) 2005-07-12
AU2002245019A1 (en) 2002-07-30
EP1358156B1 (de) 2007-02-21

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties