DE60026350D1 - Diaryl piperidyl-pyrrol-derivate als antiprotozoenmittel - Google Patents
Diaryl piperidyl-pyrrol-derivate als antiprotozoenmittelInfo
- Publication number
- DE60026350D1 DE60026350D1 DE60026350T DE60026350T DE60026350D1 DE 60026350 D1 DE60026350 D1 DE 60026350D1 DE 60026350 T DE60026350 T DE 60026350T DE 60026350 T DE60026350 T DE 60026350T DE 60026350 D1 DE60026350 D1 DE 60026350D1
- Authority
- DE
- Germany
- Prior art keywords
- tozenes
- antiprotro
- diaryl
- piperidyl
- pyrrol derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/116—Heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K50/00—Feeding-stuffs specially adapted for particular animals
- A23K50/70—Feeding-stuffs specially adapted for particular animals for birds
- A23K50/75—Feeding-stuffs specially adapted for particular animals for birds for poultry
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Polymers & Plastics (AREA)
- Animal Husbandry (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- Birds (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US16514299P | 1999-11-12 | 1999-11-12 | |
US165142P | 1999-11-12 | ||
PCT/US2000/030747 WO2001034149A1 (en) | 1999-11-12 | 2000-11-09 | Diaryl piperidyl pyrrole derivatives as antiprotozoal agents |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60026350D1 true DE60026350D1 (de) | 2006-04-27 |
DE60026350T2 DE60026350T2 (de) | 2006-11-09 |
Family
ID=22597609
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60026350T Expired - Lifetime DE60026350T2 (de) | 1999-11-12 | 2000-11-09 | Diaryl piperidyl-pyrrol-derivate als antiprotozoenmittel |
Country Status (11)
Country | Link |
---|---|
US (2) | US6291480B1 (de) |
EP (1) | EP1278520B1 (de) |
JP (1) | JP4722360B2 (de) |
AT (1) | ATE318600T1 (de) |
AU (1) | AU781552B2 (de) |
CA (1) | CA2390100C (de) |
DE (1) | DE60026350T2 (de) |
ES (1) | ES2257336T3 (de) |
NZ (1) | NZ518718A (de) |
WO (1) | WO2001034149A1 (de) |
ZA (1) | ZA200203685B (de) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU1596101A (en) * | 1999-11-12 | 2001-06-06 | Merck & Co., Inc. | Aliphatic amine substituted piperidyl diaryl pyrrole derivatives as antiprotozoal agents |
CN1526011A (zh) * | 2001-07-10 | 2004-09-01 | IDECҩ�﹫˾ | 抑制凋亡过程及改善细胞性能 |
WO2003022838A1 (en) * | 2001-09-05 | 2003-03-20 | Smithkline Beecham Plc | Pyridine substituted furan derivatives as raf kinase inhibitors |
BRPI0411221A (pt) * | 2003-06-11 | 2006-07-18 | Sankyo Co | composto, medicamento, métodos para inibir a produção de citocinas inflamatórias, e para a prevenção ou tratamento de doenças associadas com citocinas inflamatórias, método para o tratamento ou alìvio de febre, dor e/ou inflamação e, métodos para a prevenção ou tratamento de artrite reumatóide, de osteoartrite, de doença septicêmica, psorìase, doença de crohn, colite ulcerativa, diabete melito ou, hepatite |
NZ568694A (en) | 2005-11-09 | 2011-09-30 | Zalicus Inc | Method, compositions, and kits for the treatment of medical conditions |
MX359921B (es) * | 2013-02-08 | 2018-10-16 | Luoda Pharma Pty Ltd | Métodos de tratamiento tópico para infecciones microbianas. |
RU2659205C1 (ru) * | 2017-06-01 | 2018-06-28 | Федеральное государственное бюджетное научное учреждение "Прикаспийский зональный научно-исследовательский ветеринарный институт" | Способ профилактики кокцидиоза цыплят-бройлеров при выращивании их на мясо |
BE1028700B1 (nl) * | 2020-10-13 | 2022-05-16 | Poulpharm Bvba | Werkwijze voor het testen van de efficiëntie van anti-parasitaire (coccidiose) middelen bij pluimvee en konijnen |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4153703A (en) * | 1977-06-30 | 1979-05-08 | Uniroyal, Inc. | Method of controlling insects and acarids with certain aryl-substituted thiazoles |
WO1996017841A1 (fr) * | 1994-12-06 | 1996-06-13 | Nippon Soda Co., Ltd. | Composes de pyridylpyrrole, processus de production et bactericide agro-horticole |
US5792778A (en) * | 1995-08-10 | 1998-08-11 | Merck & Co., Inc. | 2-substituted aryl pyrroles, compositions containing such compounds and methods of use |
JP3294616B2 (ja) * | 1995-08-10 | 2002-06-24 | メルク エンド カンパニー インコーポレーテッド | 2−置換アリールピロール、このような化合物を含む組成物及び使用方法 |
WO1997016426A1 (en) * | 1995-10-31 | 1997-05-09 | Merck & Co., Inc. | Substituted aryl pyrroles, compositions containing such compounds and methods of use |
JPH09194477A (ja) * | 1996-01-18 | 1997-07-29 | Nippon Soda Co Ltd | 新規なピリジルピロール化合物、製法および農園芸用殺菌剤 |
WO1997048725A1 (en) * | 1996-06-21 | 1997-12-24 | Peptech Limited | Novel peptides for prevention and treatment of infection |
JP2000080094A (ja) * | 1998-07-02 | 2000-03-21 | Sankyo Co Ltd | 5員ヘテロアリ―ル化合物 |
WO2000001688A1 (fr) * | 1998-07-02 | 2000-01-13 | Sankyo Company, Limited | Composes heteroaryle a cinq elements |
AU4315100A (en) * | 1999-04-28 | 2000-11-17 | Sankyo Company Limited | Preventive or inhibitory agents for hepatopathy |
JP2001010957A (ja) * | 1999-04-28 | 2001-01-16 | Sankyo Co Ltd | 肝障害の予防または抑制剤 |
-
2000
- 2000-11-09 JP JP2001536147A patent/JP4722360B2/ja not_active Expired - Lifetime
- 2000-11-09 AU AU15904/01A patent/AU781552B2/en not_active Ceased
- 2000-11-09 ES ES00978439T patent/ES2257336T3/es not_active Expired - Lifetime
- 2000-11-09 DE DE60026350T patent/DE60026350T2/de not_active Expired - Lifetime
- 2000-11-09 EP EP00978439A patent/EP1278520B1/de not_active Expired - Lifetime
- 2000-11-09 AT AT00978439T patent/ATE318600T1/de not_active IP Right Cessation
- 2000-11-09 CA CA002390100A patent/CA2390100C/en not_active Expired - Lifetime
- 2000-11-09 NZ NZ518718A patent/NZ518718A/en not_active IP Right Cessation
- 2000-11-09 WO PCT/US2000/030747 patent/WO2001034149A1/en active IP Right Grant
- 2000-11-10 US US09/710,147 patent/US6291480B1/en not_active Expired - Lifetime
- 2000-11-10 US US09/709,959 patent/US6384052B1/en not_active Expired - Lifetime
-
2002
- 2002-05-09 ZA ZA200203685A patent/ZA200203685B/en unknown
Also Published As
Publication number | Publication date |
---|---|
NZ518718A (en) | 2004-03-26 |
DE60026350T2 (de) | 2006-11-09 |
ES2257336T3 (es) | 2006-08-01 |
JP2003527336A (ja) | 2003-09-16 |
CA2390100A1 (en) | 2001-05-17 |
CA2390100C (en) | 2010-01-05 |
WO2001034149A1 (en) | 2001-05-17 |
EP1278520B1 (de) | 2006-03-01 |
AU1590401A (en) | 2001-06-06 |
JP4722360B2 (ja) | 2011-07-13 |
US6291480B1 (en) | 2001-09-18 |
ZA200203685B (en) | 2003-06-05 |
EP1278520A1 (de) | 2003-01-29 |
US6384052B1 (en) | 2002-05-07 |
ATE318600T1 (de) | 2006-03-15 |
EP1278520A4 (de) | 2003-05-02 |
AU781552B2 (en) | 2005-05-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8327 | Change in the person/name/address of the patent owner |
Owner name: MERCK & CO., INC., RAHWAY, N.J., US |
|
8327 | Change in the person/name/address of the patent owner |
Owner name: MERCK SHARP & DOHME CORP., NEW JERSEY, N.J., US |
|
R081 | Change of applicant/patentee |
Ref document number: 1278520 Country of ref document: EP Owner name: SCHERING CORPORATION, US Free format text: FORMER OWNER: MERCK SHARP & DOHME CORP., 07065-0900 RAHWAY, US Effective date: 20121213 |
|
R082 | Change of representative |
Ref document number: 1278520 Country of ref document: EP Representative=s name: ABITZ & PARTNER, DE Effective date: 20121213 |