DE3566611D1 - Lysine esters used as absorption enhancing agents - Google Patents
Lysine esters used as absorption enhancing agentsInfo
- Publication number
- DE3566611D1 DE3566611D1 DE8585400771T DE3566611T DE3566611D1 DE 3566611 D1 DE3566611 D1 DE 3566611D1 DE 8585400771 T DE8585400771 T DE 8585400771T DE 3566611 T DE3566611 T DE 3566611T DE 3566611 D1 DE3566611 D1 DE 3566611D1
- Authority
- DE
- Germany
- Prior art keywords
- enhancing agents
- esters used
- absorption enhancing
- lysine esters
- lysine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0031—Rectum, anus
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Emergency Medicine (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/604,349 US4749694A (en) | 1984-04-26 | 1984-04-26 | Novel lysine esters used as absorption |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3566611D1 true DE3566611D1 (en) | 1989-01-12 |
Family
ID=24419249
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8585400771T Expired DE3566611D1 (en) | 1984-04-26 | 1985-04-18 | Lysine esters used as absorption enhancing agents |
Country Status (4)
Country | Link |
---|---|
US (1) | US4749694A (de) |
EP (1) | EP0162747B1 (de) |
JP (1) | JPS60233041A (de) |
DE (1) | DE3566611D1 (de) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4729989A (en) * | 1985-06-28 | 1988-03-08 | Merck & Co., Inc. | Enhancement of absorption of drugs from gastrointestinal tract using choline ester salts |
US4994451A (en) * | 1988-01-19 | 1991-02-19 | Bristol-Myers Company | Cephalosporin salts and injectable compositions |
US4910301A (en) * | 1985-08-05 | 1990-03-20 | Bristol-Myers Company | Cefepime cephalosporin salts |
US5244891A (en) * | 1985-08-05 | 1993-09-14 | Bristol-Myers Squibb Company | Injectable compositions of cefepime dihydrochloride hydrate |
IT1233836B (it) * | 1988-01-13 | 1992-04-21 | Euroresearch Srl | Sali idrosolubili dell'acido (+)2-(4 fluorofenil)-alfa-metil-5 benzoxazolo acetato. |
DE3806852A1 (de) * | 1988-03-03 | 1989-09-14 | Knoll Ag | Neue (alpha)-aminodicarbonsaeure-derivate, ihre herstellung und verwendung |
US8987263B2 (en) * | 2002-10-10 | 2015-03-24 | Meir Shinitzky | Basic esters of fatty alcohols and their use as anti-inflammatory or immunomodulatory agents |
US7151092B2 (en) * | 2002-10-31 | 2006-12-19 | Metabasis Therapeutics, Inc. | Cytarabine monophosphate prodrugs |
FR2925491B1 (fr) * | 2007-12-19 | 2010-09-03 | Oz Biosciences Sas | Nouvelle classe de lipides cationiques pour le transport d'agents actifs dans les cellules |
JP6030630B2 (ja) * | 2011-04-14 | 2016-11-24 | ノヴォ ノルディスク アー/エス | 経口ペプチド送達のための脂肪酸アシル化アミノ酸 |
AU2015217221A1 (en) | 2014-02-13 | 2016-08-11 | Ligand Pharmaceuticals, Inc. | Prodrug compounds and their uses |
EP3164136A4 (de) | 2014-07-02 | 2018-04-04 | Ligand Pharmaceuticals, Inc. | Prodrug-verbindungen und verwendungen davon |
US9920003B2 (en) * | 2014-08-19 | 2018-03-20 | Archer Daniels Midland Company | Non-ionic amphiphiles and methods of making the same |
AU2019207625A1 (en) | 2018-01-09 | 2020-07-30 | Ligand Pharmaceuticals, Inc. | Acetal compounds and therapeutic uses thereof |
EP4051258A4 (de) * | 2019-10-29 | 2024-01-10 | Tranexamic Technologies, LLC | Synergistische kombinationen von synthetischen lysinanaloga, derivaten, mimetika oder prodrugs und pharmazeutischen mitteln zur verbesserten wirksamkeit |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL272185A (de) * | 1960-12-05 | |||
CH448122A (de) * | 1963-10-14 | 1967-12-15 | Hoffmann La Roche | Verfahren zur Herstellung von Estern |
JPS5339410B2 (de) * | 1973-12-21 | 1978-10-21 | ||
US4154956A (en) * | 1973-12-21 | 1979-05-15 | Toray Industries, Inc. | Method for producing lysine ester |
GB1476432A (en) * | 1974-12-05 | 1977-06-16 | Beecham Group Ltd | Pharmaceutical compositions containing penicillin salts |
GB1477672A (en) * | 1975-01-30 | 1977-06-22 | Beecham Group Ltd | Penicillin compositions |
DE2742411B1 (de) * | 1977-09-21 | 1979-01-18 | Beiersdorf Ag | Zahn- und Mundpflegemittel |
JPS5767513A (en) * | 1980-10-14 | 1982-04-24 | Asahi Chem Ind Co Ltd | Novel drug composition for rectal administration |
-
1984
- 1984-04-26 US US06/604,349 patent/US4749694A/en not_active Expired - Fee Related
-
1985
- 1985-04-18 DE DE8585400771T patent/DE3566611D1/de not_active Expired
- 1985-04-18 EP EP85400771A patent/EP0162747B1/de not_active Expired
- 1985-04-26 JP JP60089123A patent/JPS60233041A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
US4749694A (en) | 1988-06-07 |
JPS60233041A (ja) | 1985-11-19 |
EP0162747B1 (de) | 1988-12-07 |
EP0162747A1 (de) | 1985-11-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |