DE3483308D1 - Semicarbazid-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen. - Google Patents

Semicarbazid-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.

Info

Publication number
DE3483308D1
DE3483308D1 DE8484114005T DE3483308T DE3483308D1 DE 3483308 D1 DE3483308 D1 DE 3483308D1 DE 8484114005 T DE8484114005 T DE 8484114005T DE 3483308 T DE3483308 T DE 3483308T DE 3483308 D1 DE3483308 D1 DE 3483308D1
Authority
DE
Germany
Prior art keywords
production
pharmaceutical compositions
compositions containing
semicarbazide derivatives
semicarbazide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE8484114005T
Other languages
English (en)
Inventor
Osamu Nakaguchi
Norihiko Shimazaki
Yoshio Kawai
Masashi Hashimoto
Michie Nakatuka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838330978A external-priority patent/GB8330978D0/en
Priority claimed from GB848417453A external-priority patent/GB8417453D0/en
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE3483308D1 publication Critical patent/DE3483308D1/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D203/00Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/26Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/04Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/28Nitrogen atoms
    • C07D295/32Nitrogen atoms acylated with carboxylic or carbonic acids, or their nitrogen or sulfur analogues
DE8484114005T 1983-11-21 1984-11-20 Semicarbazid-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen. Expired - Fee Related DE3483308D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838330978A GB8330978D0 (en) 1983-11-21 1983-11-21 Semicarbazide derivatives
GB848417453A GB8417453D0 (en) 1984-07-09 1984-07-09 Semicarbazide derivatives

Publications (1)

Publication Number Publication Date
DE3483308D1 true DE3483308D1 (de) 1990-10-31

Family

ID=26287019

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8484114005T Expired - Fee Related DE3483308D1 (de) 1983-11-21 1984-11-20 Semicarbazid-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.

Country Status (3)

Country Link
US (1) US4725608A (de)
EP (1) EP0144853B1 (de)
DE (1) DE3483308D1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4866173A (en) * 1982-09-22 1989-09-12 Rorer Pharmaceutical Corporation Therapeutic substituted semicarbazides
US4694004A (en) * 1984-07-09 1987-09-15 Fujisawa Pharmaceutical Co., Ltd. Semicarbazide derivatives, processes for preparation thereof and pharmaceutical composition comprising the same
ES2089056T3 (es) * 1990-06-16 1996-10-01 Nihon Nohyaku Co Ltd Derivados de hidrazincarboxamida, un procedimiento para la produccion de los mismos, y usos de los mismos.
MY105495A (en) * 1990-12-27 1994-10-31 Otsuka Kagaku Kk Novel process for producing semicarbazide.
DE69842004D1 (de) 1997-11-21 2010-12-30 Purdue Neuroscience Co Substituierte 2-aminoacetamide und anwendung davon
GB9727523D0 (en) 1997-12-31 1998-02-25 Pharmacia & Upjohn Spa Alpha-aminoamide derivatives useful as analgesic agents
CA2319484A1 (en) * 1998-02-04 1999-08-12 Euro-Celtique S.A. Substituted semicarbazides and the use thereof
SE9802209D0 (sv) 1998-06-22 1998-06-22 Astra Pharma Inc Novel compounds
US6281211B1 (en) 1999-02-04 2001-08-28 Euro-Celtique S.A. Substituted semicarbazides and the use thereof
KR100343266B1 (ko) * 1999-06-28 2002-07-10 주식회사 동진쎄미켐 세미카바자이드 합성방법
MXPA04002009A (es) * 2001-09-03 2004-07-08 Newron Pharm Spa Composicion farmaceutica que comprende gabapentina o un analogo de la misma y alfa-aminoamida y su uso como analgesico.
EP1438956A1 (de) * 2003-01-16 2004-07-21 Newron Pharmaceuticals S.p.A. Alpha-Aminoamidderivate die als Antimigränemittel nützlich sind
JP5319920B2 (ja) * 2004-09-10 2013-10-16 ニユーロン・フアーマシユーテイカルズ・エツセ・ピー・アー ナトリウムおよび/またはカルシウムチャンネル選択的調節因子として活性のある医薬の製造のための(ハロベンジルオキシ)ベンジルアミノ−プロパンアミドの使用

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3318680A (en) * 1961-10-24 1967-05-09 Du Pont Method for the control of weeds
US3285957A (en) * 1964-02-13 1966-11-15 Monsanto Co Diphenyl semicarbazides
FR1521959A (fr) * 1966-05-07 1968-04-19 Basf Ag Dérivés de semicarbazides et mélanges herbicides renfermant ces dérivés
CH480309A (de) * 1966-08-11 1969-10-31 Ciba Geigy Verfahren zur Herstellung von Thiosemicarbazidverbindungen
CH480308A (de) * 1966-08-11 1969-10-31 Ciba Geigy Verfahren zur Herstellung von Thiosemicarbazid-Verbindungen
US3511875A (en) * 1968-04-12 1970-05-12 Du Pont Herbicidal alkylcarbamoyloxy semicarbazides
IL38138A (en) * 1970-11-19 1974-07-31 Ciba Geigy Ag Process and compositions containing thiourea derivatives for the promotion of fruit abscission
DE2221812A1 (de) * 1972-05-04 1973-11-15 Bayer Ag Verfahren zur herstellung von thiosemicarbaziden
US4013669A (en) * 1973-01-05 1977-03-22 Fisons Limited Ester-pyridinium compounds as acaricides
US4088653A (en) * 1976-08-23 1978-05-09 Canadian Patents And Developments Limited Tetrahydropyridyl derivatives
GB1574019A (en) * 1977-01-14 1980-09-03 Joullie International Sa Therapeutically useful 3,4,5-trimethoxybenzene derivatives
IT1141008B (it) * 1979-09-10 1986-10-01 Energy Conversion Devices Inc Composizione a base di tellurio per la formazione di immagini

Also Published As

Publication number Publication date
EP0144853B1 (de) 1990-09-26
US4725608A (en) 1988-02-16
EP0144853A3 (en) 1986-01-29
EP0144853A2 (de) 1985-06-19

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee