DE3364524D1 - Polymorphic forms of 5-(3-(2-(2,2,2-trifluoroethyl)-guanidino)-pyrazol-1-yl) valeramide - Google Patents
Polymorphic forms of 5-(3-(2-(2,2,2-trifluoroethyl)-guanidino)-pyrazol-1-yl) valeramideInfo
- Publication number
- DE3364524D1 DE3364524D1 DE8383304851T DE3364524T DE3364524D1 DE 3364524 D1 DE3364524 D1 DE 3364524D1 DE 8383304851 T DE8383304851 T DE 8383304851T DE 3364524 T DE3364524 T DE 3364524T DE 3364524 D1 DE3364524 D1 DE 3364524D1
- Authority
- DE
- Germany
- Prior art keywords
- valeramide
- guanidino
- pyrazol
- trifluoroethyl
- polymorphic forms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8225154 | 1982-09-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE3364524D1 true DE3364524D1 (en) | 1986-08-21 |
Family
ID=10532675
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE8383304851T Expired DE3364524D1 (en) | 1982-09-03 | 1983-08-23 | Polymorphic forms of 5-(3-(2-(2,2,2-trifluoroethyl)-guanidino)-pyrazol-1-yl) valeramide |
Country Status (21)
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8401751D0 (en) * | 1984-01-24 | 1984-02-29 | Ici Plc | Guanidine derivatives |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1233818A (en) * | 1981-03-09 | 1988-03-08 | David J. Gilman | Guanidine derivatives as histamine h-2 receptor antagonists |
-
1983
- 1983-08-02 GB GB838320820A patent/GB8320820D0/en active Pending
- 1983-08-09 IE IE1874/83A patent/IE55805B1/xx unknown
- 1983-08-11 AU AU17897/83A patent/AU1789783A/en not_active Abandoned
- 1983-08-19 DK DK3800/83A patent/DK380083D0/da not_active Application Discontinuation
- 1983-08-21 IL IL69533A patent/IL69533A/xx unknown
- 1983-08-22 ZA ZA836196A patent/ZA836196B/xx unknown
- 1983-08-23 AT AT83304851T patent/ATE20740T1/de not_active IP Right Cessation
- 1983-08-23 EP EP83304851A patent/EP0115114B1/en not_active Expired
- 1983-08-23 DE DE8383304851T patent/DE3364524D1/de not_active Expired
- 1983-08-30 FI FI833074A patent/FI833074L/fi not_active Application Discontinuation
- 1983-08-30 JP JP58157272A patent/JPS5965079A/ja active Pending
- 1983-08-31 HU HU833030A patent/HU191091B/hu unknown
- 1983-09-01 GR GR72356A patent/GR78940B/el unknown
- 1983-09-01 PT PT77278A patent/PT77278B/pt unknown
- 1983-09-01 NZ NZ205451A patent/NZ205451A/xx unknown
- 1983-09-02 SU SU833641101A patent/SU1237080A3/ru active
- 1983-09-02 ES ES525329A patent/ES525329A0/es active Granted
- 1983-09-02 NO NO833147A patent/NO833147L/no unknown
- 1983-09-02 DD DD83254489A patent/DD211342A5/de unknown
- 1983-09-02 CA CA000435933A patent/CA1198734A/en not_active Expired
- 1983-09-02 CS CS836396A patent/CS236893B2/cs unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5965079A (ja) | 1984-04-13 |
| ZA836196B (en) | 1984-07-25 |
| ATE20740T1 (de) | 1986-08-15 |
| GR78940B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1984-10-02 |
| DK380083D0 (da) | 1983-08-19 |
| SU1237080A3 (ru) | 1986-06-07 |
| FI833074A7 (fi) | 1984-03-04 |
| ES8505738A1 (es) | 1985-06-01 |
| HU191091B (en) | 1987-01-28 |
| FI833074A0 (fi) | 1983-08-30 |
| EP0115114B1 (en) | 1986-07-16 |
| AU1789783A (en) | 1984-03-08 |
| GB8320820D0 (en) | 1983-09-01 |
| PT77278A (en) | 1983-10-01 |
| FI833074L (fi) | 1984-03-04 |
| NZ205451A (en) | 1985-07-31 |
| CS236893B2 (en) | 1985-05-15 |
| PT77278B (en) | 1986-03-18 |
| ES525329A0 (es) | 1985-06-01 |
| EP0115114A1 (en) | 1984-08-08 |
| IE831874L (en) | 1984-03-03 |
| CA1198734A (en) | 1985-12-31 |
| IE55805B1 (en) | 1991-01-16 |
| NO833147L (no) | 1984-03-05 |
| IL69533A (en) | 1987-12-31 |
| DD211342A5 (de) | 1984-07-11 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES514587A0 (es) | Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico. | |
| NO152091C (no) | Analogifremgangsmaate ved fremstilling av antiinflammatorisk virksomme 5-substituerte 2,3-difenylthiofener | |
| NO156694C (no) | Analogifremgangsmaate ved fremstilling av terapeutisk aktive 10-(1,2-propadienyl)-steroider. | |
| ES513314A0 (es) | "procedimiento para la fabricacion de 1,5-disubstituido 1,2,4-triazol-3- carbamida". | |
| NO164472C (no) | Analogifremgangsmaate ved fremstilling av terapeutisk aktive substituerte 2-(monokondenserte (3,4- og 5,6)-pyridylalkylensulfinyl)-benzimidazoler. | |
| DE3364524D1 (en) | Polymorphic forms of 5-(3-(2-(2,2,2-trifluoroethyl)-guanidino)-pyrazol-1-yl) valeramide | |
| NO152697C (no) | Analogifremgangsmaate ved fremstilling av terapeutisk aktive 5-(klorfenyl)-6h-1,3,4-thiadiazin-2-aminer. | |
| DK439082A (da) | 4-acylamino-1-aza-adamantan-forbindelser samt fremgangsmaade til fremstilling deraf | |
| TR23271A (tr) | En asagi % 95.5 safliginda p-ksilol'un kazanilmasina mahsus usul | |
| IT1145279B (it) | Procedimento per la produzione di 3-(4)-formiltriciclo(5,2,1,0,2,6)-decene-8 | |
| NO153572C (no) | Analogifremgangsm¨te ved fremstilling av terapeutisk aktiv e 5-(2-(2,3-dihydro-1,4-benzodioxan-2-ylmethyl)-amino)-1-h ydroxyethyl)-2-hydroxybenzoesyre-derivater. | |
| AT362502B (de) | Verfahren zur herstellung von 7-(d-(-)-alpha- -(4-aethyl-2,3-dioxo-1-piperazincarboxamido)- -alpha-(4-hydroxyphenyl)-acetamido)-3-(5-(1- -methyl-1,2,3,4-tetrazolyl)-thiomethyl)-delta 3 -cephem-4-carbonsaeure | |
| ATE15193T1 (de) | S-(-)-1-(tert-butylamino)-3-((4-morpholino-1,2, - thiadiazol-3-yl)-oxy)-2-propanol-pamoat zur topischen verwendung bei der behandlung erhoehten intraokularen drucks. | |
| FI803179A7 (fi) | Menetelmä metallurgisen kuonan komponenttien granulometristen ominaisuuksien säätelemiseksi. | |
| JPS5227768A (en) | Preparation of 5-(beta-methylmercaptoethyl) -hydantoin | |
| PH13463A (en) | N,n-dimethylacetamide adduct of 7-(d(-)-alpha-(4-ethyl-2,3-dioxo-1-piperazine carboxamido)-(4-hydroxyphenyl)acetamido)-3-(5-(1-methy-1,2,3,4-tetrazolyl)-thiomethyl)-delta-cephem-4-carboxylic acid | |
| ES502882A0 (es) | Procedimiento de obtencion de 5-(2,4-difluorofenil)salicila-to de lisina | |
| IT8025307A0 (it) | Procedimento migliorato per la purificazione dell'acido 7-amino-3-(5-metil-1,3,4-tiadiazoli l)-3-cefem-4-carbossilico. | |
| IT8021939V0 (it) | Pinza universale per l'afferramento di teglie o simili. | |
| ES523236A0 (es) | "procedimiento para la preparacion de 2-(((5-(dimetilamino) metil-2-furanil) metil) tio) etanoamina". | |
| NO874992D0 (no) | Analogifremgangsmaate til fremstilling av 4(3h)pyrimidoner med formelen.(t) | |
| FI852810A0 (fi) | Foerfarande foer framstaellning av en n,n-dimetylacetamidaddukt av 7-/d(-)- -(4-etyl-2,3-dioxo-1 -piperazinkarboxi-amido)- -(4-hydroxifenyl)acetamido/-3-/5-(1-metyl -1,2,3,4-tetrazolyl)-tiometyl/- 3-kefem-4-karboxylsyra. | |
| IT8119398A0 (it) | Procedimento per la preparazione dell'acido 7-aperta par. quadrata d-(-)-alfa-(4-etil-2 3-diosso-1piperazino-carbonilammino)-4-idrossifenilacetammido chiusa par.quadrata -3aperta par. quadrata 5-(1-metil-1,2,3,4,-tetrazolil)tiometilchiusa par. quadrata -delta 3-cefem-4-carbossilico. | |
| ES511038A0 (es) | "procedimiento para la preparacion de 5-(1-hidroxi-2-(1-metil-3-fenilpropil-amino)etil) salicilamida". | |
| JPS5248693A (en) | Synthesis of noncyclic c-nucleosides |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition | ||
| 8339 | Ceased/non-payment of the annual fee |