DE3362266D1 - Penicillanic acid dioxide prodrug - Google Patents

Penicillanic acid dioxide prodrug

Info

Publication number
DE3362266D1
DE3362266D1 DE8383302891T DE3362266T DE3362266D1 DE 3362266 D1 DE3362266 D1 DE 3362266D1 DE 8383302891 T DE8383302891 T DE 8383302891T DE 3362266 T DE3362266 T DE 3362266T DE 3362266 D1 DE3362266 D1 DE 3362266D1
Authority
DE
Germany
Prior art keywords
prodrug
penicillanic acid
acid dioxide
dioxide
penicillanic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8383302891T
Other languages
German (de)
English (en)
Inventor
Robert Fischer Myers
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Application granted granted Critical
Publication of DE3362266D1 publication Critical patent/DE3362266D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE8383302891T 1982-05-24 1983-05-20 Penicillanic acid dioxide prodrug Expired DE3362266D1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/381,104 US4428935A (en) 1982-05-24 1982-05-24 Penicillanic acid dioxide prodrug

Publications (1)

Publication Number Publication Date
DE3362266D1 true DE3362266D1 (de) 1986-04-03

Family

ID=23503664

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8383302891T Expired DE3362266D1 (de) 1982-05-24 1983-05-20 Penicillanic acid dioxide prodrug

Country Status (7)

Country Link
US (1) US4428935A (cg-RX-API-DMAC7.html)
EP (1) EP0095341B1 (cg-RX-API-DMAC7.html)
JP (1) JPS58216191A (cg-RX-API-DMAC7.html)
DE (1) DE3362266D1 (cg-RX-API-DMAC7.html)
DK (1) DK226983A (cg-RX-API-DMAC7.html)
GR (1) GR79260B (cg-RX-API-DMAC7.html)
IE (1) IE55577B1 (cg-RX-API-DMAC7.html)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4681943A (en) * 1984-11-30 1987-07-21 The Dow Chemical Company 1-acyl-1-(2-pyridinyl)semicarbazides
US4946959A (en) * 1984-11-30 1990-08-07 The Dow Chemical Company Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols
CA2078217C (en) * 1990-04-13 2000-02-22 Dennis M. Godek Process for sultamicillin intermediate
US7189351B2 (en) * 2001-10-25 2007-03-13 Spherix Incorporated D-tagatose as an anti-biofilm agent
PA8579701A1 (es) * 2002-08-23 2005-05-24 Pfizer Prod Inc Profarmaco inhibidor de beta-lactamasa
JP2006526612A (ja) * 2003-06-05 2006-11-24 ファイザー・プロダクツ・インク ベータ−ラクタマーゼ阻害剤・プロドラッグ
WO2005105073A1 (en) * 2004-04-27 2005-11-10 Medicinova, Inc. Phenoxyalkycarboxylic acid derivatives in the treatment of inflammatory diseases
ES2547258T3 (es) 2006-12-10 2015-10-02 Chongxi Yu Sistemas de administración transdérmica de antibióticos beta-lactama
RU2586287C2 (ru) * 2009-06-10 2016-06-10 Текфилдз Байокем Ко., Лтд. Композиции или пролекарства противомикробных и родственных противомикробным соединений, обладающие высокой проникающей способностью
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
ES2885698T3 (es) 2009-06-25 2021-12-15 Alkermes Pharma Ireland Ltd Profármacos de compuestos nh-ácidos
PL2445502T5 (pl) 2009-06-25 2023-03-13 Alkermes Pharma Ireland Limited Związki heterocykliczne do leczenia zaburzeń neurologicznych i psychologicznych
US8592427B2 (en) 2010-06-24 2013-11-26 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
PT2685979T (pt) 2011-03-18 2016-12-02 Alkermes Pharma Ireland Ltd Composições farmacêuticas injetáveis compreendendo um antipsicótico solúvel em água, laurato de sorbitano e polissorbato 20
PL2736510T3 (pl) * 2011-07-28 2017-07-31 Kempharm, Inc. Proleki metylofenidatu, procesy ich wytwarzania i stosowania
NZ722096A (en) 2011-12-15 2016-11-25 Alkermes Pharma Ireland Ltd Prodrugs of secondary amine compounds
CA2867121C (en) 2012-03-19 2021-05-25 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
JP6219918B2 (ja) 2012-03-19 2017-10-25 アルカームス ファーマ アイルランド リミテッド グリセロールエステルを含む医薬組成物
AU2013235526B2 (en) 2012-03-19 2017-11-30 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising benzyl alcohol
US9193685B2 (en) 2012-09-19 2015-11-24 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
EP2903614B1 (en) * 2012-10-05 2021-09-29 Sphaera Pharma Pte. Ltd Novel compounds, their synthesis and their uses
WO2015143145A1 (en) 2014-03-20 2015-09-24 Alkermes Pharma Ireland Limited Aripiprazole formulations having increased injection speeds
EP3761983A1 (en) 2018-03-05 2021-01-13 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
JP7406566B2 (ja) * 2019-04-17 2023-12-27 イクシェル ファーマ エルエルシー フマル酸モノメチルのプロドラッグ

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1255034A (en) * 1968-09-06 1971-11-24 Beecham Group Ltd Penicillin esters
NL7401782A (cg-RX-API-DMAC7.html) * 1973-02-14 1974-08-16
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド
US4234579A (en) 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4244951A (en) 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4376767A (en) * 1981-01-02 1983-03-15 Merck & Co., Inc. Pyridylmethyl esters of selected bio-affecting carboxylic acids
US4323499A (en) 1981-01-05 1982-04-06 Pfizer Inc. 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids

Also Published As

Publication number Publication date
JPS58216191A (ja) 1983-12-15
EP0095341A1 (en) 1983-11-30
IE831203L (en) 1983-11-24
DK226983D0 (da) 1983-05-20
US4428935A (en) 1984-01-31
IE55577B1 (en) 1990-11-07
GR79260B (cg-RX-API-DMAC7.html) 1984-10-22
DK226983A (da) 1983-11-25
EP0095341B1 (en) 1986-02-26

Similar Documents

Publication Publication Date Title
DE3362266D1 (de) Penicillanic acid dioxide prodrug
DE3368052D1 (de) 4-chloro-2-phenylimidazole-5-acetic acid derivatives
NO1998011I1 (no) Tiludronsyre
FI810352L (fi) Beta-lactam-antibioter
FR2538262B1 (fr) Voiture-jouet radioguidee
FI834503A0 (fi) Anordning att anvaendas vid automatisk och kontinuerlig framstaellning av fyllda hoeljesprodukter
FI831190A7 (fi) Fenoksialkyylikarboksyylihappojohdan- naisia.
AT388055B (de) Zielfernrohr
DK272083D0 (da) Oxazoleddikesyrederivater
FI833529L (fi) Foeremaol avsett att anvaendas vid automatisk och kontinuerlig framstaellning av fyllda hoeljesprodukter
DK504883D0 (da) Benzoesyrederivater
DK572581A (da) Cephalosporinderivater
DE3360053D1 (de) 3-benzoyl-2-mercaptopropionic acid derivatives
DK617084D0 (da) Prostatriensyrederivater
FI832635L (fi) Foerfarande foer framstaellning av anhydrid av n-formyl-l-aspartinsyra
DK575181A (da) Fluormethylthioeddikesyrefrbindelser
DK155731C (da) 3-brom-4-fluor-benzoesyreamid
PT77664A (pt) Cephalosporin esteres
FI841769A7 (fi) Foerfarande foer regenerering av blandningar innehaollande svavelsyra och metallsulfater till svavelsyra och metalloxider.
FI832385L (fi) Kefalosporin-antibiotika
DE3467164D1 (de) Pyrrole-2-acetylamino acid derivatives
DK553983A (da) Carbaminsyreestere
DK315383D0 (da) Carbaminsyreestere
FR2536911B1 (fr) Photodetecteur
AT364218B (de) Phosphorsaeurebeize

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8328 Change in the person/name/address of the agent

Free format text: LEDERER, F., DIPL.-CHEM. DR., PAT.-ANW., 8000 MUENCHEN

8339 Ceased/non-payment of the annual fee