DE3269422D1 - Pharmaceutical amides, and preparation, formulations and use thereof - Google Patents

Pharmaceutical amides, and preparation, formulations and use thereof

Info

Publication number
DE3269422D1
DE3269422D1 DE8282108860T DE3269422T DE3269422D1 DE 3269422 D1 DE3269422 D1 DE 3269422D1 DE 8282108860 T DE8282108860 T DE 8282108860T DE 3269422 T DE3269422 T DE 3269422T DE 3269422 D1 DE3269422 D1 DE 3269422D1
Authority
DE
Germany
Prior art keywords
sup
sub
alkyl
carbon atoms
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8282108860T
Other languages
English (en)
Inventor
Samuel Wilkinson
George William Hardy
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wellcome Foundation Ltd
Original Assignee
Wellcome Foundation Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Foundation Ltd filed Critical Wellcome Foundation Ltd
Application granted granted Critical
Publication of DE3269422D1 publication Critical patent/DE3269422D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Glass Compositions (AREA)
  • Manufacturing Cores, Coils, And Magnets (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
DE8282108860T 1981-09-25 1982-09-24 Pharmaceutical amides, and preparation, formulations and use thereof Expired DE3269422D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8129053 1981-09-25

Publications (1)

Publication Number Publication Date
DE3269422D1 true DE3269422D1 (en) 1986-04-03

Family

ID=10524742

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8282108860T Expired DE3269422D1 (en) 1981-09-25 1982-09-24 Pharmaceutical amides, and preparation, formulations and use thereof

Country Status (10)

Country Link
US (1) US4504492A (de)
EP (1) EP0075896B1 (de)
JP (1) JPS5877852A (de)
AT (1) ATE18201T1 (de)
AU (1) AU8866882A (de)
DE (1) DE3269422D1 (de)
DK (1) DK425382A (de)
GB (1) GB2108118B (de)
NZ (1) NZ201998A (de)
ZA (1) ZA827000B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0225292A3 (de) * 1985-12-06 1988-11-30 Ciba-Geigy Ag Einige N-substituierte Buttersäureamidderivate
US5166212A (en) * 1985-12-06 1992-11-24 Ciba-Geigy Corporation Certain n-substituted butyramide derivatives
DK77487A (da) * 1986-03-11 1987-09-12 Hoffmann La Roche Hydroxylaminderivater
FR2609289B1 (fr) * 1987-01-06 1991-03-29 Bellon Labor Sa Roger Nouveaux composes a activite d'inhibiteurs de collagenase, procede pour les preparer et compositions pharmaceutiques contenant ces composes
CA1337400C (en) * 1987-06-08 1995-10-24 Norma G. Delaney Inhibitors of neutral endopeptidase
US4931430A (en) * 1987-12-14 1990-06-05 E. R. Squibb & Sons, Inc. Method for preventing or treating anxiety employing an ACE inhibitor
US5599951A (en) * 1989-09-15 1997-02-04 Societe Civile Bioprojet Amino acid derivatives, the process for their preparation and their applications to therapy
FR2652087B1 (fr) * 1989-09-15 1993-10-15 Bioprojet Ste Civile Derives d'amino-acides, leur procede de preparation et leurs applications therapeutiques.
US5098889A (en) * 1990-09-17 1992-03-24 E. R. Squibb & Sons, Inc. Method for preventing or inhibiting loss of cognitive function employing a combination of an ace inhibitor and a drug that acts at serotonin receptors
US5756825A (en) * 1992-09-08 1998-05-26 Safavy; Ahmad Hydroxamic acid-based bifunctional chelating compounds
CA2358578A1 (en) * 1999-01-02 2000-07-13 Aventis Pharma Deutschland Gmbh Novel malonic acid derivatives, processes for their preparation, their use and pharmaceutical compositions containing them (inhibition of factor xa activity)
EP1127884A1 (de) 2000-02-26 2001-08-29 Aventis Pharma Deutschland GmbH Neue Malonsäure Derivaie, Verfahren zu ihrer Herstellung, ihre Verwendung als Inhibitor der Faktor XA Aktivtät und pharmazeutische Zusammensetzungen diese enthaltend
CA2580694A1 (en) * 2004-09-23 2006-03-30 Alexander Michalow Methods for regulating neurotransmitter systems by inducing counteradaptations
US20080045610A1 (en) * 2004-09-23 2008-02-21 Alexander Michalow Methods for regulating neurotransmitter systems by inducing counteradaptations
JP6599094B2 (ja) 2014-11-13 2019-10-30 株式会社ミツトヨ 光学装置

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4105789A (en) * 1976-05-10 1978-08-08 E. R. Squibb & Sons, Inc. Carboxyalkylacylamino acids
US4228184A (en) * 1976-05-10 1980-10-14 E. R. Squibb & Sons, Inc. Carboxyalkylacylamino acids
GB2074571B (en) * 1980-04-11 1984-02-15 Wellcome Found Alpha-benzyl-substituted amides
FR2480747A1 (fr) * 1980-04-17 1981-10-23 Roques Bernard Derives d'acides amines et leur application therapeutique
DE3042482A1 (de) * 1980-11-11 1982-06-24 A. Nattermann & Cie GmbH, 5000 Köln N-benzoyl- (omega) -anilinoalkancarbonsaeuren, -salze und -ester, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
EP0075334A3 (de) * 1981-09-25 1984-03-21 The Wellcome Foundation Limited Pharmazeutisch wirksame Verbindungen und ihre Herstellung, Formulierungen und deren Verwendung
FR2518088B1 (fr) * 1981-12-16 1987-11-27 Roques Bernard Nouveaux derives d'aminoacides, et leur application therapeutique

Also Published As

Publication number Publication date
EP0075896A2 (de) 1983-04-06
GB2108118B (en) 1985-09-11
NZ201998A (en) 1985-11-08
ZA827000B (en) 1984-05-30
DK425382A (da) 1983-03-26
ATE18201T1 (de) 1986-03-15
EP0075896B1 (de) 1986-02-26
US4504492A (en) 1985-03-12
EP0075896A3 (en) 1983-07-20
JPS5877852A (ja) 1983-05-11
GB2108118A (en) 1983-05-11
AU8866882A (en) 1983-03-31

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Legal Events

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8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee